BR112021020673A2 - Processo para a preparação de derivados de oxadiazol microbiocidas - Google Patents
Processo para a preparação de derivados de oxadiazol microbiocidasInfo
- Publication number
- BR112021020673A2 BR112021020673A2 BR112021020673A BR112021020673A BR112021020673A2 BR 112021020673 A2 BR112021020673 A2 BR 112021020673A2 BR 112021020673 A BR112021020673 A BR 112021020673A BR 112021020673 A BR112021020673 A BR 112021020673A BR 112021020673 A2 BR112021020673 A2 BR 112021020673A2
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- oxadiazole derivatives
- microbiocidal
- microbiocidal oxadiazole
- activity
- Prior art date
Links
- 230000003641 microbiacidal effect Effects 0.000 title abstract 4
- 238000000034 method Methods 0.000 title abstract 3
- 150000004866 oxadiazoles Chemical class 0.000 title abstract 2
- XDOXQQBUPUADQB-UHFFFAOYSA-N 5-(trifluoromethyl)-1,2,4-oxadiazole Chemical class FC(F)(F)C1=NC=NO1 XDOXQQBUPUADQB-UHFFFAOYSA-N 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 230000000855 fungicidal effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
processo para a preparação de derivados de oxadiazol microbiocidas. a presente invenção se refere a um processo de acordo com o esquema 1 para a preparação de derivados de 5-trifluorometil-1,2,4-oxadiazol microbiocidas da fórmula (i) adequados para uso, por exemplo, como ingredientes ativos, que têm atividade microbicida, em particular, atividade fungicida.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN201911015611 | 2019-04-18 | ||
PCT/EP2020/060746 WO2020212513A1 (en) | 2019-04-18 | 2020-04-16 | Process for the preparation of microbiocidal oxadiazole derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112021020673A2 true BR112021020673A2 (pt) | 2021-12-07 |
Family
ID=70292983
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112021020673A BR112021020673A2 (pt) | 2019-04-18 | 2020-04-16 | Processo para a preparação de derivados de oxadiazol microbiocidas |
Country Status (12)
Country | Link |
---|---|
US (1) | US20220194907A1 (pt) |
EP (1) | EP3956318A1 (pt) |
JP (1) | JP2022529006A (pt) |
CN (1) | CN113748105B (pt) |
AR (1) | AR118673A1 (pt) |
BR (1) | BR112021020673A2 (pt) |
CL (1) | CL2021002713A1 (pt) |
CO (1) | CO2021013497A2 (pt) |
IL (1) | IL286566A (pt) |
MX (1) | MX2021012542A (pt) |
UY (1) | UY38667A (pt) |
WO (1) | WO2020212513A1 (pt) |
Families Citing this family (34)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2021266044A1 (en) | 2020-04-28 | 2022-11-24 | Basf Se | Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution F129L in the mitochondrial cytochrome b protein conferring resistance to Qo inhibitors IV |
CN115460920A (zh) | 2020-04-28 | 2022-12-09 | 巴斯夫欧洲公司 | 嗜球果伞素类型化合物防除在线粒体细胞色素b蛋白中含有赋予对Qo抑制剂II的耐受性的氨基酸替代F129L的植物病原性真菌的用途 |
CA3170923A1 (en) | 2020-04-28 | 2021-11-04 | Basf Se | Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors i |
CA3172204A1 (en) | 2020-04-28 | 2021-11-04 | Basf Se | Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors ii |
WO2022008303A1 (en) | 2020-07-08 | 2022-01-13 | Basf Se | Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors vi |
