CH554858A - Verfahren zur herstellung von methyl-n-acetal-6,7-aziridino-6-desamino-7-desoxy-(alpha)-thiolincosamidinen. - Google Patents

Verfahren zur herstellung von methyl-n-acetal-6,7-aziridino-6-desamino-7-desoxy-(alpha)-thiolincosamidinen.

Info

Publication number
CH554858A
CH554858A CH854674A CH854674A CH554858A CH 554858 A CH554858 A CH 554858A CH 854674 A CH854674 A CH 854674A CH 854674 A CH854674 A CH 854674A CH 554858 A CH554858 A CH 554858A
Authority
CH
Switzerland
Prior art keywords
thiolincosamidines
desamino
aziridino
desoxy
acetal
Prior art date
Application number
CH854674A
Other languages
German (de)
English (en)
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of CH554858A publication Critical patent/CH554858A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08G—MACROMOLECULAR COMPOUNDS OBTAINED OTHERWISE THAN BY REACTIONS ONLY INVOLVING UNSATURATED CARBON-TO-CARBON BONDS
    • C08G18/00—Polymeric products of isocyanates or isothiocyanates
    • C08G18/06—Polymeric products of isocyanates or isothiocyanates with compounds having active hydrogen
    • C08G18/28—Polymeric products of isocyanates or isothiocyanates with compounds having active hydrogen characterised by the compounds used containing active hydrogen
    • C08G18/30—Low-molecular-weight compounds
    • C08G18/38—Low-molecular-weight compounds having heteroatoms other than oxygen
    • C08G18/3855—Low-molecular-weight compounds having heteroatoms other than oxygen having sulfur
    • C08G18/3863—Low-molecular-weight compounds having heteroatoms other than oxygen having sulfur containing groups having sulfur atoms between two carbon atoms, the sulfur atoms being directly linked to carbon atoms or other sulfur atoms
    • C08G18/3865—Low-molecular-weight compounds having heteroatoms other than oxygen having sulfur containing groups having sulfur atoms between two carbon atoms, the sulfur atoms being directly linked to carbon atoms or other sulfur atoms containing groups having one sulfur atom between two carbon atoms
    • C08G18/3868—Low-molecular-weight compounds having heteroatoms other than oxygen having sulfur containing groups having sulfur atoms between two carbon atoms, the sulfur atoms being directly linked to carbon atoms or other sulfur atoms containing groups having one sulfur atom between two carbon atoms the sulfur atom belonging to a sulfide group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
    • C07H15/16—Lincomycin; Derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Polymers & Plastics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Cephalosporin Compounds (AREA)
CH854674A 1970-04-06 1971-03-19 Verfahren zur herstellung von methyl-n-acetal-6,7-aziridino-6-desamino-7-desoxy-(alpha)-thiolincosamidinen. CH554858A (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2611970A 1970-04-06 1970-04-06

Publications (1)

Publication Number Publication Date
CH554858A true CH554858A (de) 1974-10-15

Family

ID=21830031

Family Applications (2)

Application Number Title Priority Date Filing Date
CH854674A CH554858A (de) 1970-04-06 1971-03-19 Verfahren zur herstellung von methyl-n-acetal-6,7-aziridino-6-desamino-7-desoxy-(alpha)-thiolincosamidinen.
CH405671A CH556325A (de) 1970-04-06 1971-03-19 Verfahren zur herstellung von alkyl-7-desoxy-7(s)-or-(alpha)-thiolincosaminiden.

Family Applications After (1)

Application Number Title Priority Date Filing Date
CH405671A CH556325A (de) 1970-04-06 1971-03-19 Verfahren zur herstellung von alkyl-7-desoxy-7(s)-or-(alpha)-thiolincosaminiden.

Country Status (14)

Country Link
US (1) US3702322A (nl)
JP (1) JPS5527071B1 (nl)
BE (1) BE765370A (nl)
CA (1) CA945149A (nl)
CH (2) CH554858A (nl)
DE (4) DE2167180C3 (nl)
DK (1) DK134489B (nl)
ES (1) ES389524A1 (nl)
FR (1) FR2092009B1 (nl)
GB (1) GB1311438A (nl)
IL (1) IL36435A (nl)
NL (1) NL170960C (nl)
SE (2) SE385011B (nl)
ZA (1) ZA711709B (nl)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3853843A (en) * 1972-12-13 1974-12-10 Upjohn Co Derivatives of thiolincosaminide compounds
US3870699A (en) * 1973-03-06 1975-03-11 Upjohn Co Lincomycin analogs
WO2003020736A1 (en) * 2001-08-28 2003-03-13 Pharmacia Corporation Crystaline clindamycin free base
US7199105B2 (en) * 2002-08-15 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
CA2493799A1 (en) * 2002-08-15 2004-02-26 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
US7256177B2 (en) 2003-06-17 2007-08-14 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
US7199106B2 (en) 2003-06-17 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antimicrobial activity
US7361743B2 (en) * 2004-02-11 2008-04-22 Pfizer Inc Lincomycin derivatives possessing antibacterial activity

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1467501A (fr) * 1965-10-20 1967-01-27 Upjohn Co 7-halogéno-7-deoxylincomycine et 7-halogéno-7-dexoyepilincomycine, leurs analogues et isomères et leurs procédés de fabrication

Also Published As

Publication number Publication date
FR2092009A1 (nl) 1972-01-21
NL7104221A (nl) 1971-10-08
IL36435A0 (en) 1971-05-26
BE765370A (fr) 1971-10-06
NL170960B (nl) 1982-08-16
DE2116066B2 (de) 1980-01-17
DE2167180C3 (de) 1981-07-30
CA945149A (en) 1974-04-09
SE385011B (sv) 1976-05-31
CH556325A (de) 1974-11-29
DE2116066C3 (de) 1980-11-13
GB1311438A (en) 1973-03-28
DE2167181C3 (de) 1981-07-02
DE2116066A1 (de) 1971-11-04
FR2092009B1 (nl) 1974-09-27
SE409209B (sv) 1979-08-06
NL170960C (nl) 1983-01-17
ZA711709B (en) 1972-01-26
ES389524A1 (es) 1974-03-16
DE2167182B1 (de) 1981-01-08
DK134489C (nl) 1977-04-25
DK134489B (da) 1976-11-15
DE2167181B1 (de) 1980-11-27
JPS5527071B1 (nl) 1980-07-17
IL36435A (en) 1975-04-25
DE2167182C3 (de) 1981-09-17
US3702322A (en) 1972-11-07
DE2167180B1 (de) 1980-12-18

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Legal Events

Date Code Title Description
PL Patent ceased