CL2004000805A1 - Compuestos derivados de 7-aza-quinazolina sustituida, inhibidores de quinasa p38; procedimiento de preparacion; composicion farmaceutica; y su uso para tratar artritis, enfermedad de crohn, alzheimer, asma, ataque al corazon. - Google Patents
Compuestos derivados de 7-aza-quinazolina sustituida, inhibidores de quinasa p38; procedimiento de preparacion; composicion farmaceutica; y su uso para tratar artritis, enfermedad de crohn, alzheimer, asma, ataque al corazon.Info
- Publication number
- CL2004000805A1 CL2004000805A1 CL200400805A CL2004000805A CL2004000805A1 CL 2004000805 A1 CL2004000805 A1 CL 2004000805A1 CL 200400805 A CL200400805 A CL 200400805A CL 2004000805 A CL2004000805 A CL 2004000805A CL 2004000805 A1 CL2004000805 A1 CL 2004000805A1
- Authority
- CL
- Chile
- Prior art keywords
- quinazolina
- quinasa
- aza
- crohn
- alzheimer
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pulmonology (AREA)
- Biomedical Technology (AREA)
- Cardiology (AREA)
- Physical Education & Sports Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Hematology (AREA)
- Psychiatry (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Urology & Nephrology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US46322903P | 2003-04-16 | 2003-04-16 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2004000805A1 true CL2004000805A1 (es) | 2005-02-04 |
Family
ID=33300055
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL200400805A CL2004000805A1 (es) | 2003-04-16 | 2004-04-15 | Compuestos derivados de 7-aza-quinazolina sustituida, inhibidores de quinasa p38; procedimiento de preparacion; composicion farmaceutica; y su uso para tratar artritis, enfermedad de crohn, alzheimer, asma, ataque al corazon. |
Country Status (16)
Country | Link |
---|---|
US (2) | US7189731B2 (es) |
EP (1) | EP1620105B1 (es) |
JP (1) | JP2006523640A (es) |
KR (1) | KR20060006037A (es) |
CN (1) | CN1774250A (es) |
AR (1) | AR044515A1 (es) |
AU (1) | AU2004229163A1 (es) |
BR (1) | BRPI0409405A (es) |
CA (1) | CA2520785A1 (es) |
CL (1) | CL2004000805A1 (es) |
DE (1) | DE602004004259T2 (es) |
ES (1) | ES2279361T3 (es) |
MX (1) | MXPA05010975A (es) |
RU (1) | RU2005135329A (es) |
TW (1) | TW200503722A (es) |
WO (1) | WO2004091625A1 (es) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102004020908A1 (de) * | 2004-04-28 | 2005-11-17 | Grünenthal GmbH | Substituierte 5,6,7,8,-Tetrahydro-pyrido[4,3-d]pyrimidin-2-yl- und 5,6,7,8,-Tetrahydro-chinazolin-2-yl-Verbindungen |
US20090131430A1 (en) * | 2004-11-23 | 2009-05-21 | Palle Venkata P | Pyrido'2,3-dipyrimidines as anti-inflammatory agents |
ES2303758B1 (es) * | 2006-02-20 | 2009-08-13 | Laboratorios Almirall S.A. | Nuevos derivados de piridin-3-amina. |
EP1992344A1 (en) | 2007-05-18 | 2008-11-19 | Institut Curie | P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation |
BRPI1011505A2 (pt) | 2009-03-11 | 2016-03-22 | Auckland Uniservices Ltd | formas de pró-drogas de inibidores de quinase e sua aplicação em terapia |
WO2011028135A1 (en) | 2009-09-02 | 2011-03-10 | Auckland Uniservices Limited | Kinase inhibitors, prodrug forms thereof and their use in therapy |
WO2017151409A1 (en) | 2016-02-29 | 2017-09-08 | University Of Florida Research Foundation, Incorporated | Chemotherapeutic methods |
US10342786B2 (en) | 2017-10-05 | 2019-07-09 | Fulcrum Therapeutics, Inc. | P38 kinase inhibitors reduce DUX4 and downstream gene expression for the treatment of FSHD |
WO2019071144A1 (en) | 2017-10-05 | 2019-04-11 | Fulcrum Therapeutics, Inc. | USE OF P38 INHIBITORS TO REDUCE DUX4 EXPRESSION |
Family Cites Families (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1199768A (en) * | 1966-10-31 | 1970-07-22 | Pfizer & Co C | Nitrogen Heterocycles and process for their preparation |
JPS4936700A (es) * | 1972-08-16 | 1974-04-05 | ||
US4672116A (en) * | 1985-12-20 | 1987-06-09 | Ortho Pharmaceutical Corporation | Substituted 5,6-dialkoxyquinazoline derivatives |
