CH619685A5 - Process for the preparation of 3-fluoro-D-alanine or 2-deutero-3-fluoro-D-alanine - Google Patents

Process for the preparation of 3-fluoro-D-alanine or 2-deutero-3-fluoro-D-alanine Download PDF

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Publication number
CH619685A5
CH619685A5 CH1459075A CH1459075A CH619685A5 CH 619685 A5 CH619685 A5 CH 619685A5 CH 1459075 A CH1459075 A CH 1459075A CH 1459075 A CH1459075 A CH 1459075A CH 619685 A5 CH619685 A5 CH 619685A5
Authority
CH
Switzerland
Prior art keywords
reacted
alanine
fluoro
deutero
substituted
Prior art date
Application number
CH1459075A
Other languages
German (de)
English (en)
Inventor
Donald Floyd Reinhold
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/525,708 external-priority patent/US3976689A/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of CH619685A5 publication Critical patent/CH619685A5/de

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/04Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C229/20Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B53/00Asymmetric syntheses
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N37/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/44Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing at least one carboxylic group or a thio analogue, or a derivative thereof, and a nitrogen atom attached to the same carbon skeleton by a single or double bond, this nitrogen atom not being a member of a derivative or of a thio analogue of a carboxylic group, e.g. amino-carboxylic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • C07B59/001Acyclic or carbocyclic compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/04Formation of amino groups in compounds containing carboxyl groups
    • C07C227/06Formation of amino groups in compounds containing carboxyl groups by addition or substitution reactions, without increasing the number of carbon atoms in the carbon skeleton of the acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/05Isotopically modified compounds, e.g. labelled

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Indole Compounds (AREA)
CH1459075A 1974-11-20 1975-11-11 Process for the preparation of 3-fluoro-D-alanine or 2-deutero-3-fluoro-D-alanine CH619685A5 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/525,708 US3976689A (en) 1972-02-03 1974-11-20 Process for preparing 3-fluoro-D-alanine and its deutero analogs

Publications (1)

Publication Number Publication Date
CH619685A5 true CH619685A5 (en) 1980-10-15

Family

ID=24094311

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1459075A CH619685A5 (en) 1974-11-20 1975-11-11 Process for the preparation of 3-fluoro-D-alanine or 2-deutero-3-fluoro-D-alanine

Country Status (9)

Country Link
JP (1) JPS5175020A (enrdf_load_html_response)
CH (1) CH619685A5 (enrdf_load_html_response)
DD (1) DD124972A5 (enrdf_load_html_response)
DK (1) DK515575A (enrdf_load_html_response)
ES (1) ES442779A1 (enrdf_load_html_response)
FI (1) FI753167A7 (enrdf_load_html_response)
NL (1) NL7513137A (enrdf_load_html_response)
NO (1) NO753750L (enrdf_load_html_response)
SE (1) SE7512699L (enrdf_load_html_response)

Also Published As

Publication number Publication date
DD124972A5 (enrdf_load_html_response) 1977-03-23
NL7513137A (nl) 1976-05-24
SE7512699L (sv) 1976-05-21
ES442779A1 (es) 1977-09-16
FI753167A7 (enrdf_load_html_response) 1976-05-21
DK515575A (da) 1976-05-21
NO753750L (enrdf_load_html_response) 1976-05-21
JPS5175020A (en) 1976-06-29

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