SI2332940T1 - Azaindoli, uporabni kot inhibitorji jak in drugih protein-kinaz - Google Patents

Azaindoli, uporabni kot inhibitorji jak in drugih protein-kinaz

Info

Publication number
SI2332940T1
SI2332940T1 SI200531659T SI200531659T SI2332940T1 SI 2332940 T1 SI2332940 T1 SI 2332940T1 SI 200531659 T SI200531659 T SI 200531659T SI 200531659 T SI200531659 T SI 200531659T SI 2332940 T1 SI2332940 T1 SI 2332940T1
Authority
SI
Slovenia
Prior art keywords
jak
inhibitors
protein kinases
azaindoles useful
azaindoles
Prior art date
Application number
SI200531659T
Other languages
English (en)
Slovenian (sl)
Inventor
Francesco Salituro
Luc Farmer
Randy Bethiel
Edmund Harrington
Jeremy Green
John Court
Jon Come
David Lauffer
Alex Aronov
Hayley Binch
Dean Boyall
Jean-Damien Charrier
Simon Everitt
Damien Fraysse
Michael Mortimore
Francoise Pierard
Daniel Robinson
Joanne Pinder
Tiansheng Wang
Albert Pierce
Jian Wang
Original Assignee
Vertex Pharmaceuticals Incorporated
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharmaceuticals Incorporated filed Critical Vertex Pharmaceuticals Incorporated
Priority claimed from EP10182365A external-priority patent/EP2332940B1/en
Publication of SI2332940T1 publication Critical patent/SI2332940T1/sl

Links

SI200531659T 2004-03-30 2005-03-30 Azaindoli, uporabni kot inhibitorji jak in drugih protein-kinaz SI2332940T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US55750304P 2004-03-30 2004-03-30
US62559904P 2004-11-05 2004-11-05
EP10182365A EP2332940B1 (en) 2004-03-30 2005-03-30 Azaindoles useful as inhibitors of JAK and other protein kinases

Publications (1)

Publication Number Publication Date
SI2332940T1 true SI2332940T1 (sl) 2013-03-29

Family

ID=37955154

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200531659T SI2332940T1 (sl) 2004-03-30 2005-03-30 Azaindoli, uporabni kot inhibitorji jak in drugih protein-kinaz

Country Status (4)

Country Link
CN (1) CN100569772C (xx)
SI (1) SI2332940T1 (xx)
UA (1) UA87494C2 (xx)
ZA (1) ZA200607981B (xx)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA025520B1 (ru) * 2009-05-22 2017-01-30 Инсайт Холдингс Корпорейшн N-(ГЕТЕРО)АРИЛПИРРОЛИДИНОВЫЕ ПРОИЗВОДНЫЕ ПИРАЗОЛ-4-ИЛ-ПИРРОЛО[2,3-d]ПИРИМИДИНОВ И ПИРРОЛ-3-ИЛ-ПИРРОЛО[2,3-d]ПИРИМИДИНОВ В КАЧЕСТВЕ ИНГИБИТОРОВ ЯНУС-КИНАЗЫ
WO2011094273A1 (en) * 2010-01-27 2011-08-04 Vertex Pharmaceuticals Incorporated Pyrazolopyridine kinase inhibitors
KR20130094693A (ko) * 2010-04-30 2013-08-26 셀좀 리미티드 Ｊａｋ 저해제로서의 피라졸 화합물
KR20130128436A (ko) * 2010-12-16 2013-11-26 버텍스 파마슈티칼스 인코포레이티드 인플루엔자 바이러스 복제의 억제제
RU2013132683A (ru) * 2010-12-16 2015-01-27 Вертекс Фармасьютикалз Инкорпорейтед Ингибиторы репликации вирусов гриппа
CN103492381A (zh) * 2010-12-16 2014-01-01 沃泰克斯药物股份有限公司 流感病毒复制的抑制剂
DE102011009961A1 (de) * 2011-02-01 2012-08-02 Merck Patent Gmbh 7-Azaindolderivate
EP2487159A1 (en) * 2011-02-11 2012-08-15 MSD Oss B.V. RorgammaT inhibitors
ES2804528T3 (es) * 2011-07-05 2021-02-08 Vertex Pharma Procesos y productos intermedios para la producción de azaindoles
US10647693B2 (en) * 2016-08-30 2020-05-12 North & South Brother Pharmacy Investment Company Limited Inhibitors of influenza virus replication, application methods and uses thereof
CN110128421B (zh) * 2018-02-09 2020-08-11 新发药业有限公司 一种5-卤代-7-氮杂吲哚的简便制备方法
CN108299426B (zh) * 2018-03-20 2020-09-04 宝鸡文理学院 一种[1,2,4]-三唑并[4,3-a]吡啶类化合物及其合成方法

Also Published As

Publication number Publication date
CN100569772C (zh) 2009-12-16
ZA200607981B (en) 2008-06-25
CN1938303A (zh) 2007-03-28
UA87494C2 (xx) 2009-07-27

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