ZA202109419B - Heteroaromatic inhibitors of astacin proteinases - Google Patents

Heteroaromatic inhibitors of astacin proteinases

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Publication number
ZA202109419B
ZA202109419B ZA2021/09419A ZA202109419A ZA202109419B ZA 202109419 B ZA202109419 B ZA 202109419B ZA 2021/09419 A ZA2021/09419 A ZA 2021/09419A ZA 202109419 A ZA202109419 A ZA 202109419A ZA 202109419 B ZA202109419 B ZA 202109419B
Authority
ZA
South Africa
Prior art keywords
astacin
proteinases
heteroaromatic
inhibitors
heteroaromatic inhibitors
Prior art date
Application number
ZA2021/09419A
Other languages
English (en)
Inventor
Daniel Ramsbeck
Kathrin Tan
Dagmar Schlenzig
Mirko Buchholz
Holger Cynis
Stephan Schilling
Original Assignee
Vivoryon Therapeutics N V
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vivoryon Therapeutics N V filed Critical Vivoryon Therapeutics N V
Publication of ZA202109419B publication Critical patent/ZA202109419B/en

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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
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