CH558374A - Verfahren zur herstellung von arylsubstituierten piperazinylalkyl- bezw. alkenyl- chinazolon-(4)-derivaten. - Google Patents
Verfahren zur herstellung von arylsubstituierten piperazinylalkyl- bezw. alkenyl- chinazolon-(4)-derivaten.Info
- Publication number
- CH558374A CH558374A CH450074A CH450074A CH558374A CH 558374 A CH558374 A CH 558374A CH 450074 A CH450074 A CH 450074A CH 450074 A CH450074 A CH 450074A CH 558374 A CH558374 A CH 558374A
- Authority
- CH
- Switzerland
- Prior art keywords
- chinazolone
- alkenyl
- aryl
- derivatives
- production
- Prior art date
Links
- -1 PIPERAZINYL Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19702027645 DE2027645A1 (de) | 1970-06-05 | 1970-06-05 | Piperazinylalkyl chinazolon (4) den vate, Verfahren zu deren Herstellung und sie enthaltende Arzneimittel |
Publications (1)
Publication Number | Publication Date |
---|---|
CH558374A true CH558374A (de) | 1975-01-31 |
Family
ID=5773104
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CH450074A CH558374A (de) | 1970-06-05 | 1971-06-02 | Verfahren zur herstellung von arylsubstituierten piperazinylalkyl- bezw. alkenyl- chinazolon-(4)-derivaten. |
CH802071A CH557829A (de) | 1970-06-05 | 1971-06-02 | Verfahren zur herstellung von arylsubstituierten piperazinyl-alkyl- bzw. -alkenyl-chinazolon-(4)-derivaten. |
CH450174A CH569732A5 (forum.php) | 1970-06-05 | 1971-06-02 |
Family Applications After (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CH802071A CH557829A (de) | 1970-06-05 | 1971-06-02 | Verfahren zur herstellung von arylsubstituierten piperazinyl-alkyl- bzw. -alkenyl-chinazolon-(4)-derivaten. |
CH450174A CH569732A5 (forum.php) | 1970-06-05 | 1971-06-02 |
Country Status (10)
Country | Link |
---|---|
US (1) | US3984555A (forum.php) |
AT (3) | AT317899B (forum.php) |
BE (1) | BE768137A (forum.php) |
CA (1) | CA951319A (forum.php) |
CH (3) | CH558374A (forum.php) |
DE (1) | DE2027645A1 (forum.php) |
FR (1) | FR2100726B1 (forum.php) |
GB (1) | GB1331522A (forum.php) |
LU (1) | LU63267A1 (forum.php) |
NL (1) | NL7107695A (forum.php) |
Families Citing this family (32)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4287341A (en) * | 1979-11-01 | 1981-09-01 | Pfizer Inc. | Alkoxy-substituted-6-chloro-quinazoline-2,4-diones |
US6723727B1 (en) * | 1996-12-20 | 2004-04-20 | Hoechst Aktiengesellschaft | Substituted purine derivatives, processes for their preparation, their use, and compositions comprising them |
EP0903344B1 (en) * | 1997-08-21 | 2011-01-26 | Shiseido Co., Ltd. | Quinazolin-4-one derivatives, their preparation and their use as hair growth promoters or in external compositions for skin |
WO2001025234A1 (en) * | 1999-10-01 | 2001-04-12 | Advanced Medicine, Inc. | Quinazolinones and analogues and their use as local anesthetics |
US6667300B2 (en) * | 2000-04-25 | 2003-12-23 | Icos Corporation | Inhibitors of human phosphatidylinositol 3-kinase delta |
EP3029041B1 (en) * | 2000-04-25 | 2020-03-04 | ICOS Corporation | Inhibitors of human phosphatidyl-inositol 3-kinase delta |
AUPR201600A0 (en) * | 2000-12-11 | 2001-01-11 | Fujisawa Pharmaceutical Co., Ltd. | Quinazolinone derivative |
EP2329822A1 (en) | 2001-09-05 | 2011-06-08 | Minerva Biotechnologies Corporation | Compositions and methods of treatment of cancer |
JP2005501887A (ja) * | 2001-09-05 | 2005-01-20 | ミナーヴァ・バイオテクノロジーズ・コーポレーション | 癌の処置における組成物およびその使用 |
JP2005511581A (ja) * | 2001-11-07 | 2005-04-28 | メルク エンド カムパニー インコーポレーテッド | 有糸分裂キネシン阻害剤 |
AUPS019702A0 (en) * | 2002-01-29 | 2002-02-21 | Fujisawa Pharmaceutical Co., Ltd. | Condensed heterocyclic compounds |
US20040048853A1 (en) * | 2002-08-21 | 2004-03-11 | Gustave Bergnes | Compounds, compositions, and methods |
WO2004041755A2 (en) * | 2002-11-04 | 2004-05-21 | Nps Pharmaceuticals, Inc. | Quinazolinone compounds as calcilytics |
DE602004022819D1 (de) * | 2003-06-06 | 2009-10-08 | Vertex Pharma | Von atp-bindende kassette transportern |
US20050043239A1 (en) * | 2003-08-14 | 2005-02-24 | Jason Douangpanya | Methods of inhibiting immune responses stimulated by an endogenous factor |