EP3939961A1 (en) | 2020-07-16 | 2022-01-19 | Basf Se | Strobilurin type compounds and their use for combating phytopathogenic fungi |
EP4195928A1 (en) | 2020-08-11 | 2023-06-21 | Basf Se | Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors viii |
WO2022106304A1 (en) | 2020-11-23 | 2022-05-27 | BASF Agro B.V. | Compositions comprising mefentrifluconazole |
US20240016150A1 (en) | 2020-12-01 | 2024-01-18 | Basf Se | Mixtures containing metarylpicoxamid |
WO2022128554A1 (en) | 2020-12-15 | 2022-06-23 | Basf Se | Mixtures containing n-methoxy-n-[[4-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]phenyl]methyl]cyclopropanecarboxamide |
AR124367A1 (es) * | 2020-12-17 | 2023-03-22 | Fmc Corp | Oxadiazoles fungicidas y sus mezclas |
EP4266885A1 (en) | 2020-12-23 | 2023-11-01 | Basf Se | Pesticidal mixtures |
EP4018830A1 (en) | 2020-12-23 | 2022-06-29 | Basf Se | Pesticidal mixtures |
CA3219311A1 (en) | 2021-05-18 | 2022-11-24 | Basf Se | New substituted quinolines as fungicides |
IL308534A (en) | 2021-05-18 | 2024-01-01 | Basf Se | New converted pyridines as fungicides |
CA3218900A1 (en) | 2021-05-18 | 2022-11-24 | Wassilios Grammenos | New substituted pyridines as fungicides |
EP4367101A1 (en) | 2021-07-08 | 2024-05-15 | Basf Se | Preparation of substituted amidoximes |
CN117642391A (zh) * | 2021-07-14 | 2024-03-01 | 巴斯夫欧洲公司 | 用于生产三氟乙酸烷基酯的方法 |
CN117794908A (zh) | 2021-08-02 | 2024-03-29 | 巴斯夫欧洲公司 | (3-喹啉基)-喹唑啉 |
WO2023011958A1 (en) | 2021-08-02 | 2023-02-09 | Basf Se | (3-pirydyl)-quinazoline |
WO2023072670A1 (en) | 2021-10-28 | 2023-05-04 | Basf Se | Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors x |
WO2023072671A1 (en) | 2021-10-28 | 2023-05-04 | Basf Se | Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors ix |
EP4198023A1 (en) | 2021-12-16 | 2023-06-21 | Basf Se | Pesticidally active thiosemicarbazone compounds |
WO2023208447A1 (en) | 2022-04-25 | 2023-11-02 | Basf Se | An emulsifiable concentrate having a (substituted) benzaldehyde-based solvent system |
WO2024018016A1 (en) | 2022-07-21 | 2024-01-25 | Syngenta Crop Protection Ag | Crystalline forms of 1,2,4-oxadiazole fungicides |
EP4342885A1 (en) | 2022-09-20 | 2024-03-27 | Basf Se | N-(3-(aminomethyl)-phenyl)-5-(4-phenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-amine derivatives and similar compounds as pesticides |
EP4361126A1 (en) | 2022-10-24 | 2024-05-01 | Basf Se | Use of strobilurin type compounds for combating phytopathogenic fungi containing an amino acid substitution f129l in the mitochondrial cytochrome b protein conferring resistance to qo inhibitors xv |
WO2024104813A1 (en) | 2022-11-14 | 2024-05-23 | Basf Se | Fungicidal mixture comprising substituted pyridines |
WO2024104815A1 (en) | 2022-11-16 | 2024-05-23 | Basf Se | Substituted benzodiazepines as fungicides |
WO2024104818A1 (en) | 2022-11-16 | 2024-05-23 | Basf Se | Substituted benzodiazepines as fungicides |
WO2024104814A1 (en) | 2022-11-16 | 2024-05-23 | Basf Se | Fungicidal mixture comprising substituted pyridines |
WO2024104822A1 (en) | 2022-11-16 | 2024-05-23 | Basf Se | Substituted tetrahydrobenzodiazepine as fungicides |
