MX2021012542A - Proceso para la preparacion de derivados de oxadiazol microbiocidas. - Google Patents

Proceso para la preparacion de derivados de oxadiazol microbiocidas.

Info

Publication number
MX2021012542A
MX2021012542A MX2021012542A MX2021012542A MX2021012542A MX 2021012542 A MX2021012542 A MX 2021012542A MX 2021012542 A MX2021012542 A MX 2021012542A MX 2021012542 A MX2021012542 A MX 2021012542A MX 2021012542 A MX2021012542 A MX 2021012542A
Authority
MX
Mexico
Prior art keywords
preparation
oxadiazole derivatives
microbiocidal
microbiocidal oxadiazole
activity
Prior art date
Application number
MX2021012542A
Other languages
English (en)
Inventor
Edouard Godineau
Régis Jean Georges Mondiere
Thomas James Hoffman
Wolfgang Stutz
Sujit Kumar Ghorai
Anup Jawalekar
Original Assignee
Syngenta Crop Protection Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Crop Protection Ag filed Critical Syngenta Crop Protection Ag
Publication of MX2021012542A publication Critical patent/MX2021012542A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

La presente invención se refiere a un proceso de acuerdo con el esquema de reacción 1 para la preparación de derivados de 5-trifluorometil-1,2,4-oxadiazol microbiocidas de fórmula (I) adecuados para su uso, por ejemplo, como principios activos, que tienen actividad microbiocida, en particular, actividad fungicida. (ver Fórmulas) Esquema de reacción 1.
MX2021012542A 2019-04-18 2020-04-16 Proceso para la preparacion de derivados de oxadiazol microbiocidas. MX2021012542A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN201911015611 2019-04-18
PCT/EP2020/060746 WO2020212513A1 (en) 2019-04-18 2020-04-16 Process for the preparation of microbiocidal oxadiazole derivatives

Publications (1)

Publication Number Publication Date
MX2021012542A true MX2021012542A (es) 2021-11-12

Family

ID=70292983

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2021012542A MX2021012542A (es) 2019-04-18 2020-04-16 Proceso para la preparacion de derivados de oxadiazol microbiocidas.

Country Status (12)

Country Link
US (1) US20220194907A1 (es)
EP (1) EP3956318A1 (es)
JP (1) JP2022529006A (es)
CN (1) CN113748105A (es)
AR (1) AR118673A1 (es)
BR (1) BR112021020673A2 (es)
CL (1) CL2021002713A1 (es)
CO (1) CO2021013497A2 (es)
IL (1) IL286566A (es)
MX (1) MX2021012542A (es)
UY (1) UY38667A (es)
WO (1) WO2020212513A1 (es)

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US20230172204A1 (en) 2020-04-28 2023-06-08 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors iii
CN115460919A (zh) 2020-04-28 2022-12-09 巴斯夫欧洲公司 嗜球果伞素类型化合物防除在线粒体细胞色素b蛋白中含有赋予对Qo抑制剂IV的耐受性的氨基酸替代F129L的植物病原性真菌的用途
US20230172207A1 (en) 2020-04-28 2023-06-08 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors i
CA3171545A1 (en) 2020-04-28 2021-11-04 Andreas Koch Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors i
BR112023000163A2 (pt) 2020-07-08 2023-01-31 Basf Se Compostos, composições agroquímicas, uso dos compostos e método para combater fungos fitopatogênicos
EP3939961A1 (en) 2020-07-16 2022-01-19 Basf Se Strobilurin type compounds and their use for combating phytopathogenic fungi
CN116056576A (zh) 2020-08-11 2023-05-02 巴斯夫欧洲公司 嗜球果伞素类型化合物防除在线粒体细胞色素b蛋白中含有赋予对Qo抑制剂VIII的耐受性的氨基酸替代F129L的植物病原性真菌的用途
WO2022106304A1 (en) 2020-11-23 2022-05-27 BASF Agro B.V. Compositions comprising mefentrifluconazole
WO2022117373A1 (en) 2020-12-01 2022-06-09 Basf Se Mixtures containing metarylpicoxamid
WO2022128554A1 (en) 2020-12-15 2022-06-23 Basf Se Mixtures containing n-methoxy-n-[[4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]cyclopropanecarboxamide
AR124367A1 (es) * 2020-12-17 2023-03-22 Fmc Corp Oxadiazoles fungicidas y sus mezclas
EP4018830A1 (en) 2020-12-23 2022-06-29 Basf Se Pesticidal mixtures
WO2022136000A1 (en) 2020-12-23 2022-06-30 Basf Se Pesticidal mixtures
BR112023023989A2 (pt) 2021-05-18 2024-01-30 Basf Se Compostos, composição, método para combater fungos fitopatogênicos e semente
WO2022243107A1 (en) 2021-05-18 2022-11-24 Basf Se New substituted pyridines as fungicides
CN117355519A (zh) 2021-05-18 2024-01-05 巴斯夫欧洲公司 用作杀真菌剂的新型取代吡啶类
WO2023280630A1 (en) 2021-07-08 2023-01-12 Basf Se Preparation of substituted amidoximes
WO2023285176A1 (en) * 2021-07-14 2023-01-19 Basf Se A process for producing alkyl trifluoroacetates
WO2023011957A1 (en) 2021-08-02 2023-02-09 Basf Se (3-quinolyl)-quinazoline
WO2023011958A1 (en) 2021-08-02 2023-02-09 Basf Se (3-pirydyl)-quinazoline
WO2023072670A1 (en) 2021-10-28 2023-05-04 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors x
WO2023072671A1 (en) 2021-10-28 2023-05-04 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors ix
EP4198023A1 (en) 2021-12-16 2023-06-21 Basf Se Pesticidally active thiosemicarbazone compounds
WO2023208447A1 (en) 2022-04-25 2023-11-02 Basf Se An emulsifiable concentrate having a (substituted) benzaldehyde-based solvent system
WO2024018016A1 (en) 2022-07-21 2024-01-25 Syngenta Crop Protection Ag Crystalline forms of 1,2,4-oxadiazole fungicides
EP4342885A1 (en) 2022-09-20 2024-03-27 Basf Se N-(3-(aminomethyl)-phenyl)-5-(4-phenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-amine derivatives and similar compounds as pesticides
EP4361126A1 (en) 2022-10-24 2024-05-01 Basf Se Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors xv

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Also Published As

Publication number Publication date
JP2022529006A (ja) 2022-06-16
CL2021002713A1 (es) 2022-05-27
CN113748105A (zh) 2021-12-03
EP3956318A1 (en) 2022-02-23
IL286566A (en) 2021-10-31
US20220194907A1 (en) 2022-06-23
CO2021013497A2 (es) 2022-01-28
WO2020212513A1 (en) 2020-10-22
UY38667A (es) 2020-11-30
BR112021020673A2 (pt) 2021-12-07
AR118673A1 (es) 2021-10-20

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