CN1035112C - 用于生产二嗪基哌啶衍生物的改进方法 - Google Patents

用于生产二嗪基哌啶衍生物的改进方法 Download PDF

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Publication number
CN1035112C
CN1035112C CN90108728A CN90108728A CN1035112C CN 1035112 C CN1035112 C CN 1035112C CN 90108728 A CN90108728 A CN 90108728A CN 90108728 A CN90108728 A CN 90108728A CN 1035112 C CN1035112 C CN 1035112C
Authority
CN
China
Prior art keywords
diazine
described method
pyrrolidone
formula
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
CN90108728A
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English (en)
Chinese (zh)
Other versions
CN1051357A (zh
Inventor
加里·D·马丁
约瑟夫·L·米尼利
罗纳德·J·马特森
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Co
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of CN1051357A publication Critical patent/CN1051357A/zh
Application granted granted Critical
Publication of CN1035112C publication Critical patent/CN1035112C/zh
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CN90108728A 1989-10-27 1990-10-25 用于生产二嗪基哌啶衍生物的改进方法 Expired - Lifetime CN1035112C (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US42838289A 1989-10-27 1989-10-27
US428,382 1989-10-27
US58558990A 1990-09-20 1990-09-20
US585589 1990-09-20
US585,589 1990-09-20

Publications (2)

Publication Number Publication Date
CN1051357A CN1051357A (zh) 1991-05-15
CN1035112C true CN1035112C (zh) 1997-06-11

Family

ID=27027734

Family Applications (1)

Application Number Title Priority Date Filing Date
CN90108728A Expired - Lifetime CN1035112C (zh) 1989-10-27 1990-10-25 用于生产二嗪基哌啶衍生物的改进方法

Country Status (9)

Country Link
KR (1) KR910007913A (no)
CN (1) CN1035112C (no)
AT (1) AT398972B (no)
ES (1) ES2026060A6 (no)
FI (1) FI95468C (no)
GR (1) GR1001134B (no)
NO (1) NO176715C (no)
PT (1) PT95712B (no)
YU (1) YU203390A (no)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100432283B1 (ko) * 2001-10-27 2004-05-22 한국과학기술연구원 무스카린성 아세틸콜린 수용체에 작용하는테트라하이드로피리딘 유도체
KR20200047989A (ko) 2018-10-29 2020-05-08 이수완 튜닝이 용이한 바이올린

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4826843A (en) * 1985-07-08 1989-05-02 Bristol-Myers Cerebral function enhancing diazinylpiperidine derivatives

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU206878B (en) * 1989-10-27 1993-01-28 Bristol Myers Squibb Co Process for producing 1-//1-/2-/trifluoromethyl/-4-pyrimidinyl/-4-piperidinyl/-methyl/-2-pirrolidinone

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4826843A (en) * 1985-07-08 1989-05-02 Bristol-Myers Cerebral function enhancing diazinylpiperidine derivatives

Also Published As

Publication number Publication date
FI905226A0 (fi) 1990-10-24
FI95468B (fi) 1995-10-31
PT95712B (pt) 1998-01-30
PT95712A (pt) 1991-09-13
YU203390A (sh) 1993-10-20
AT398972B (de) 1995-02-27
NO904588L (no) 1991-04-29
ATA214890A (de) 1994-07-15
NO176715C (no) 1995-05-16
CN1051357A (zh) 1991-05-15
NO904588D0 (no) 1990-10-24
NO176715B (no) 1995-02-06
GR1001134B (el) 1993-04-28
GR900100777A (en) 1992-03-20
ES2026060A6 (es) 1992-04-01
KR910007913A (ko) 1991-05-30
FI95468C (fi) 1996-02-12

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Legal Events

Date Code Title Description
C06 Publication
PB01 Publication
C10 Entry into substantive examination
SE01 Entry into force of request for substantive examination
C14 Grant of patent or utility model
GR01 Patent grant
C15 Extension of patent right duration from 15 to 20 years for appl. with date before 31.12.1992 and still valid on 11.12.2001 (patent law change 1993)
OR01 Other related matters
C17 Cessation of patent right
CX01 Expiry of patent term

Expiration termination date: 20101025

Granted publication date: 19970611