WO2005016349A1 (en) * | 2003-08-14 | 2005-02-24 | Icos Corporation | Methods of inhibiting leukocyte accumulation |
USRE44638E1 (en) | 2004-05-13 | 2013-12-10 | Icos Corporation | Quinazolinones as inhibitors of human phosphatidylinositol 3-kinase delta |
EP1755609A1 (en) * | 2004-05-25 | 2007-02-28 | Icos Corporation | Methods for treating and/or preventing aberrant proliferation of hematopoietic cells |
CA2598409A1 (en) * | 2005-02-17 | 2006-08-24 | Icos Corporation | Phosphoinositide 3-kinase inhibitors for inhibiting leukocyte accumulation |
CA2680789C (en) * | 2006-03-28 | 2016-02-16 | Atir Holding S.A. | Heterocyclic compounds and uses thereof in the treatment of sexual disorders |
KR20160091440A (ko) | 2008-11-13 | 2016-08-02 | 길리아드 칼리스토가 엘엘씨 | 혈액 종양에 대한 요법 |
US9492449B2 (en) | 2008-11-13 | 2016-11-15 | Gilead Calistoga Llc | Therapies for hematologic malignancies |
BRPI1012333A2 (pt) | 2009-03-24 | 2016-03-29 | Gilead Calistoga Llc | atropisômeros de derivados de 2-purinil-3-tolil-quinazolinonas e métodos de uso |
ES2548253T3 (es) * | 2009-04-20 | 2015-10-15 | Gilead Calistoga Llc | Métodos para el tratamiento de tumores sólidos |
EP2456443A1 (en) | 2009-07-21 | 2012-05-30 | Gilead Calistoga LLC | Treatment of liver disorders with pi3k inhibitors |
BRPI1003506B1 (pt) | 2010-09-24 | 2019-12-03 | Ache Int Bvi Ltd | composto alquil-piperazino-fenil-4(3h)quinazolinonas e uso do composto alquil-piperazino-fenil-4(3h)quinazolinonas associado aos receptores serotoninérgicos 5-ht1a e 5-ht2a |
WO2012140642A1 (en) * | 2011-04-10 | 2012-10-18 | Atir Holding S.A. | Heterocyclic compounds and uses thereof in the treatment of sexual disorders |
KR20140133590A (ko) | 2012-03-05 | 2014-11-19 | 길리아드 칼리스토가 엘엘씨 | (s)-2-(1-(9h-퓨린-6-일아미노)프로필)-5-플루오로-3-페닐퀴나졸린-4(3h)-온의 다형체 형태 |
IN2015MN00002A (forum.php) | 2012-07-09 | 2015-10-16 | Lupin Ltd | |
EP3083623A1 (en) | 2013-12-20 | 2016-10-26 | Gilead Calistoga LLC | Polymorphic forms of a hydrochloride salt of (s) -2-(9h-purin-6-ylamino) propyl) -5-fluoro-3-phenylquinazolin-4 (3h) -one |
EA201690990A1 (ru) | 2013-12-20 | 2016-11-30 | Джилид Калистога Ллс | Способы получения ингибиторов фосфатидилинозитол-3-киназы |
JP6455995B2 (ja) | 2014-06-13 | 2019-01-23 | ギリアード サイエンシーズ, インコーポレイテッド | ホスファチジルイノシトール3−キナーゼ阻害剤 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1053063A (forum.php) * | 1963-05-18 |
-
1970
- 1970-06-05 DE DE19702027645 patent/DE2027645A1/de active Pending
-
1971
- 1971-05-28 US US05/148,100 patent/US3984555A/en not_active Expired - Lifetime
- 1971-06-01 AT AT244273A patent/AT317899B/de not_active IP Right Cessation
- 1971-06-01 AT AT470571A patent/AT318615B/de not_active IP Right Cessation
- 1971-06-01 AT AT244173A patent/AT318628B/de not_active IP Right Cessation
- 1971-06-02 CH CH450074A patent/CH558374A/xx not_active IP Right Cessation
- 1971-06-02 CH CH802071A patent/CH557829A/xx not_active IP Right Cessation
- 1971-06-02 CH CH450174A patent/CH569732A5/xx not_active IP Right Cessation
- 1971-06-02 LU LU63267D patent/LU63267A1/xx unknown
- 1971-06-03 GB GB1880371*[A patent/GB1331522A/en not_active Expired
- 1971-06-03 CA CA114,709,A patent/CA951319A/en not_active Expired
- 1971-06-04 BE BE768137A patent/BE768137A/xx unknown
- 1971-06-04 NL NL7107695A patent/NL7107695A/xx unknown
- 1971-06-04 FR FR7120368A patent/FR2100726B1/fr not_active Expired
Also Published As
Publication number | Publication date |
---|---|
LU63267A1 (forum.php) | 1972-08-23 |
FR2100726B1 (forum.php) | 1975-10-10 |
CH557829A (de) | 1975-01-15 |
AT317899B (de) | 1974-09-25 |
CA951319A (en) | 1974-07-16 |
US3984555A (en) | 1976-10-05 |
GB1331522A (en) | 1973-09-26 |
NL7107695A (forum.php) | 1971-12-07 |
AT318615B (de) | 1974-11-11 |
AT318628B (de) | 1974-11-11 |
FR2100726A1 (forum.php) | 1972-03-24 |
BE768137A (fr) | 1971-12-06 |
CH569732A5 (forum.php) | 1975-11-28 |
DE2027645A1 (de) | 1971-12-09 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PL | Patent ceased |