CL2009000490A1 - Procesos de preparacion de (fenilsulfanilfenil)piperidinas a partir de una n-bencil-piperidona; los intermediarios considerados; y la preparacion de uno de ellos. - Google Patents

Procesos de preparacion de (fenilsulfanilfenil)piperidinas a partir de una n-bencil-piperidona; los intermediarios considerados; y la preparacion de uno de ellos.

Info

Publication number
CL2009000490A1
CL2009000490A1 CL2009000490A CL2009000490A CL2009000490A1 CL 2009000490 A1 CL2009000490 A1 CL 2009000490A1 CL 2009000490 A CL2009000490 A CL 2009000490A CL 2009000490 A CL2009000490 A CL 2009000490A CL 2009000490 A1 CL2009000490 A1 CL 2009000490A1
Authority
CL
Chile
Prior art keywords
preparation
phenylsulfanylphenyl
piperidone
intermediaries
piperidines
Prior art date
Application number
CL2009000490A
Other languages
English (en)
Spanish (es)
Inventor
Michael Harold Rock
Sebastian Brandes
Original Assignee
H Lundbeck As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by H Lundbeck As filed Critical H Lundbeck As
Publication of CL2009000490A1 publication Critical patent/CL2009000490A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/52—Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CL2009000490A 2008-03-03 2009-03-02 Procesos de preparacion de (fenilsulfanilfenil)piperidinas a partir de una n-bencil-piperidona; los intermediarios considerados; y la preparacion de uno de ellos. CL2009000490A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DKPA200800314 2008-03-03

Publications (1)

Publication Number Publication Date
CL2009000490A1 true CL2009000490A1 (es) 2010-04-16

Family

ID=40547924

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2009000490A CL2009000490A1 (es) 2008-03-03 2009-03-02 Procesos de preparacion de (fenilsulfanilfenil)piperidinas a partir de una n-bencil-piperidona; los intermediarios considerados; y la preparacion de uno de ellos.

Country Status (28)

Country Link
US (1) US8362255B2 (OSRAM)
EP (1) EP2260024B1 (OSRAM)
JP (1) JP5564439B2 (OSRAM)
KR (1) KR20100122914A (OSRAM)
CN (1) CN101959859B (OSRAM)
AR (1) AR070737A1 (OSRAM)
AT (1) ATE539055T1 (OSRAM)
AU (1) AU2009221170B2 (OSRAM)
BR (1) BRPI0908166A2 (OSRAM)
CA (1) CA2715579A1 (OSRAM)
CL (1) CL2009000490A1 (OSRAM)
CO (1) CO6290758A2 (OSRAM)
CY (1) CY1113887T1 (OSRAM)
DK (1) DK2260024T3 (OSRAM)
EA (1) EA017855B1 (OSRAM)
ES (1) ES2377862T3 (OSRAM)
HR (1) HRP20120118T1 (OSRAM)
IL (1) IL207471A (OSRAM)
MX (1) MX2010008729A (OSRAM)
NZ (1) NZ587593A (OSRAM)
PL (1) PL2260024T3 (OSRAM)
PT (1) PT2260024E (OSRAM)
RS (1) RS52128B (OSRAM)
SI (1) SI2260024T1 (OSRAM)
TW (1) TW200940505A (OSRAM)
UA (1) UA98698C2 (OSRAM)
WO (1) WO2009109541A1 (OSRAM)
ZA (1) ZA201006135B (OSRAM)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8299095B2 (en) * 2006-06-16 2012-10-30 H. Lundbeck A/S Crystalline forms of 4-[2-(4-methylphenylsulfanyl)-phenyl] piperidine with combined serotonin and norepinephrine reuptake inhibition and uses thereof
JP2012163850A (ja) * 2011-02-08 2012-08-30 Nippon Sheet Glass Co Ltd 正立等倍レンズアレイプレート、光走査ユニット、画像読取装置および画像書込装置
US8987457B2 (en) 2012-05-21 2015-03-24 Novartis Ag Ring-substituted N-pyridinyl amides as kinase inhibitors
CN104710345B (zh) * 2013-12-17 2017-09-05 江苏恩华药业股份有限公司 用于制备4‑（2‑（4‑甲基苯基硫基））苯基哌啶的化合物、其制备方法及应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2324087A (en) * 1997-04-10 1998-10-14 Merck & Co Inc Preparation of (S)-3-Carbethoxy-3-benzylpiperidine
WO2001046147A1 (en) 1999-12-20 2001-06-28 Eli Lilly And Company A process for preparing 4-substituted piperidines
UA81749C2 (uk) * 2001-10-04 2008-02-11 Х. Луннбек А/С Фенілпіперазинові похідні як інгібітори зворотного захоплення серотоніну
UA81300C2 (en) * 2003-04-04 2007-12-25 Lundbeck & Co As H Derivates of 4-(2-fenilsulfanilfenil)-1,2,3,6-tetrahydropiridin as retarding agents of serotonin recapture
DK1626720T3 (da) * 2003-04-04 2008-12-01 Lundbeck & Co As H 4-(2-Phenylsulfanyl-phenyl)-piperidinderivater som serotonin-genoptagelseshæmmer
US8299095B2 (en) * 2006-06-16 2012-10-30 H. Lundbeck A/S Crystalline forms of 4-[2-(4-methylphenylsulfanyl)-phenyl] piperidine with combined serotonin and norepinephrine reuptake inhibition and uses thereof

Also Published As

Publication number Publication date
CA2715579A1 (en) 2009-09-11
PT2260024E (pt) 2012-03-06
WO2009109541A1 (en) 2009-09-11
EP2260024A1 (en) 2010-12-15
KR20100122914A (ko) 2010-11-23
HK1153458A1 (en) 2012-03-30
US8362255B2 (en) 2013-01-29
AU2009221170A1 (en) 2009-09-11
US20110054178A1 (en) 2011-03-03
ES2377862T3 (es) 2012-04-02
IL207471A (en) 2014-06-30
CO6290758A2 (es) 2011-06-20
SI2260024T1 (sl) 2012-04-30
EA201071025A1 (ru) 2011-02-28
NZ587593A (en) 2012-03-30
CY1113887T1 (el) 2016-07-27
EA017855B1 (ru) 2013-03-29
BRPI0908166A2 (pt) 2015-08-11
AU2009221170B2 (en) 2013-08-22
CN101959859B (zh) 2013-08-14
RS52128B (sr) 2012-08-31
AR070737A1 (es) 2010-04-28
ZA201006135B (en) 2011-10-26
PL2260024T3 (pl) 2012-04-30
JP2011513358A (ja) 2011-04-28
ATE539055T1 (de) 2012-01-15
MX2010008729A (es) 2010-09-24
HRP20120118T1 (hr) 2012-03-31
EP2260024B1 (en) 2011-12-28
UA98698C2 (en) 2012-06-11
JP5564439B2 (ja) 2014-07-30
CN101959859A (zh) 2011-01-26
TW200940505A (en) 2009-10-01
IL207471A0 (en) 2010-12-30
DK2260024T3 (da) 2012-02-27

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