CH558374A - Verfahren zur herstellung von arylsubstituierten piperazinylalkyl- bezw. alkenyl- chinazolon-(4)-derivaten. - Google Patents
Verfahren zur herstellung von arylsubstituierten piperazinylalkyl- bezw. alkenyl- chinazolon-(4)-derivaten.Info
- Publication number
- CH558374A CH558374A CH450074A CH450074A CH558374A CH 558374 A CH558374 A CH 558374A CH 450074 A CH450074 A CH 450074A CH 450074 A CH450074 A CH 450074A CH 558374 A CH558374 A CH 558374A
- Authority
- CH
- Switzerland
- Prior art keywords
- chinazolone
- alkenyl
- aryl
- derivatives
- production
- Prior art date
Links
- -1 PIPERAZINYL Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19702027645 DE2027645A1 (de) | 1970-06-05 | 1970-06-05 | Piperazinylalkyl chinazolon (4) den vate, Verfahren zu deren Herstellung und sie enthaltende Arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CH558374A true CH558374A (de) | 1975-01-31 |
Family
ID=5773104
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH802071A CH557829A (de) | 1970-06-05 | 1971-06-02 | Verfahren zur herstellung von arylsubstituierten piperazinyl-alkyl- bzw. -alkenyl-chinazolon-(4)-derivaten. |
| CH450074A CH558374A (de) | 1970-06-05 | 1971-06-02 | Verfahren zur herstellung von arylsubstituierten piperazinylalkyl- bezw. alkenyl- chinazolon-(4)-derivaten. |
| CH450174A CH569732A5 (OSRAM) | 1970-06-05 | 1971-06-02 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH802071A CH557829A (de) | 1970-06-05 | 1971-06-02 | Verfahren zur herstellung von arylsubstituierten piperazinyl-alkyl- bzw. -alkenyl-chinazolon-(4)-derivaten. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH450174A CH569732A5 (OSRAM) | 1970-06-05 | 1971-06-02 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US3984555A (OSRAM) |
| AT (3) | AT318628B (OSRAM) |
| BE (1) | BE768137A (OSRAM) |
| CA (1) | CA951319A (OSRAM) |
| CH (3) | CH557829A (OSRAM) |
| DE (1) | DE2027645A1 (OSRAM) |
| FR (1) | FR2100726B1 (OSRAM) |
| GB (1) | GB1331522A (OSRAM) |
| LU (1) | LU63267A1 (OSRAM) |
| NL (1) | NL7107695A (OSRAM) |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4287341A (en) * | 1979-11-01 | 1981-09-01 | Pfizer Inc. | Alkoxy-substituted-6-chloro-quinazoline-2,4-diones |
| US6723727B1 (en) * | 1996-12-20 | 2004-04-20 | Hoechst Aktiengesellschaft | Substituted purine derivatives, processes for their preparation, their use, and compositions comprising them |
| EP0903344B1 (en) * | 1997-08-21 | 2011-01-26 | Shiseido Co., Ltd. | Quinazolin-4-one derivatives, their preparation and their use as hair growth promoters or in external compositions for skin |
| US6436919B1 (en) | 1999-10-01 | 2002-08-20 | Theravance Inc. | Local anesthetic compounds |
| US6667300B2 (en) | 2000-04-25 | 2003-12-23 | Icos Corporation | Inhibitors of human phosphatidylinositol 3-kinase delta |
| EP2223922B1 (en) * | 2000-04-25 | 2016-03-02 | ICOS Corporation | Inhibitors of human phosphatidyl-inositol 3-kinase delta |
| AUPR201600A0 (en) * | 2000-12-11 | 2001-01-11 | Fujisawa Pharmaceutical Co., Ltd. | Quinazolinone derivative |
| EP2329822A1 (en) | 2001-09-05 | 2011-06-08 | Minerva Biotechnologies Corporation | Compositions and methods of treatment of cancer |
| CA2459584A1 (en) * | 2001-09-05 | 2003-03-13 | Cynthia C. Bamdad | Compositions and use thereof in the treatment of cancer |
| WO2003039460A2 (en) * | 2001-11-07 | 2003-05-15 | Merck & Co., Inc. | Mitotic kinesin inhibitors |