WO2024104823A1 (en) | 2022-11-16 | 2024-05-23 | Basf Se | New substituted tetrahydrobenzoxazepine |
EP4389210A1 (en) | 2022-12-21 | 2024-06-26 | Basf Se | Heteroaryl compounds for the control of invertebrate pests |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MXPA04003169A (es) | 2001-10-03 | 2004-07-08 | Pharmacia Corp | Profarmacos de compuestos policiclicos sustituidos utiles para inhibicion selectiva de la cascada de coagulacion. |
AU2006332694A1 (en) | 2005-12-30 | 2007-07-12 | Alantos Pharmaceuticals, Holding, Inc. | Substituted bis-amide metalloprotease inhibitors |
MY148430A (en) * | 2006-03-23 | 2013-04-30 | Biota Scient Management | Antibacterial agents |
WO2009022746A1 (ja) | 2007-08-10 | 2009-02-19 | Nippon Soda Co., Ltd. | 含窒素複素環化合物および有害生物防除剤 |
WO2013066838A1 (en) | 2011-10-31 | 2013-05-10 | Glaxosmithkline Llc | Compounds and methods |
WO2013066839A2 (en) | 2011-10-31 | 2013-05-10 | Glaxosmithkline Llc | Compounds and methods |
CN104302358B (zh) * | 2012-03-07 | 2017-12-05 | 癌症研究协会:皇家癌症医院 | 3‑芳基‑5‑取代的异喹啉‑1‑酮化合物和它们的治疗用途 |
HUE050030T2 (hu) * | 2015-10-02 | 2020-11-30 | Syngenta Participations Ag | Mikrobiocid oxadiazol-származékok |
US11066396B2 (en) * | 2016-06-23 | 2021-07-20 | Merck Sharp & Dohme Corp. | 3-aryl- heteroaryl substituted 5-trifluoromethyl oxadiazoles as histonedeacetylase 6 (HDAC6) inhibitors |
WO2018177880A1 (en) * | 2017-03-31 | 2018-10-04 | Syngenta Participations Ag | Fungicidal compositions |
MX2019011239A (es) | 2017-03-31 | 2019-10-21 | Syngenta Participations Ag | Composiciones fungicidas. |
WO2018184985A1 (en) * | 2017-04-05 | 2018-10-11 | Syngenta Participations Ag | Microbiocidal oxadiazole derivatives |
BR112019024993A2 (pt) * | 2017-06-02 | 2020-06-16 | Syngenta Participations Ag | Composições fungicidas |
-
2020
- 2020-04-15 AR ARP200101052A patent/AR118673A1/es unknown
- 2020-04-16 EP EP20719634.6A patent/EP3956318A1/en active Pending
- 2020-04-16 WO PCT/EP2020/060746 patent/WO2020212513A1/en active Application Filing
- 2020-04-16 JP JP2021561026A patent/JP2022529006A/ja active Pending
- 2020-04-16 US US17/594,469 patent/US20220194907A1/en active Pending
- 2020-04-16 CN CN202080029013.5A patent/CN113748105B/zh active Active
- 2020-04-16 MX MX2021012542A patent/MX2021012542A/es unknown
- 2020-04-16 BR BR112021020673A patent/BR112021020673A2/pt unknown
- 2020-04-16 UY UY0001038667A patent/UY38667A/es unknown
-
2021
- 2021-09-22 IL IL286566A patent/IL286566A/en unknown
- 2021-10-11 CO CONC2021/0013497A patent/CO2021013497A2/es unknown
- 2021-10-15 CL CL2021002713A patent/CL2021002713A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
US20220194907A1 (en) | 2022-06-23 |
CN113748105A (zh) | 2021-12-03 |
IL286566A (en) | 2021-10-31 |
CL2021002713A1 (es) | 2022-05-27 |
UY38667A (es) | 2020-11-30 |
JP2022529006A (ja) | 2022-06-16 |
CO2021013497A2 (es) | 2022-01-28 |
AR118673A1 (es) | 2021-10-20 |
WO2020212513A1 (en) | 2020-10-22 |
CN113748105B (zh) | 2024-06-11 |
EP3956318A1 (en) | 2022-02-23 |
MX2021012542A (es) | 2021-11-12 |
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