CN100569772C - 用作jak和其它蛋白激酶抑制剂的氮杂吲哚 - Google Patents
用作jak和其它蛋白激酶抑制剂的氮杂吲哚 Download PDFInfo
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- CN100569772C CN100569772C CNB2005800103488A CN200580010348A CN100569772C CN 100569772 C CN100569772 C CN 100569772C CN B2005800103488 A CNB2005800103488 A CN B2005800103488A CN 200580010348 A CN200580010348 A CN 200580010348A CN 100569772 C CN100569772 C CN 100569772C
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CNB2005800103488A Expired - Fee Related CN100569772C (zh) | 2004-03-30 | 2005-03-30 | 用作jak和其它蛋白激酶抑制剂的氮杂吲哚 |
Country Status (4)
Country | Link |
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CN (1) | CN100569772C (xx) |
SI (1) | SI2332940T1 (xx) |
UA (1) | UA87494C2 (xx) |
ZA (1) | ZA200607981B (xx) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
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BRPI1012159B1 (pt) * | 2009-05-22 | 2022-01-25 | Incyte Holdings Corporation | Compostos derivados de n-(hetero)aril-pirrolidina de pirazol-4-il-pirrolo[2,3-d] pirimidinas e pirrol-3-il-pirrolo[2,3-d] pirimidinas como inibidores de janus cinase, composições farmacêuticas compreendendo os referidos compostos e usos dos mesmos |
JP5769733B2 (ja) * | 2010-01-27 | 2015-08-26 | バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated | ピラゾロピリジンキナーゼ阻害剤 |
KR20130094693A (ko) * | 2010-04-30 | 2013-08-26 | 셀좀 리미티드 | Jak 저해제로서의 피라졸 화합물 |
CA2822062A1 (en) * | 2010-12-16 | 2012-06-21 | Vertex Pharmaceuticals Incorporated | Inhibitors of influenza viruses replication |
EP2651941A1 (en) * | 2010-12-16 | 2013-10-23 | Vertex Pharmaceuticals Incorporated | Inhibitors of influenza viruses replication |
RU2013132681A (ru) * | 2010-12-16 | 2015-01-27 | Вертекс Фармасьютикалз Инкорпорейтед | Ингибиторы репликации вирусов гриппа |
DE102011009961A1 (de) * | 2011-02-01 | 2012-08-02 | Merck Patent Gmbh | 7-Azaindolderivate |
EP2487159A1 (en) * | 2011-02-11 | 2012-08-15 | MSD Oss B.V. | RorgammaT inhibitors |
PT3141548T (pt) * | 2011-07-05 | 2020-07-10 | Vertex Pharma | Processos e intermediários para a produção de azaindóis |
CN109641868B (zh) * | 2016-08-30 | 2021-12-03 | 广东东阳光药业有限公司 | 流感病毒复制抑制剂及其使用方法和用途 |
CN110128421B (zh) * | 2018-02-09 | 2020-08-11 | 新发药业有限公司 | 一种5-卤代-7-氮杂吲哚的简便制备方法 |
CN108299426B (zh) * | 2018-03-20 | 2020-09-04 | 宝鸡文理学院 | 一种[1,2,4]-三唑并[4,3-a]吡啶类化合物及其合成方法 |
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2005
- 2005-03-30 UA UAA200611365A patent/UA87494C2/ru unknown
- 2005-03-30 SI SI200531659T patent/SI2332940T1/sl unknown
- 2005-03-30 ZA ZA200607981A patent/ZA200607981B/en unknown
- 2005-03-30 CN CNB2005800103488A patent/CN100569772C/zh not_active Expired - Fee Related
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CN1938303A (zh) | 2007-03-28 |
ZA200607981B (en) | 2008-06-25 |
UA87494C2 (xx) | 2009-07-27 |
SI2332940T1 (sl) | 2013-03-29 |
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