CN104109128B - 卡博替尼苹果酸盐及其制备方法 - Google Patents
卡博替尼苹果酸盐及其制备方法 Download PDFInfo
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- CN104109128B CN104109128B CN201310164410.5A CN201310164410A CN104109128B CN 104109128 B CN104109128 B CN 104109128B CN 201310164410 A CN201310164410 A CN 201310164410A CN 104109128 B CN104109128 B CN 104109128B
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
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CN201310164410.5A CN104109128B (zh) | 2013-04-19 | 2013-04-19 | 卡博替尼苹果酸盐及其制备方法 |
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CN104109128A CN104109128A (zh) | 2014-10-22 |
CN104109128B true CN104109128B (zh) | 2016-10-05 |
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Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
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US11814356B1 (en) | 2023-03-29 | 2023-11-14 | Apotex Inc. | Salt of cabozantinib |
Families Citing this family (1)
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CN108341773A (zh) * | 2017-01-21 | 2018-07-31 | 南京华威医药科技开发有限公司 | 卡博替尼苹果酸盐的晶型ii |
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EP2210607B1 (en) * | 2003-09-26 | 2011-08-17 | Exelixis Inc. | N-[3-fluoro-4-({6-(methyloxy)-7-[(3-morpholin-4-ylpropyl)oxy]quinolin-4-yl}oxy)phenyl]-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide for the treatment of cancer |
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Cited By (1)
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US11814356B1 (en) | 2023-03-29 | 2023-11-14 | Apotex Inc. | Salt of cabozantinib |
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Effective date of registration: 20221205 Address after: 102199 Floor 2, Building 1, Yard 2, Kechuang 8th Street, Beijing Economic and Technological Development Zone, Daxing District, Beijing (Yizhuang Cluster, High end Industrial Zone, Beijing Pilot Free Trade Zone) Patentee after: Beijing Zhengda Innovation Medicine Co.,Ltd. Address before: 222069 No. 16 Jinqiao Road, Dapu Industrial Zone, Lianyungang Economic and Technological Development Zone, Lianyungang City, Jiangsu Province Patentee before: LIANYUNGANG RUNZHONG PHARMACEUTICAL Co.,Ltd. |