CL2021002713A1 - Procedimiento para la preparación de derivados de oxadiazol microbiocidas. - Google Patents

Procedimiento para la preparación de derivados de oxadiazol microbiocidas.

Info

Publication number
CL2021002713A1
CL2021002713A1 CL2021002713A CL2021002713A CL2021002713A1 CL 2021002713 A1 CL2021002713 A1 CL 2021002713A1 CL 2021002713 A CL2021002713 A CL 2021002713A CL 2021002713 A CL2021002713 A CL 2021002713A CL 2021002713 A1 CL2021002713 A1 CL 2021002713A1
Authority
CL
Chile
Prior art keywords
preparation
procedure
oxadiazole derivatives
microbiocidal
microbiocidal oxadiazole
Prior art date
Application number
CL2021002713A
Other languages
English (en)
Inventor
Régis Jean Georges Mondiere
Edouard Godineau
Thomas James Hoffman
Wolfgang Stutz
Sujit Kumar Ghorai
Anup Jawalekar
Original Assignee
Syngenta Crop Protection Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Crop Protection Ag filed Critical Syngenta Crop Protection Ag
Publication of CL2021002713A1 publication Critical patent/CL2021002713A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

La presente invención se refiere a un procedimiento de acuerdo con el esquema 1 para la preparación de derivados de 5- trifluorometil-1,2,4-oxadiazol microbiocidas de fórmula (I) adecuados para su uso, por ejemplo, como principios activos, que tienen actividad microbiocida, en particular, actividad fungicida.
CL2021002713A 2019-04-18 2021-10-15 Procedimiento para la preparación de derivados de oxadiazol microbiocidas. CL2021002713A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN201911015611 2019-04-18

Publications (1)

Publication Number Publication Date
CL2021002713A1 true CL2021002713A1 (es) 2022-05-27

Family

ID=70292983

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2021002713A CL2021002713A1 (es) 2019-04-18 2021-10-15 Procedimiento para la preparación de derivados de oxadiazol microbiocidas.

Country Status (12)

Country Link
US (1) US20220194907A1 (es)
EP (1) EP3956318A1 (es)
JP (1) JP2022529006A (es)
CN (1) CN113748105B (es)
AR (1) AR118673A1 (es)
BR (1) BR112021020673A2 (es)
CL (1) CL2021002713A1 (es)
CO (1) CO2021013497A2 (es)
IL (1) IL286566A (es)
MX (1) MX2021012542A (es)
UY (1) UY38667A (es)
WO (1) WO2020212513A1 (es)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3172284A1 (en) 2020-04-28 2021-11-04 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors i
WO2021219388A1 (en) 2020-04-28 2021-11-04 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors iii
KR20230005261A (ko) 2020-04-28 2023-01-09 바스프 에스이 Qo 억제제 II 에 대한 내성을 부여하는 미토콘드리아 시토크롬 b 단백질 내에 아미노산 치환 F129L 을 함유하는 식물병원성 진균의 퇴치를 위한 스트로빌루린 유형 화합물의 용도
JP2023527660A (ja) 2020-04-28 2023-06-30 ビーエーエスエフ ソシエタス・ヨーロピア ミトコンドリアチトクロムｂタンパク質中にＱｏ阻害剤Ｉに対して耐性を付与するアミノ酸置換Ｆ１２９Ｌを含む植物病原性菌類を駆除するためのストロビルリン型化合物の使用
US20230255200A1 (en) 2020-07-08 2023-08-17 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors vi
EP3939961A1 (en) 2020-07-16 2022-01-19 Basf Se Strobilurin type compounds and their use for combating phytopathogenic fungi
US20230357152A1 (en) 2020-08-11 2023-11-09 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors viii
WO2022106304A1 (en) 2020-11-23 2022-05-27 BASF Agro B.V. Compositions comprising mefentrifluconazole
US20240016150A1 (en) 2020-12-01 2024-01-18 Basf Se Mixtures containing metarylpicoxamid
WO2022128554A1 (en) 2020-12-15 2022-06-23 Basf Se Mixtures containing n-methoxy-n-[[4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]cyclopropanecarboxamide
AR124367A1 (es) * 2020-12-17 2023-03-22 Fmc Corp Oxadiazoles fungicidas y sus mezclas
WO2022136000A1 (en) 2020-12-23 2022-06-30 Basf Se Pesticidal mixtures
EP4018830A1 (en) 2020-12-23 2022-06-29 Basf Se Pesticidal mixtures
CA3218900A1 (en) 2021-05-18 2022-11-24 Wassilios Grammenos New substituted pyridines as fungicides
CN117355518A (zh) 2021-05-18 2024-01-05 巴斯夫欧洲公司 用作杀真菌剂的新型取代吡啶类
CN117355520A (zh) 2021-05-18 2024-01-05 巴斯夫欧洲公司 用作杀真菌剂的新型取代喹啉类
MX2024000380A (es) 2021-07-08 2024-01-29 Basf Se Preparacion de amidoximas sustituidas.
IL310047A (en) * 2021-07-14 2024-03-01 Basf Se A process for producing alkyl trifluoroacetates
AU2022321882A1 (en) 2021-08-02 2024-02-15 Basf Se (3-pirydyl)-quinazoline
KR20240042626A (ko) 2021-08-02 2024-04-02 바스프 에스이 (3-퀴놀릴)-퀴나졸린
WO2023072671A1 (en) 2021-10-28 2023-05-04 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors ix
WO2023072670A1 (en) 2021-10-28 2023-05-04 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors x
EP4198023A1 (en) 2021-12-16 2023-06-21 Basf Se Pesticidally active thiosemicarbazone compounds
WO2023208447A1 (en) 2022-04-25 2023-11-02 Basf Se An emulsifiable concentrate having a (substituted) benzaldehyde-based solvent system
WO2024018016A1 (en) 2022-07-21 2024-01-25 Syngenta Crop Protection Ag Crystalline forms of 1,2,4-oxadiazole fungicides
EP4342885A1 (en) 2022-09-20 2024-03-27 Basf Se N-(3-(aminomethyl)-phenyl)-5-(4-phenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-amine derivatives and similar compounds as pesticides
EP4361126A1 (en) 2022-10-24 2024-05-01 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors xv
WO2024104813A1 (en) 2022-11-14 2024-05-23 Basf Se Fungicidal mixture comprising substituted pyridines
WO2024104818A1 (en) 2022-11-16 2024-05-23 Basf Se Substituted benzodiazepines as fungicides
WO2024104815A1 (en) 2022-11-16 2024-05-23 Basf Se Substituted benzodiazepines as fungicides
WO2024104823A1 (en) 2022-11-16 2024-05-23 Basf Se New substituted tetrahydrobenzoxazepine
WO2024104814A1 (en) 2022-11-16 2024-05-23 Basf Se Fungicidal mixture comprising substituted pyridines
WO2024104822A1 (en) 2022-11-16 2024-05-23 Basf Se Substituted tetrahydrobenzodiazepine as fungicides
EP4389210A1 (en) 2022-12-21 2024-06-26 Basf Se Heteroaryl compounds for the control of invertebrate pests

