CA3142992A1 - Heteroaromatic inhibitors of astacin proteinases - Google Patents

Heteroaromatic inhibitors of astacin proteinases Download PDF

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Publication number
CA3142992A1
CA3142992A1 CA3142992A CA3142992A CA3142992A1 CA 3142992 A1 CA3142992 A1 CA 3142992A1 CA 3142992 A CA3142992 A CA 3142992A CA 3142992 A CA3142992 A CA 3142992A CA 3142992 A1 CA3142992 A1 CA 3142992A1
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Canada
Prior art keywords
alkyl
independently selected
group
carboxy
aryl
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CA3142992A
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English (en)
French (fr)
Inventor
Daniel Ramsbeck
Kathrin Tan
Dagmar Schlenzig
Mirko Buchholz
Holger Cynis
Stephan Schilling
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Vivoryon Therapeutics NV
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Vivoryon Therapeutics NV
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Priority to CA3300715A priority Critical patent/CA3300715A1/en
Publication of CA3142992A1 publication Critical patent/CA3142992A1/en
Pending legal-status Critical Current

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    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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CA3300715A1 (en) 2026-03-02
EP3750878A1 (en) 2020-12-16
EP3750878B1 (en) 2025-05-14
KR102930913B1 (ko) 2026-02-27
BR112021024327A2 (pt) 2022-01-11
EP3750878C0 (en) 2025-05-14
KR20260036022A (ko) 2026-03-13
CN114585608B (zh) 2026-03-17
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