US5084463A (en) * | 1989-12-11 | 1992-01-28 | American Home Products Corporation | N-quinolinyl alkyl-substituted 1-aryloxy-2-propanolamine and propylamine derivatives possessing class III antiarrhythmic activity |
US20020061879A1 (en) * | 1996-02-02 | 2002-05-23 | Garvey David S. | Nitrosated and nitrosylated alpha-adrenergic receptor antagonist compounds, compositions and their uses |
EP1014953B1 (en) | 1997-03-05 | 2012-04-25 | Sugen, Inc. | Formulations for hydrophobic pharmaceutical agents |
US6313294B1 (en) * | 1998-02-04 | 2001-11-06 | Development Center For Biotechnology | Process for preparing amides |
AU1071301A (en) | 1999-11-01 | 2001-05-14 | Eli Lilly And Company | Pharmaceutical compounds |
EP1235815A1 (en) | 1999-11-22 | 2002-09-04 | Warner-Lambert Company | Quinazolines and their use for inhibiting cyclin-dependent kinase enzymes |
EP1110552A1 (en) | 1999-12-22 | 2001-06-27 | Aventis Pharma S.A. | Use of a compound with affinity for the mitochondrial benzodiazepine receptor in cancer therapy |
WO2001064646A2 (en) | 2000-03-01 | 2001-09-07 | Tularik Inc. | Hydrazones and analogs as cholesterol lowering agents |
MXPA03000708A (es) | 2000-07-26 | 2003-06-04 | Smithkline Beecham Plc | Aminopiperidin quinolinas y sus analogos azaisostericos con actividad antibacteriana. |
AUPR213700A0 (en) | 2000-12-18 | 2001-01-25 | Biota Scientific Management Pty Ltd | Antiviral agents |
KR100639772B1 (ko) * | 2001-02-12 | 2006-10-30 | 에프. 호프만-라 로슈 아게 | 6-치환된 피리도-피리미딘 |
DE60231868D1 (de) | 2001-04-24 | 2009-05-20 | Purdue Research Foundation | Folat-mimetika und deren folatrezeptorbindende konjugate |
WO2002090360A1 (en) * | 2001-05-10 | 2002-11-14 | Smithkline Beecham Corporation | Compounds useful as kinase inhibitors for the treatment of hyperproliferative diseases |
ATE374201T1 (de) * | 2002-08-06 | 2007-10-15 | Hoffmann La Roche | 6-alkoxypyridopyrimidine als inhibitoren der p-38-map-kinase |
-
2004
- 2004-04-13 KR KR1020057019705A patent/KR20060006037A/ko not_active Application Discontinuation
- 2004-04-13 RU RU2005135329/04A patent/RU2005135329A/ru not_active Application Discontinuation
- 2004-04-13 CN CNA2004800099562A patent/CN1774250A/zh active Pending
- 2004-04-13 BR BRPI0409405-0A patent/BRPI0409405A/pt not_active Application Discontinuation
- 2004-04-13 JP JP2006505106A patent/JP2006523640A/ja active Pending
- 2004-04-13 ES ES04726958T patent/ES2279361T3/es not_active Expired - Lifetime
- 2004-04-13 AU AU2004229163A patent/AU2004229163A1/en not_active Abandoned
- 2004-04-13 MX MXPA05010975A patent/MXPA05010975A/es not_active Application Discontinuation
- 2004-04-13 WO PCT/EP2004/003883 patent/WO2004091625A1/en active IP Right Grant
- 2004-04-13 DE DE602004004259T patent/DE602004004259T2/de not_active Expired - Fee Related
- 2004-04-13 CA CA002520785A patent/CA2520785A1/en not_active Abandoned
- 2004-04-13 EP EP04726958A patent/EP1620105B1/en not_active Expired - Lifetime
- 2004-04-15 CL CL200400805A patent/CL2004000805A1/es unknown
- 2004-04-15 US US10/824,980 patent/US7189731B2/en not_active Expired - Fee Related
- 2004-04-15 TW TW093110567A patent/TW200503722A/zh unknown
- 2004-04-15 AR ARP040101263A patent/AR044515A1/es unknown
-
2007
- 2007-01-09 US US11/651,320 patent/US20070135459A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
DE602004004259T2 (de) | 2007-11-15 |
TW200503722A (en) | 2005-02-01 |
CA2520785A1 (en) | 2004-10-28 |
EP1620105A1 (en) | 2006-02-01 |
EP1620105B1 (en) | 2007-01-10 |
CN1774250A (zh) | 2006-05-17 |
BRPI0409405A (pt) | 2006-04-25 |
US20070135459A1 (en) | 2007-06-14 |
US20040209903A1 (en) | 2004-10-21 |
RU2005135329A (ru) | 2006-08-10 |
US7189731B2 (en) | 2007-03-13 |
MXPA05010975A (es) | 2005-11-28 |
AU2004229163A1 (en) | 2004-10-28 |
KR20060006037A (ko) | 2006-01-18 |
DE602004004259D1 (de) | 2007-02-22 |
JP2006523640A (ja) | 2006-10-19 |
ES2279361T3 (es) | 2007-08-16 |
WO2004091625A1 (en) | 2004-10-28 |
AR044515A1 (es) | 2005-09-14 |
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