CN103509008A - 吡唑取代的氨基-杂芳基化合物的衍生物 - Google Patents
吡唑取代的氨基-杂芳基化合物的衍生物 Download PDFInfo
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- CN103509008A CN103509008A CN201210326710.4A CN201210326710A CN103509008A CN 103509008 A CN103509008 A CN 103509008A CN 201210326710 A CN201210326710 A CN 201210326710A CN 103509008 A CN103509008 A CN 103509008A
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Images
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US201261663221P | 2012-06-22 | 2012-06-22 | |
| US61/663,221 | 2012-06-22 | ||
| US201261680885P | 2012-08-08 | 2012-08-08 | |
| US61/680,885 | 2012-08-08 |
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| CN103509008A true CN103509008A (zh) | 2014-01-15 |
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| CN (1) | CN103509008A (https=) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
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| CN103304552A (zh) * | 2012-03-09 | 2013-09-18 | 广东东阳光药业有限公司 | 取代的吡啶化合物及其使用方法和用途 |
| CN104650049A (zh) * | 2013-08-28 | 2015-05-27 | 广东东阳光药业有限公司 | 取代的吡啶化合物及其使用方法和用途 |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3381925B1 (en) * | 2015-11-27 | 2020-12-16 | Chia Tai Tianqing Pharmaceutical Group Co., Ltd. | Deuterium-modified brigatinib derivatives, pharmaceutical compositions comprising same, and use thereof |
| EP3415518B1 (en) | 2016-03-03 | 2020-07-08 | Shenzhen TargetRx, Inc. | Macrocycle and composition comprising thereof |
| CN114437058A (zh) * | 2020-10-30 | 2022-05-06 | 珠海宇繁生物科技有限责任公司 | 氘代hpk1激酶抑制剂及其制备方法和应用 |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101023064A (zh) * | 2004-08-26 | 2007-08-22 | 辉瑞大药厂 | 作为蛋白激酶抑制剂的对映异构体纯的氨基杂芳基化合物 |
| CN101967140A (zh) * | 2010-09-14 | 2011-02-09 | 郑州泰基鸿诺药物科技有限公司 | 氘代克里唑蒂尼及其衍生物、制备方法和应用 |
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| DE602006018354D1 (de) * | 2005-12-05 | 2010-12-30 | Pfizer Prod Inc | Verfahren zur behandlung von abnormalem zellwachstum |
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- 2012-09-06 JP JP2012195912A patent/JP2014005265A/ja active Pending
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101023064A (zh) * | 2004-08-26 | 2007-08-22 | 辉瑞大药厂 | 作为蛋白激酶抑制剂的对映异构体纯的氨基杂芳基化合物 |
| CN101967140A (zh) * | 2010-09-14 | 2011-02-09 | 郑州泰基鸿诺药物科技有限公司 | 氘代克里唑蒂尼及其衍生物、制备方法和应用 |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103304552A (zh) * | 2012-03-09 | 2013-09-18 | 广东东阳光药业有限公司 | 取代的吡啶化合物及其使用方法和用途 |
| CN103304552B (zh) * | 2012-03-09 | 2016-12-28 | 广东东阳光药业有限公司 | 取代的吡啶化合物及其使用方法和用途 |
| CN104650049A (zh) * | 2013-08-28 | 2015-05-27 | 广东东阳光药业有限公司 | 取代的吡啶化合物及其使用方法和用途 |
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| JP2014005265A (ja) | 2014-01-16 |
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