CA2977367A1 - Methods and compositions for decreasing gastric emptying - Google Patents
Methods and compositions for decreasing gastric emptying Download PDFInfo
- Publication number
- CA2977367A1 CA2977367A1 CA2977367A CA2977367A CA2977367A1 CA 2977367 A1 CA2977367 A1 CA 2977367A1 CA 2977367 A CA2977367 A CA 2977367A CA 2977367 A CA2977367 A CA 2977367A CA 2977367 A1 CA2977367 A1 CA 2977367A1
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- alkyl
- group
- agent
- optionally substituted
- treating
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| CN103429571A (zh) | 2010-12-22 | 2013-12-04 | 普渡制药公司 | 作为钠通道阻断剂的取代吡啶 |
| WO2013030665A1 (en) | 2011-09-02 | 2013-03-07 | Purdue Pharma L.P. | Pyrimidines as sodium channel blockers |
| WO2014096941A1 (en) | 2012-12-20 | 2014-06-26 | Purdue Pharma L.P. | Cyclic sulfonamides as sodium channel blockers |
| US9120786B2 (en) | 2013-03-04 | 2015-09-01 | Purdue Pharma, L.P. | Triazine carboxamides as sodium channel blockers |
| CN105073728A (zh) | 2013-03-15 | 2015-11-18 | 全球血液疗法股份有限公司 | 化合物及其用于调节血红蛋白的用途 |
| WO2015031036A1 (en) | 2013-08-26 | 2015-03-05 | Purdue Pharma L.P. | Azaspiro[4.5] decane derivatives and use thereof |
| US9828348B2 (en) | 2013-11-08 | 2017-11-28 | Purdue Pharma L.P. | Benzimidazole derivatives and use thereof |
| EA201992707A1 (ru) | 2013-11-18 | 2020-06-30 | Глобал Блад Терапьютикс, Инк. | Соединения и их применения для модуляции гемоглобина |
| AU2014370407B2 (en) | 2013-12-23 | 2018-03-29 | Purdue Pharma L.P. | Indazoles and use thereof |
| US9994571B2 (en) | 2013-12-26 | 2018-06-12 | Purdue Pharma L.P. | 10-substituted morphinan hydantoins |
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| CN107613965A (zh) * | 2015-02-19 | 2018-01-19 | 普渡制药公司 | 用于减少胃排空的方法和组合物 |
| CN106397426A (zh) * | 2016-03-29 | 2017-02-15 | 广东环境保护工程职业学院 | 一种1，3，4-噻二唑类化合物及其制备方法 |
| US12605388B2 (en) | 2024-09-25 | 2026-04-21 | Azurity Pharmaceuticals Ireland Limited | Lamotrigine salts, co-crystals, and compositions |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
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| MXPA04000411A (es) | 2001-07-16 | 2004-03-18 | Euro Celtique Sa | Tiazolidinonas arilo sustituidas y uso de las mismas. |
| AR036873A1 (es) | 2001-09-07 | 2004-10-13 | Euro Celtique Sa | Piridinas aril sustituidas a, composiciones farmaceuticas y el uso de las mismas para la preparacion de un medicamento |
| DK1483247T3 (da) | 2002-03-13 | 2009-08-17 | Euro Celtique Sa | Arylsubstituerede pyrimidiner og anvendelsen deraf |
| JP2006504660A (ja) | 2002-07-31 | 2006-02-09 | ユーロ−セルティーク エス．エイ． | アリール置換ベンゾイミダゾール類およびナトリウムチャネルブロッカーとしてのそれらの使用 |
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| EP1533298A1 (en) * | 2003-11-21 | 2005-05-25 | Newron Pharmaceuticals S.p.A. | 3-aminopyrrolidone derivatives |
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| US20070020194A1 (en) * | 2005-06-08 | 2007-01-25 | Greenway Frank L Iii | Nasally administered appetite suppressant |
| WO2007083239A1 (en) | 2006-01-23 | 2007-07-26 | Pfizer Limited | Pyridine derivatives as sodium channel modulators |
| JPWO2008044770A1 (ja) * | 2006-10-13 | 2010-02-18 | 味の素株式会社 | ４−ヒドロキシイソロイシンを含む胃排出抑制剤 |
| CN101553256B (zh) | 2006-11-01 | 2013-01-30 | 普渡制药公司 | 苯基丙酰胺化合物及其用途 |