| AUPS019702A0 (en) * | 2002-01-29 | 2002-02-21 | Fujisawa Pharmaceutical Co., Ltd. | Condensed heterocyclic compounds |
| EP1539180A4 (en) * | 2002-08-21 | 2006-08-30 | Cytokinetics Inc | COMPOUNDS, COMPOSITIONS AND METHODS |
| US20060052345A1 (en) * | 2002-11-04 | 2006-03-09 | Nps Pharmaceuticals, Inc. | Quinazolinone compounds as calcilytics |
| ATE440825T1 (de) * | 2003-06-06 | 2009-09-15 | Vertex Pharma | Pyrimidin-derivate zur verwendung als modulatoren von atp-bindende kassette transportern |
| WO2005016349A1 (en) * | 2003-08-14 | 2005-02-24 | Icos Corporation | Methods of inhibiting leukocyte accumulation |
| US20050043239A1 (en) * | 2003-08-14 | 2005-02-24 | Jason Douangpanya | Methods of inhibiting immune responses stimulated by an endogenous factor |
| WO2005113554A2 (en) * | 2004-05-13 | 2005-12-01 | Icos Corporation | Method of preparing 3-phenyl-2-[9h-purin-6-ylamino)-methyl]-3h-quinazolin-4-one and substituted and related compounds |
| WO2005117889A1 (en) * | 2004-05-25 | 2005-12-15 | Icos Corporation | Methods for treating and/or preventing aberrant proliferation of hematopoietic |
| US20080287469A1 (en) * | 2005-02-17 | 2008-11-20 | Diacovo Thomas G | Phosphoinositide 3-Kinase Inhibitors for Inhibiting Leukocyte Accumulation |
| EP2233472B1 (en) * | 2006-03-28 | 2014-01-15 | Atir Holding S.A. | Heterocyclic compounds and uses thereof in the treatment of sexual disorders |
| SG195655A1 (en) | 2008-11-13 | 2013-12-30 | Gilead Calistoga Llc | Therapies for hematologic malignancies |
| US9492449B2 (en) | 2008-11-13 | 2016-11-15 | Gilead Calistoga Llc | Therapies for hematologic malignancies |
| CN102439012A (zh) | 2009-03-24 | 2012-05-02 | 吉里德卡利斯托加公司 | 2-嘌呤基-3-甲苯基-喹唑啉酮衍生物的阻转异构体和使用方法 |
| AP2011005956A0 (en) * | 2009-04-20 | 2011-10-31 | Gilead Calistoga Llc | Methods of treatment for solid tumors. |
| CA2768843A1 (en) | 2009-07-21 | 2011-01-27 | Gilead Calistoga Llc | Treatment of liver disorders with pi3k inhibitors |
| BRPI1003506B1 (pt) | 2010-09-24 | 2019-12-03 | Ache Int Bvi Ltd | composto alquil-piperazino-fenil-4(3h)quinazolinonas e uso do composto alquil-piperazino-fenil-4(3h)quinazolinonas associado aos receptores serotoninérgicos 5-ht1a e 5-ht2a |
| EP2697206B1 (en) | 2011-04-10 | 2019-04-03 | Atir Holding S.A. | Heterocyclic compounds and uses thereof in the treatment of sexual disorders |
| PL2834241T3 (pl) | 2012-03-05 | 2021-07-12 | Gilead Calistoga Llc | Formy polimorficzne (s)-2-(1-(9h-puryn-6-yloamino)propylo)-5-fluoro-3-fenylochinazolin-4(3h)-onu |
| WO2014009872A1 (en) | 2012-07-09 | 2014-01-16 | Lupin Limited | Tetrahydroquinazolinone derivatives as parp inhibitors |
| JP2017500319A (ja) | 2013-12-20 | 2017-01-05 | ギリアード カリストガ エルエルシー | （ｓ）−２−（１−（９ｈ−プリン−６−イルアミノ）プロピル）−５−フルオロ−３−フェニルキナゾリン−４（３ｈ）−オンの塩酸塩の多形形態 |
| CA2934531C (en) | 2013-12-20 | 2020-02-25 | Gilead Calistoga Llc | Process methods for phosphatidylinositol 3-kinase inhibitors |
| WO2015191726A1 (en) | 2014-06-13 | 2015-12-17 | Gilead Sciences, Inc. | Phosphatidylinositol 3-kinase inhibitors |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1053063A (OSRAM) * | 1963-05-18 |
-
1970
- 1970-06-05 DE DE19702027645 patent/DE2027645A1/de active Pending
-
1971
- 1971-05-28 US US05/148,100 patent/US3984555A/en not_active Expired - Lifetime
- 1971-06-01 AT AT244173A patent/AT318628B/de not_active IP Right Cessation