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003028729A2 (en) 2001-10-03 2003-04-10 Pharmacia Corporation Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
CA2635580A1 (en) 2005-12-30 2007-07-12 Alantos Pharmaceuticals Holding, Inc. Substituted bis-amide metalloprotease inhibitors
NZ571271A (en) * 2006-03-23 2011-10-28 Biota Europe Ltd The use of benzamide or pyridinamide derivatives as antibacterial agents
EP2186804B1 (en) 2007-08-10 2015-06-17 Nippon Soda Co., Ltd. Nitrogen-containing heterocyclic compound and pest control agent
WO2013066838A1 (en) 2011-10-31 2013-05-10 Glaxosmithkline Llc Compounds and methods
WO2013066839A2 (en) 2011-10-31 2013-05-10 Glaxosmithkline Llc Compounds and methods
WO2013132253A1 (en) 2012-03-07 2013-09-12 Institute Of Cancer Research: Royal Cancer Hospital (The) 3-aryl-5-substituted-isoquinolin-1-one compounds and their therapeutic use
WO2017055473A1 (en) 2015-10-02 2017-04-06 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
US11066396B2 (en) * 2016-06-23 2021-07-20 Merck Sharp & Dohme Corp. 3-aryl- heteroaryl substituted 5-trifluoromethyl oxadiazoles as histonedeacetylase 6 (HDAC6) inhibitors
US11974572B2 (en) * 2017-03-31 2024-05-07 Sygenta Participations Ag Fungicidal compositions
WO2018177880A1 (en) * 2017-03-31 2018-10-04 Syngenta Participations Ag Fungicidal compositions
WO2018184985A1 (en) * 2017-04-05 2018-10-11 Syngenta Participations Ag Microbiocidal oxadiazole derivatives
WO2018219773A1 (en) * 2017-06-02 2018-12-06 Syngenta Participations Ag Fungicidal compositions

Also Published As

Publication number Publication date
MX2021012542A (es) 2021-11-12
US20220194907A1 (en) 2022-06-23
BR112021020673A2 (pt) 2021-12-07
CN113748105A (zh) 2021-12-03
AR118673A1 (es) 2021-10-20
JP2022529006A (ja) 2022-06-16
IL286566A (en) 2021-10-31
UY38667A (es) 2020-11-30
WO2020212513A1 (en) 2020-10-22
CO2021013497A2 (es) 2022-01-28
CN113748105B (zh) 2024-06-11
EP3956318A1 (en) 2022-02-23

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