| CA2693588C (en) | 2007-07-13 | 2015-11-17 | Icagen, Inc. | Sodium channel inhibitors |
| US8853250B2 (en) | 2007-07-13 | 2014-10-07 | Icagen, Inc. | Sodium channel inhibitors |
| JP2013530180A (ja) | 2010-06-16 | 2013-07-25 | パーデュー、ファーマ、リミテッド、パートナーシップ | アリール置換インドールおよびその使用 |
| WO2012004664A2 (en) | 2010-07-07 | 2012-01-12 | Purdue Pharma L.P. | Analogs of sodium channel peptide toxin |
| JP2013531687A (ja) | 2010-07-16 | 2013-08-08 | パーデュー、ファーマ、リミテッド、パートナーシップ | ナトリウムチャネル遮断剤としてのピリジン化合物 |
| EP2616441B1 (en) | 2010-09-17 | 2019-08-07 | Purdue Pharma L.P. | Pyridine compounds and the uses thereof |
| EP2625169B1 (en) | 2010-10-05 | 2015-03-25 | Purdue Pharma L.P. | Quinazoline compounds as sodium channel blockers |
| CN103429571A (zh) | 2010-12-22 | 2013-12-04 | 普渡制药公司 | 作为钠通道阻断剂的取代吡啶 |
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| EA023375B1 (ru) | 2011-10-26 | 2016-05-31 | Пфайзер Лимитед | Производные (4-фенилимидазол-2-ил)этиламина в качестве модуляторов натриевых каналов |
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| WO2013136170A1 (en) | 2012-03-16 | 2013-09-19 | Purdue Pharma L.P. | Substituted pyridines as sodium channel blockers |
| WO2014016673A1 (en) | 2012-07-27 | 2014-01-30 | Purdue Pharma L.P. | Sodium channel blocking peptides and the use thereof |
| US9637458B2 (en) | 2013-03-04 | 2017-05-02 | Jeffrey Lockman | Pyrimidine carboxamides as sodium channel blockers |
| CA3082427A1 (en) | 2013-03-15 | 2014-09-25 | Purdue Pharma L.P. | Carboxamide derivatives and use thereof |
| CN107613965A (zh) * | 2015-02-19 | 2018-01-19 | 普渡制药公司 | 用于减少胃排空的方法和组合物 |
-
2016
- 2016-02-19 CN CN201680021578.2A patent/CN107613965A/zh active Pending
- 2016-02-19 EP EP16753165.6A patent/EP3258925B1/en active Active
- 2016-02-19 MX MX2017010682A patent/MX2017010682A/es unknown
- 2016-02-19 KR KR1020177025621A patent/KR20170117170A/ko not_active Withdrawn
- 2016-02-19 BR BR112017017619A patent/BR112017017619A2/pt not_active Application Discontinuation
- 2016-02-19 WO PCT/US2016/018715 patent/WO2016134283A1/en not_active Ceased
- 2016-02-19 CA CA2977367A patent/CA2977367A1/en not_active Abandoned
- 2016-02-19 US US15/048,530 patent/US9763955B2/en active Active
- 2016-02-19 JP JP2017543916A patent/JP6762308B2/ja active Active
- 2016-02-19 AU AU2016219879A patent/AU2016219879A1/en not_active Abandoned
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- 2017-08-10 IL IL253949A patent/IL253949A0/en unknown
- 2017-08-18 US US15/680,737 patent/US10143696B2/en active Active
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| US10143696B2 (en) | 2018-12-04 |
| JP6762308B2 (ja) | 2020-09-30 |
| PH12017501393A1 (en) | 2018-01-08 |
| EP3258925B1 (en) | 2023-03-29 |
| US9763955B2 (en) | 2017-09-19 |
| US20160243129A1 (en) | 2016-08-25 |
| JP2018509397A (ja) | 2018-04-05 |
| EP3258925A4 (en) | 2019-01-09 |
| WO2016134283A1 (en) | 2016-08-25 |
| US20170340646A1 (en) | 2017-11-30 |
| KR20170117170A (ko) | 2017-10-20 |
| EP3258925A1 (en) | 2017-12-27 |
| MX2017010682A (es) | 2018-04-24 |
| CN107613965A (zh) | 2018-01-19 |
| BR112017017619A2 (pt) | 2018-05-08 |
| IL253949A0 (en) | 2017-10-31 |
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| EEER | Examination request |
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| FZDE | Discontinued |
Effective date: 20191206 |