CN102319433A - 包含嘧啶的nnrti和rt抑制剂的组合 - Google Patents
包含嘧啶的nnrti和rt抑制剂的组合 Download PDFInfo
- Publication number
- CN102319433A CN102319433A CN2011102800883A CN201110280088A CN102319433A CN 102319433 A CN102319433 A CN 102319433A CN 2011102800883 A CN2011102800883 A CN 2011102800883A CN 201110280088 A CN201110280088 A CN 201110280088A CN 102319433 A CN102319433 A CN 102319433A
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- CN
- China
- Prior art keywords
- amino
- combination
- pharmaceutically acceptable
- nrti
- acceptable salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (12)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US49977103P | 2003-09-03 | 2003-09-03 | |
| EP03103275.8 | 2003-09-03 | ||
| EP03103275 | 2003-09-03 | ||
| US60/499771 | 2003-09-03 | ||
| EP03103319 | 2003-09-08 | ||
| EP03103319.4 | 2003-09-08 | ||
| EP03103335 | 2003-09-10 | ||
| EP03103335.0 | 2003-09-10 | ||
| EP03103668 | 2003-10-02 | ||
| EP03103668.4 | 2003-10-02 | ||
| US50848603P | 2003-10-03 | 2003-10-03 | |
| US60/508486 | 2003-10-03 |
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| CN2004800254267A Division CN101060844B (zh) | 2003-09-03 | 2004-09-03 | 包含嘧啶的nnrti和rt抑制剂的组合 |
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| KR (2) | KR101638999B1 (es) |
| CN (1) | CN102319433A (es) |
| DK (1) | DK1663240T4 (es) |
| EA (1) | EA014840B1 (es) |
| ES (1) | ES2542017T5 (es) |
| HU (1) | HUE025576T2 (es) |
| PT (1) | PT1663240E (es) |
| SI (1) | SI1663240T2 (es) |
| TW (1) | TWI365744B (es) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003016306A1 (en) * | 2001-08-13 | 2003-02-27 | Janssen Pharmaceutica N.V. | Hiv inhibiting pyrimidines derivatives |
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2004
- 2004-09-02 TW TW093126446A patent/TWI365744B/zh active
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- 2004-09-03 CN CN2011102800883A patent/CN102319433A/zh active Pending
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- 2004-09-03 KR KR1020137024817A patent/KR101638999B1/ko active IP Right Grant
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- 2004-09-03 DK DK04787096.9T patent/DK1663240T4/da active
- 2004-09-03 KR KR1020117025799A patent/KR101539245B1/ko active IP Right Grant
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003016306A1 (en) * | 2001-08-13 | 2003-02-27 | Janssen Pharmaceutica N.V. | Hiv inhibiting pyrimidines derivatives |
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| Title |
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| GILEAD SCIENCES INC: "《internet article[online]》", 11 August 2003 * |
Also Published As
| Publication number | Publication date |
|---|---|
| ES2542017T3 (es) | 2015-07-29 |
| EA200600522A1 (ru) | 2006-08-25 |
| KR20110132475A (ko) | 2011-12-07 |
| ES2542017T5 (es) | 2023-06-15 |
| DK1663240T3 (en) | 2015-07-20 |
| KR101539245B1 (ko) | 2015-07-27 |
| SI1663240T2 (sl) | 2023-05-31 |
| KR20130127515A (ko) | 2013-11-22 |
| DK1663240T4 (da) | 2023-04-17 |
| TWI365744B (en) | 2012-06-11 |
| TW200524612A (en) | 2005-08-01 |
| PT1663240E (pt) | 2015-09-01 |
| SI1663240T1 (sl) | 2015-10-30 |
| HUE025576T2 (en) | 2016-04-28 |
| EA014840B1 (ru) | 2011-02-28 |
| KR101638999B1 (ko) | 2016-07-12 |
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