CN101438288A - 谷氨酰胺合成酶的磷酰基转移酶活性的调节 - Google Patents

谷氨酰胺合成酶的磷酰基转移酶活性的调节 Download PDF

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CN101438288A
CN101438288A CNA2006800545929A CN200680054592A CN101438288A CN 101438288 A CN101438288 A CN 101438288A CN A2006800545929 A CNA2006800545929 A CN A2006800545929A CN 200680054592 A CN200680054592 A CN 200680054592A CN 101438288 A CN101438288 A CN 101438288A
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compound
atp
adenylylation
alkyl
heteroaryl
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科林·彼得·凯尼恩
林登·凯里·奥德菲尔德
克里斯蒂安·韦南德·范德-韦斯特许仁
阿曼达·路易丝·鲁索
克里斯托弗·约翰·帕金森
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CNA2006800545929A 2006-03-15 2006-03-15 谷氨酰胺合成酶的磷酰基转移酶活性的调节 Pending CN101438288A (zh)

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PCT/IB2006/000565 WO2007105023A1 (fr) 2006-03-15 2006-03-15 Modulation de l'activite phosphoryl transferase de la glutamine synthetase

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Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103709164A (zh) * 2013-12-04 2014-04-09 浙江工业大学 一种腺嘌呤的合成方法
CN109456329A (zh) * 2018-11-19 2019-03-12 威海迪素制药有限公司 一种泛昔洛韦的制备方法
CN113967207A (zh) * 2021-11-22 2022-01-25 重庆医科大学 4-异硫脲基丁腈盐酸盐在治疗分枝杆菌感染中的应用

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CA2660758A1 (fr) 2006-08-24 2008-02-27 Astrazeneca Ab Derives de la morpholino pyrimidine utiles dans le traitement de maladies proliferatives
WO2008130669A1 (fr) * 2007-04-20 2008-10-30 The Research Foundation Of State University Of New York Benzimidazoles et compositions pharmaceutiques de ceux-ci
WO2008134553A1 (fr) * 2007-04-26 2008-11-06 Xenon Pharmaceuticals Inc. Procédés de traitement de maladies associées aux canaux sodiques au moyen de composés bicycliques
EP2176238B1 (fr) 2007-07-09 2012-04-18 AstraZeneca AB Dérivés de morpholino pyrimidine utilisés dans des maladies liées à une kinase mtor et/ou à pi3k
US8871751B2 (en) 2008-01-18 2014-10-28 The Board Of Trustees Of The University Of Illinois Compositions and methods relating to nuclear hormone and steroid hormone receptors including inhibitors of estrogen receptor alpha-mediated gene expression and inhibition of breast cancer
WO2010116302A1 (fr) * 2009-04-07 2010-10-14 University Of The Witwatersrand, Johannesburg Dérivés d'imidazo[1,2-a] pyridine-6-carboxamides, leur utilisation pour le traitement du cancer du côlon et leur procédé de fabrication
EP2440533B1 (fr) * 2009-06-12 2015-09-23 Socpra-Sciences Et Génie S.E.C. Composés se liant à un ribocommutateur guanine et leur utilisation en tant qu'antibiotiques
SA111320519B1 (ar) 2010-06-11 2014-07-02 Astrazeneca Ab مركبات بيريميدينيل للاستخدام كمثبطات atr
UA115388C2 (uk) 2013-11-21 2017-10-25 Пфайзер Інк. 2,6-заміщені пуринові похідні та їх застосування в лікуванні проліферативних захворювань
CN104974098A (zh) * 2015-06-30 2015-10-14 苏州开元民生科技股份有限公司 2,5-二氨基-4,6-二羟基嘧啶盐酸盐的合成方法
IL297543A (en) 2017-11-30 2022-12-01 Arrakis Therapeutics Inc Nucleic acid-binding photoprobes and their uses
US10702525B1 (en) * 2019-09-04 2020-07-07 United Arab Emirates University Pyrimidine derivatives as anti-diabetic agents
CN111658646B (zh) * 2020-06-28 2021-03-02 河南工业大学 2,6-双(2-苯并咪唑基)吡啶在制备耐碳青霉烯类铜绿假单胞菌感染药物中的应用

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US4076711A (en) * 1976-04-05 1978-02-28 Schering Corporation Triazolo [4,5-d]-pyrimidines
CH630380A5 (de) * 1977-08-12 1982-06-15 Lonza Ag Verfahren zur herstellung von l-methotrexat.
US4565864A (en) * 1983-06-02 1986-01-21 Riker Laboratories, Inc. Substituted imidazo[1,2-c]pyrimidines
IT1215339B (it) * 1987-01-14 1990-02-08 Co Pharma Corp Srl Procedimento per la preparazione di 9-(idrossialchil)-ipoxantine
IT1212140B (it) * 1987-05-08 1989-11-08 Sig Gla Pharmaceuticals S P A Processo per la preparazione del 2,4-diammino-6-(1-piperidinil)-piri mi-din-n-ossido.
WO2003095448A1 (fr) * 2002-05-06 2003-11-20 Bayer Pharmaceuticals Corporation Derives de pyridinyl amino pyrimidine utilises dans le traitement des troubles de l'hyperproliferation
US20060142251A1 (en) * 2002-11-15 2006-06-29 Gunther Harth Anti-microbial agents derived from methionine sulfoximine analogues

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103709164A (zh) * 2013-12-04 2014-04-09 浙江工业大学 一种腺嘌呤的合成方法
CN109456329A (zh) * 2018-11-19 2019-03-12 威海迪素制药有限公司 一种泛昔洛韦的制备方法
CN109456329B (zh) * 2018-11-19 2021-03-09 迪嘉药业集团有限公司 一种泛昔洛韦的制备方法
CN113967207A (zh) * 2021-11-22 2022-01-25 重庆医科大学 4-异硫脲基丁腈盐酸盐在治疗分枝杆菌感染中的应用

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