CN102753513B - 制备芳基和杂芳基乙酸衍生物的方法 - Google Patents
制备芳基和杂芳基乙酸衍生物的方法 Download PDFInfo
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- CN102753513B CN102753513B CN201180009550.4A CN201180009550A CN102753513B CN 102753513 B CN102753513 B CN 102753513B CN 201180009550 A CN201180009550 A CN 201180009550A CN 102753513 B CN102753513 B CN 102753513B
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- China
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- hydrogen
- alkyl
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
- C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
- C07C67/333—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton
- C07C67/343—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
- C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
- C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/612—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US29608110P | 2010-01-19 | 2010-01-19 | |
| EP10151081.6 | 2010-01-19 | ||
| US61/296,081 | 2010-01-19 | ||
| EP10151081 | 2010-01-19 | ||
| PCT/EP2011/050456 WO2011089072A1 (de) | 2010-01-19 | 2011-01-14 | Verfahren zur herstellung von aryl- und heteroarylessigsäure-derivaten |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN102753513A CN102753513A (zh) | 2012-10-24 |
| CN102753513B true CN102753513B (zh) | 2015-03-18 |
Family
ID=42245969
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN201180009550.4A Active CN102753513B (zh) | 2010-01-19 | 2011-01-14 | 制备芳基和杂芳基乙酸衍生物的方法 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US8507688B2 (https=) |
| EP (1) | EP2526081B1 (https=) |
| JP (1) | JP5899119B2 (https=) |
| KR (1) | KR101773070B1 (https=) |
| CN (1) | CN102753513B (https=) |
| DK (1) | DK2526081T3 (https=) |
| ES (1) | ES2546487T3 (https=) |
| IL (1) | IL220787A (https=) |
| IN (1) | IN2012DN06383A (https=) |
| WO (1) | WO2011089072A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR112013022282B1 (pt) * | 2011-03-02 | 2019-03-26 | Bayer Intellectual Property Gmbh | Processo para a preparação de derivados de ácidos aril- e heteroaril acético |
| JP7353295B2 (ja) | 2018-04-10 | 2023-09-29 | バイエル・アクチエンゲゼルシヤフト | ２，６－ジアルキルフェニル酢酸の製造方法 |
| CN113121341A (zh) * | 2019-12-31 | 2021-07-16 | 江苏中旗科技股份有限公司 | 一种合成2,6-二乙基-4-甲基苯乙酸酯的方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2736053B1 (fr) * | 1995-06-28 | 1997-09-19 | Sanofi Sa | Nouvelles 1-phenylalkyl-1,2,3,6-tetrahydropyridines |
| CN1152860C (zh) | 1995-06-30 | 2004-06-09 | 拜尔公司 | 二烷基-卤代苯基取代的酮-烯醇 |
| AU4614100A (en) * | 1999-05-17 | 2000-12-05 | Teijin Limited | Cyanobiphenyl derivatives |
| DE10111262A1 (de) | 2001-03-09 | 2002-09-12 | Studiengesellschaft Kohle Mbh | Verfahren zur Herstellung von Vinyl- Aryl- und Heteroarylessigsäuren und ihrer Devivate |
| WO2003009936A2 (en) * | 2001-07-23 | 2003-02-06 | Andrew Bruce Holmes | Palladium-catalysed carbon-carbon bond forming reactions in compressed carbon dioxide |
-
2011
- 2011-01-14 CN CN201180009550.4A patent/CN102753513B/zh active Active
- 2011-01-14 EP EP11700418.4A patent/EP2526081B1/de active Active
- 2011-01-14 ES ES11700418.4T patent/ES2546487T3/es active Active
- 2011-01-14 KR KR1020127021635A patent/KR101773070B1/ko active Active
- 2011-01-14 DK DK11700418.4T patent/DK2526081T3/en active
- 2011-01-14 WO PCT/EP2011/050456 patent/WO2011089072A1/de not_active Ceased
- 2011-01-14 JP JP2012548446A patent/JP5899119B2/ja active Active
- 2011-01-14 IN IN6383DEN2012 patent/IN2012DN06383A/en unknown
- 2011-01-19 US US13/009,453 patent/US8507688B2/en active Active
-
2012
- 2012-07-05 IL IL220787A patent/IL220787A/en active IP Right Grant
Non-Patent Citations (2)
| Title |
|---|
| E. Paetzold,et al..Efficient two-phase Suzuki reaction catalyzed by palladium complexes with water-soluble phosphine ligands and detergents as phase transfer reagents.《Journal of Molecular Catalysis A: Chemical》.2000,第152卷69-76. * |
| Pd-catalyzed synthesis of arylacetic acid derivatives from boronic acids;Lukas J. Gooßen;《Chemical Communication》;20010321;669–670 * |
Also Published As
| Publication number | Publication date |
|---|---|
| JP5899119B2 (ja) | 2016-04-06 |
| WO2011089072A1 (de) | 2011-07-28 |
| EP2526081B1 (de) | 2015-07-01 |
| KR20120116491A (ko) | 2012-10-22 |
| US20110184180A1 (en) | 2011-07-28 |
| EP2526081A1 (de) | 2012-11-28 |
| JP2013517255A (ja) | 2013-05-16 |
| DK2526081T3 (en) | 2015-10-05 |
| CN102753513A (zh) | 2012-10-24 |
| US8507688B2 (en) | 2013-08-13 |
| ES2546487T3 (es) | 2015-09-24 |
| IL220787A (en) | 2015-05-31 |
| IN2012DN06383A (https=) | 2015-10-02 |
| KR101773070B1 (ko) | 2017-09-12 |
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Legal Events
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| C06 | Publication | ||
| PB01 | Publication | ||
| C10 | Entry into substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| C14 | Grant of patent or utility model | ||
| GR01 | Patent grant | ||
| TR01 | Transfer of patent right | ||
| TR01 | Transfer of patent right |
Effective date of registration: 20240115 Address after: 50 Alfred Nobel Street, Monheim, Rhine, Germany 40789 Patentee after: BAYER CROPSCIENCE AG Address before: Germany Patentee before: BAYER INTELLECTUAL PROPERTY GmbH |