CN100379733C - 三唑类抗真菌药物及其制备方法 - Google Patents
三唑类抗真菌药物及其制备方法 Download PDFInfo
- Publication number
- CN100379733C CN100379733C CNB021292973A CN02129297A CN100379733C CN 100379733 C CN100379733 C CN 100379733C CN B021292973 A CNB021292973 A CN B021292973A CN 02129297 A CN02129297 A CN 02129297A CN 100379733 C CN100379733 C CN 100379733C
- Authority
- CN
- China
- Prior art keywords
- compound
- formula
- fluorine
- triazol
- alcohol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Description
化合物 | MIC(μg/mL)曲霉菌属 | 足放线菌属 |
56789 | 9.10.250.0520.519 | 268.00.94137 |
Claims (10)
Priority Applications (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CNB021292973A CN100379733C (zh) | 2002-10-08 | 2002-10-08 | 三唑类抗真菌药物及其制备方法 |
CN200710079858A CN100579977C (zh) | 2002-10-08 | 2002-10-08 | 制备三唑类抗真菌药物的方法 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CNB021292973A CN100379733C (zh) | 2002-10-08 | 2002-10-08 | 三唑类抗真菌药物及其制备方法 |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN200710079858A Division CN100579977C (zh) | 2002-10-08 | 2002-10-08 | 制备三唑类抗真菌药物的方法 |
Publications (2)
Publication Number | Publication Date |
---|---|
CN1488629A CN1488629A (zh) | 2004-04-14 |
CN100379733C true CN100379733C (zh) | 2008-04-09 |
Family
ID=34144102
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CNB021292973A Expired - Lifetime CN100379733C (zh) | 2002-10-08 | 2002-10-08 | 三唑类抗真菌药物及其制备方法 |
CN200710079858A Expired - Fee Related CN100579977C (zh) | 2002-10-08 | 2002-10-08 | 制备三唑类抗真菌药物的方法 |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN200710079858A Expired - Fee Related CN100579977C (zh) | 2002-10-08 | 2002-10-08 | 制备三唑类抗真菌药物的方法 |
Country Status (1)
Country | Link |
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CN (2) | CN100379733C (zh) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20080194820A1 (en) | 2004-12-14 | 2008-08-14 | Venkataraman Sundaram | Process For Preparing Voriconazole |
WO2007132354A2 (en) * | 2006-02-01 | 2007-11-22 | Medichem, S.A. | Process for preparing voriconazole, new polymorphic form of intermediate thereof, and uses thereof |
EP2545039A1 (en) | 2010-03-10 | 2013-01-16 | Synthon BV | A process for making voriconazole |
AR082536A1 (es) * | 2010-08-26 | 2012-12-12 | Bayer Cropscience Ag | Derivados de 5-yodo-triazol |
CN111518041A (zh) * | 2020-04-24 | 2020-08-11 | 湖南复瑞生物医药技术有限责任公司 | 一种2’4’-二氟-2-[1-(1h-1,2,4-三唑基)]苯乙酮的制备方法 |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1100421A (zh) * | 1990-02-02 | 1995-03-22 | 美国辉瑞有限公司 | 含三唑类的药用组合物的制备方法 |
-
2002
- 2002-10-08 CN CNB021292973A patent/CN100379733C/zh not_active Expired - Lifetime
- 2002-10-08 CN CN200710079858A patent/CN100579977C/zh not_active Expired - Fee Related
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1100421A (zh) * | 1990-02-02 | 1995-03-22 | 美国辉瑞有限公司 | 含三唑类的药用组合物的制备方法 |
Also Published As
Publication number | Publication date |
---|---|
CN101003532A (zh) | 2007-07-25 |
CN100579977C (zh) | 2010-01-13 |
CN1488629A (zh) | 2004-04-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
C06 | Publication | ||
PB01 | Publication | ||
C10 | Entry into substantive examination | ||
SE01 | Entry into force of request for substantive examination | ||
ASS | Succession or assignment of patent right |
Owner name: NANJING KANGZE PHARMACEUTICAL TECHNOLOGY CO., LTD Free format text: FORMER OWNER: ZHANG WENGENG Effective date: 20061124 |
|
C41 | Transfer of patent application or patent right or utility model | ||
TA01 | Transfer of patent application right |
Effective date of registration: 20061124 Address after: 210015, 5, Qiaodong street, Xiaguan District, Jiangsu, Nanjing Applicant after: Nanjing Kangze Pharmaceutical Technology Inc. Co-applicant after: Zhang Wengeng Address before: 100036, room 2, unit 10, building 503, Pu Hui north, Haidian District, Beijing Applicant before: Zhang Wengeng |
|
C57 | Notification of unclear or unknown address | ||
DD01 | Delivery of document by public notice |
Addressee: Xu Yongxiang Document name: Second notice of examination advice |
|
C14 | Grant of patent or utility model | ||
GR01 | Patent grant | ||
EE01 | Entry into force of recordation of patent licensing contract |
Assignee: SHENZHEN HAIBIN PHARMACEUTICAL Co.,Ltd. Assignor: Nanjing Kangze Pharmaceutical Technology Inc.|Zhang Wengeng Contract fulfillment period: 2008.9.26 to 2022.10.7 Contract record no.: 2008990001284 Denomination of invention: Method for preparing triazole antifungal agent Granted publication date: 20080409 License type: Exclusive license Record date: 20081126 |
|
LIC | Patent licence contract for exploitation submitted for record |
Free format text: EXCLUSIVE LICENSE; TIME LIMIT OF IMPLEMENTING CONTACT: 2008.9.26 TO 2022.10.7; CHANGE OF CONTRACT Name of requester: SHENZHEN CITY HAIBIN PHARMACEUTICAL CO., LTD. Effective date: 20081126 |
|
C56 | Change in the name or address of the patentee |
Owner name: XU YONGXIANG Free format text: FORMER NAME: KANGZU MEDICINES TECH CO., LTD., NAJING |
|
CP03 | Change of name, title or address |
Address after: Yijing garden Gulou District of Nanjing city in Jiangsu province 210005 No. 9 room 105 Patentee after: Xu Yongxiang Address before: 210015, 5, Qiaodong street, Xiaguan District, Jiangsu, Nanjing Co-patentee before: Zhang Wengeng Patentee before: Nanjing Kangze Pharmaceutical Technology Inc. |
|
CX01 | Expiry of patent term | ||
CX01 | Expiry of patent term |
Granted publication date: 20080409 |