CN101657099B - 用作ppar调节剂的取代的1,3-二氧杂环己烷 - Google Patents

用作ppar调节剂的取代的1,3-二氧杂环己烷 Download PDF

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CN101657099B
CN101657099B CN200880008902.2A CN200880008902A CN101657099B CN 101657099 B CN101657099 B CN 101657099B CN 200880008902 A CN200880008902 A CN 200880008902A CN 101657099 B CN101657099 B CN 101657099B
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ppar
compound
compounds
chlorophenyl
hex
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CN101657099A (zh
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A·S·索伦森
J-p·梅耶尔
P·阿尔伯特斯
M·S·普拉特哈玛
M·H·卡拉梅里
T·邦诺德
J·凯勒赫
D·皮尔森
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Evolva AG
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    • C07D319/04—1,3-Dioxanes; Hydrogenated 1,3-dioxanes
    • C07D319/06—1,3-Dioxanes; Hydrogenated 1,3-dioxanes not condensed with other rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
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CN200880008902.2A 2006-01-18 2008-01-18 用作ppar调节剂的取代的1,3-二氧杂环己烷 Active CN101657099B (zh)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US76024106P 2006-01-18 2006-01-18
WOPCT/IB2007/002542 2007-01-18
PCT/IB2007/002542 WO2007138485A2 (en) 2006-01-18 2007-01-18 Ppar modulators
IBPCT/IB2007/002542 2007-01-18
US60/989,806 2007-11-21
US60/989,808 2007-11-21
US60/989,805 2007-11-21

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CN101657099A CN101657099A (zh) 2010-02-24
CN101657099B true CN101657099B (zh) 2014-11-26

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CN200880008956A Pending CN101657100A (zh) 2006-01-18 2008-01-18 取代的1,3-二氧杂环己烷及其用途
CN200880008902.2A Active CN101657099B (zh) 2006-01-18 2008-01-18 用作ppar调节剂的取代的1,3-二氧杂环己烷
CN200880008866A Pending CN101646344A (zh) 2006-01-18 2008-01-18 取代的1,3-二氧杂环己烷及其应用

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US (2) US20110178112A1 (enExample)
EP (2) EP2363127A1 (enExample)
JP (3) JP2009523781A (enExample)
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AU (1) AU2007266714B2 (enExample)
CA (1) CA2637803A1 (enExample)
DK (1) DK1976509T3 (enExample)
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JP2010516700A (ja) 2007-01-18 2010-05-20 エヴォルヴァ エスアー 置換１，３−ジオキサンおよびそれらの使用
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
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WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
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US8933024B2 (en) 2010-06-18 2015-01-13 Sanofi Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
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TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
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RU2674987C1 (ru) * 2018-04-17 2018-12-14 Акционерное общество "Всесоюзный научный центр по безопасности биологически активных веществ" АО "ВНЦ БАВ" 2-Аминия-7-(диэтиламино)-4-(4-метоксибензо[d][1,3]диоксол-5-ил)-4Н-хромен-3-карбонитрила N-ацетиламиноэтаноат, проявляющий противоопухолевую активность
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JP2015180703A (ja) 2015-10-15
MX2008009241A (es) 2008-10-20
US20140288110A1 (en) 2014-09-25
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WO2007138485A2 (en) 2007-12-06
IN2015DN00502A (enExample) 2015-06-26
CN101657099A (zh) 2010-02-24
US20110178112A1 (en) 2011-07-21
EP1976509A2 (en) 2008-10-08
JP2013060465A (ja) 2013-04-04
EP2363127A1 (en) 2011-09-07
AU2007266714A1 (en) 2007-12-06
RU2008133416A (ru) 2010-02-27
RU2449999C2 (ru) 2012-05-10
PL1976509T3 (pl) 2015-07-31
CN101646344A (zh) 2010-02-10
DK1976509T3 (en) 2015-03-23
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JP2009523781A (ja) 2009-06-25

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