CA3120866A1 - Tyk2 inhibitors and uses thereof - Google Patents

Tyk2 inhibitors and uses thereof Download PDF

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Publication number
CA3120866A1
CA3120866A1 CA3120866A CA3120866A CA3120866A1 CA 3120866 A1 CA3120866 A1 CA 3120866A1 CA 3120866 A CA3120866 A CA 3120866A CA 3120866 A CA3120866 A CA 3120866A CA 3120866 A1 CA3120866 A1 CA 3120866A1
Authority
CA
Canada
Prior art keywords
nitrogen
compound
sulfur
oxygen
independently selected
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CA3120866A
Other languages
English (en)
French (fr)
Inventor
Jeremy Robert Greenwood
Craig E. Masse
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Takeda Pharmaceutical Co Ltd
Original Assignee
Nimbus Lakshmi Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nimbus Lakshmi Inc filed Critical Nimbus Lakshmi Inc
Publication of CA3120866A1 publication Critical patent/CA3120866A1/en
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CA3120866A 2018-11-30 2019-11-27 Tyk2 inhibitors and uses thereof Pending CA3120866A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862773620P 2018-11-30 2018-11-30
US62/773,620 2018-11-30
PCT/US2019/063510 WO2020112937A1 (en) 2018-11-30 2019-11-27 Tyk2 inhibitors and uses thereof

Publications (1)

Publication Number Publication Date
CA3120866A1 true CA3120866A1 (en) 2020-06-04

Family

ID=70848642

Family Applications (1)

Application Number Title Priority Date Filing Date
CA3120866A Pending CA3120866A1 (en) 2018-11-30 2019-11-27 Tyk2 inhibitors and uses thereof

Country Status (8)

Country Link
US (2) US11053241B2 (enExample)
EP (1) EP3886843A4 (enExample)
JP (2) JP7530360B2 (enExample)
CN (1) CN113271938A (enExample)
AU (1) AU2019389025B2 (enExample)
CA (1) CA3120866A1 (enExample)
IL (1) IL283409A (enExample)
WO (1) WO2020112937A1 (enExample)

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JP7530360B2 (ja) 2018-11-30 2024-08-07 武田薬品工業株式会社 Ｔｙｋ２阻害剤およびその使用
US20240067633A1 (en) * 2020-12-25 2024-02-29 Sichuan Haisco Pharmaceutical Co., Ltd. Ketohexokinase inhibitor and use thereof
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Also Published As

Publication number Publication date
US20220106306A1 (en) 2022-04-07
AU2019389025B2 (en) 2025-07-24
CN113271938A (zh) 2021-08-17
JP2024160253A (ja) 2024-11-13
US11834449B2 (en) 2023-12-05
EP3886843A4 (en) 2022-08-31
EP3886843A1 (en) 2021-10-06
JP7530360B2 (ja) 2024-08-07
US11053241B2 (en) 2021-07-06
WO2020112937A1 (en) 2020-06-04
IL283409A (en) 2021-07-29
US20200172540A1 (en) 2020-06-04
AU2019389025A1 (en) 2021-06-17
JP2022509260A (ja) 2022-01-20

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Effective date: 20231127