CA3061611A1 - Modulators of sestrin-gator2 interaction and uses thereof - Google Patents

Modulators of sestrin-gator2 interaction and uses thereof Download PDF

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Publication number
CA3061611A1
CA3061611A1 CA3061611A CA3061611A CA3061611A1 CA 3061611 A1 CA3061611 A1 CA 3061611A1 CA 3061611 A CA3061611 A CA 3061611A CA 3061611 A CA3061611 A CA 3061611A CA 3061611 A1 CA3061611 A1 CA 3061611A1
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mmol
acid
solution
ring
amino
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CA3061611A
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English (en)
French (fr)
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Eddine Saiah
George Vlasuk
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Navitor Pharmaceuticals Inc
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Publication of CA3061611A1 publication Critical patent/CA3061611A1/en
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    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyridine Compounds (AREA)
  • Steroid Compounds (AREA)
  • Crystals, And After-Treatments Of Crystals (AREA)
  • Optical Modulation, Optical Deflection, Nonlinear Optics, Optical Demodulation, Optical Logic Elements (AREA)
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CA3061611A 2017-04-26 2018-04-25 Modulators of sestrin-gator2 interaction and uses thereof Pending CA3061611A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762490280P 2017-04-26 2017-04-26
US62/490,280 2017-04-26
PCT/US2018/029288 WO2018200625A1 (en) 2017-04-26 2018-04-25 Modulators of sestrin-gator2 interaction and uses thereof

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US (4) US10912750B2 (https=)
EP (2) EP4556069A3 (https=)
JP (1) JP7179015B2 (https=)
CN (2) CN110809467B (https=)
AU (2) AU2018258355B2 (https=)
CA (1) CA3061611A1 (https=)
ES (1) ES3040534T3 (https=)
PL (1) PL3615019T3 (https=)
TW (1) TWI776886B (https=)
WO (1) WO2018200625A1 (https=)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2016342027B2 (en) 2015-10-23 2021-05-13 Navitor Pharmaceuticals, Inc. Modulators of Sestrin-GATOR2 interaction and uses thereof
PL3615019T3 (pl) 2017-04-26 2026-01-19 Navitor Pharmaceuticals, Inc. Modulator interakcji sestryna-gator2 do zastosowania w leczeniu depresji opornej na leczenie
EP3870158A4 (en) 2018-10-24 2022-08-10 Navitor Pharmaceuticals, Inc. Polymorphic compounds and uses thereof
JP7189368B2 (ja) 2018-10-30 2022-12-13 ギリアード サイエンシーズ, インコーポレイテッド アルファ4ベータ7インテグリンの阻害のための化合物
FI3873884T3 (fi) 2018-10-30 2025-02-24 Gilead Sciences Inc 3-(kinolin-8-yyli)-1,4-dihydropyrido[3,4-d]pyrimidiini-2,4-dionijohdannaisia alfa-4-beta-7-integriinin estäjinä tulehdussairauksien hoidossa
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