CN100569772C - 用作jak和其它蛋白激酶抑制剂的氮杂吲哚 - Google Patents

用作jak和其它蛋白激酶抑制剂的氮杂吲哚 Download PDF

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Publication number
CN100569772C
CN100569772C CNB2005800103488A CN200580010348A CN100569772C CN 100569772 C CN100569772 C CN 100569772C CN B2005800103488 A CNB2005800103488 A CN B2005800103488A CN 200580010348 A CN200580010348 A CN 200580010348A CN 100569772 C CN100569772 C CN 100569772C
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CN
China
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nhch
aliphatic group
nhr
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Expired - Fee Related
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CNB2005800103488A
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English (en)
Chinese (zh)
Other versions
CN1938303A (zh
Inventor
F·萨里图罗
L·法默
R·贝蒂尔
E·哈林顿
J·格林
J·考特
J·科姆
D·劳弗
A·阿罗诺夫
H·宾奇
D·博亚尔
J-D·查里尔
S·埃弗里特
D·弗雷斯
M·莫蒂默尔
F·皮耶拉尔
D·鲁滨逊
王坚
J·平德
王天生
A·皮尔斯
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Vertex Pharmaceuticals Inc
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Vertex Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by Vertex Pharmaceuticals Inc filed Critical Vertex Pharmaceuticals Inc
Publication of CN1938303A publication Critical patent/CN1938303A/zh
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Publication of CN100569772C publication Critical patent/CN100569772C/zh
Expired - Fee Related legal-status Critical Current
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CNB2005800103488A 2004-03-30 2005-03-30 用作jak和其它蛋白激酶抑制剂的氮杂吲哚 Expired - Fee Related CN100569772C (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US55750304P 2004-03-30 2004-03-30
US60/557,503 2004-03-30
US60/625,599 2004-11-05

Related Child Applications (3)

Application Number Title Priority Date Filing Date
CN201310486314.2A Division CN103554104A (zh) 2004-03-30 2005-03-30 用作jak和其它蛋白激酶抑制剂的氮杂吲哚
CN200910206575A Division CN101676285A (zh) 2004-03-30 2005-03-30 用作jak和其它蛋白激酶抑制剂的氮杂吲哚
CN2009102065762A Division CN101676286B (zh) 2004-03-30 2005-03-30 用作jak和其它蛋白激酶抑制剂的氮杂吲哚

Publications (2)

Publication Number Publication Date
CN1938303A CN1938303A (zh) 2007-03-28
CN100569772C true CN100569772C (zh) 2009-12-16

Family

ID=37955154

Family Applications (1)

Application Number Title Priority Date Filing Date
CNB2005800103488A Expired - Fee Related CN100569772C (zh) 2004-03-30 2005-03-30 用作jak和其它蛋白激酶抑制剂的氮杂吲哚

Country Status (4)

Country Link
CN (1) CN100569772C (xx)
SI (1) SI2332940T1 (xx)
UA (1) UA87494C2 (xx)
ZA (1) ZA200607981B (xx)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI1012159B1 (pt) * 2009-05-22 2022-01-25 Incyte Holdings Corporation Compostos derivados de n-(hetero)aril-pirrolidina de pirazol-4-il-pirrolo[2,3-d] pirimidinas e pirrol-3-il-pirrolo[2,3-d] pirimidinas como inibidores de janus cinase, composições farmacêuticas compreendendo os referidos compostos e usos dos mesmos
JP5769733B2 (ja) * 2010-01-27 2015-08-26 バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated ピラゾロピリジンキナーゼ阻害剤
EA201291038A1 (ru) * 2010-04-30 2013-05-30 Целльзом Лимитид Соединения пиразола в качестве ингибиторов jak
AU2011343642A1 (en) * 2010-12-16 2013-05-02 Vertex Pharmaceuticals Incorporated Inhibitors of influenza viruses replication
RU2013132717A (ru) * 2010-12-16 2015-01-27 Вертекс Фармасьютикалз Инкорпорейтед Ингибиторы репликации вирусов гриппа
WO2012083122A1 (en) * 2010-12-16 2012-06-21 Vertex Pharmaceutical Incorporated Inhibitors of influenza viruses replication
DE102011009961A1 (de) * 2011-02-01 2012-08-02 Merck Patent Gmbh 7-Azaindolderivate
EP2487159A1 (en) * 2011-02-11 2012-08-15 MSD Oss B.V. RorgammaT inhibitors
DK3141548T3 (da) * 2011-07-05 2020-07-06 Vertex Pharma Fremgangsmåder og mellemprodukter til fremstilling af azaindoler
US10647693B2 (en) * 2016-08-30 2020-05-12 North & South Brother Pharmacy Investment Company Limited Inhibitors of influenza virus replication, application methods and uses thereof
CN110128421B (zh) * 2018-02-09 2020-08-11 新发药业有限公司 一种5-卤代-7-氮杂吲哚的简便制备方法
CN108299426B (zh) * 2018-03-20 2020-09-04 宝鸡文理学院 一种[1,2,4]-三唑并[4,3-a]吡啶类化合物及其合成方法

Also Published As

Publication number Publication date
UA87494C2 (xx) 2009-07-27
CN1938303A (zh) 2007-03-28
SI2332940T1 (sl) 2013-03-29
ZA200607981B (en) 2008-06-25

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Publication Publication Date Title
CN101676286B (zh) 用作jak和其它蛋白激酶抑制剂的氮杂吲哚
CN100569772C (zh) 用作jak和其它蛋白激酶抑制剂的氮杂吲哚

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