- 1971-06-01 AT AT470571A patent/AT318615B/de not_active IP Right Cessation
- 1971-06-01 AT AT244273A patent/AT317899B/de not_active IP Right Cessation
- 1971-06-02 LU LU63267D patent/LU63267A1/xx unknown
- 1971-06-02 CH CH802071A patent/CH557829A/xx not_active IP Right Cessation
- 1971-06-02 CH CH450074A patent/CH558374A/xx not_active IP Right Cessation
- 1971-06-02 CH CH450174A patent/CH569732A5/xx not_active IP Right Cessation
- 1971-06-03 GB GB1880371*[A patent/GB1331522A/en not_active Expired
- 1971-06-03 CA CA114,709,A patent/CA951319A/en not_active Expired
- 1971-06-04 FR FR7120368A patent/FR2100726B1/fr not_active Expired
- 1971-06-04 BE BE768137A patent/BE768137A/xx unknown
- 1971-06-04 NL NL7107695A patent/NL7107695A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CH557829A (de) | 1975-01-15 |
| NL7107695A (OSRAM) | 1971-12-07 |
| AT317899B (de) | 1974-09-25 |
| AT318628B (de) | 1974-11-11 |
| BE768137A (fr) | 1971-12-06 |
| AT318615B (de) | 1974-11-11 |
| DE2027645A1 (de) | 1971-12-09 |
| FR2100726A1 (OSRAM) | 1972-03-24 |
| LU63267A1 (OSRAM) | 1972-08-23 |
| GB1331522A (en) | 1973-09-26 |
| CA951319A (en) | 1974-07-16 |
| US3984555A (en) | 1976-10-05 |
| FR2100726B1 (OSRAM) | 1975-10-10 |
| CH569732A5 (OSRAM) | 1975-11-28 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CH558374A (de) | Verfahren zur herstellung von arylsubstituierten piperazinylalkyl- bezw. alkenyl- chinazolon-(4)-derivaten. | |
| CH552607A (de) | Verfahren zur herstellung von azaspiroalkandion-derivaten. | |
| AT289065B (de) | Verfahren zur Herstellung von 2,3,6-Trimethylphenol | |
| CH547290A (de) | Verfahren zur herstellung von nitro-imidazolderivaten. | |
| CH557823A (de) | Verfahren zur herstellung von piperazinderivaten. | |
| CH550771A (de) | Verfahren zur herstellung von phenaethylaminderivaten. | |
| CH558353A (de) | Verfahren zur herstellung von isoindolinderivaten. | |
| CH550186A (de) | Verfahren zur herstellung von 5-imino-1.2.4-triazin-derivaten. | |
| CH550133A (de) | Verfahren zur herstellung von 4-methyl-pentanol-2-crotonat. | |
| CH555801A (de) | Verfahren zur herstellung von phenylaethanolamin-derivaten. | |
| CH550797A (de) | Verfahren zur herstellung von tetrahydroisochinolinderivaten. | |
| CH551984A (de) | Verfahren zur herstellung von piperazinderivaten. | |
| CH550214A (de) | Verfahren zur herstellung von cyclocopolymerisaten. | |
| CH553185A (de) | Verfahren zur herstellung von lumilysergol-derivaten. | |
| CH549567A (de) | Verfahren zur herstellung von 8-cyano-5-octanolid. | |
| CH558800A (de) | Verfahren zur herstellung von chinazolinonen. | |
| CH547775A (de) | Verfahren zur herstellung von diaethylaminopropionaniliden. | |
| CH557830A (de) | Verfahren zur herstellung von 1-aminosiochinolinen. | |
| CH547802A (de) | Verfahren zur herstellung von tetrahydropyridinderivaten. | |
| CH550809A (de) | Verfahren zur herstellung von triazol-derivaten. | |
| CH555314A (de) | Verfahren zur herstellung von cyclopropylmethylalkylaminen. | |
| CH546782A (de) | Verfahren zur herstellung von oxadiazolderivaten. | |
| CH557801A (de) | Verfahren zur herstellung von 1,1,3-trialkoxy-2-cyanopropanen. | |
| CH537891A (de) | Verfahren zur Herstellung von 2,3,6-Trimethylphenol | |
| CH547771A (de) | Verfahren zur herstellung von bornanaminderivaten. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PL | Patent ceased |