CA2977367A1 - Methods and compositions for decreasing gastric emptying - Google Patents
Methods and compositions for decreasing gastric emptying Download PDFInfo
- Publication number
- CA2977367A1 CA2977367A1 CA2977367A CA2977367A CA2977367A1 CA 2977367 A1 CA2977367 A1 CA 2977367A1 CA 2977367 A CA2977367 A CA 2977367A CA 2977367 A CA2977367 A CA 2977367A CA 2977367 A1 CA2977367 A1 CA 2977367A1
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- alkyl
- group
- agent
- optionally substituted
- treating
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| EP3255041A1 (en) | 2011-09-02 | 2017-12-13 | Purdue Pharma L.P. | Pyrimidines as sodium channel blockers |
| EP2935257B1 (en) | 2012-12-20 | 2018-02-07 | Purdue Pharma LP | Cyclic sulfonamides as sodium channel blockers |
| US9120786B2 (en) | 2013-03-04 | 2015-09-01 | Purdue Pharma, L.P. | Triazine carboxamides as sodium channel blockers |
| SG10201802911RA (en) | 2013-03-15 | 2018-05-30 | Global Blood Therapeutics Inc | Compounds and uses thereof for the modulation of hemoglobin |
| CN105612152A (zh) | 2013-08-26 | 2016-05-25 | 普渡制药公司 | 氮杂螺[4.5]癸烷衍生物及其用途 |
| US9828348B2 (en) | 2013-11-08 | 2017-11-28 | Purdue Pharma L.P. | Benzimidazole derivatives and use thereof |
| EA202092627A1 (ru) | 2013-11-18 | 2021-09-30 | Глобал Блад Терапьютикс, Инк. | Соединения и их применения для модуляции гемоглобина |
| JP6337124B2 (ja) | 2013-12-23 | 2018-06-06 | パーデュー、ファーマ、リミテッド、パートナーシップ | インダゾール及びその使用 |
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| JP6526023B2 (ja) | 2014-01-24 | 2019-06-05 | パーデュー、ファーマ、リミテッド、パートナーシップ | ピリジン類及びピリミジン類並びにその使用 |
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| IL159765A0 (en) | 2001-07-16 | 2004-06-20 | Euro Celtique Sa | Aryl substituted thiazolidinone derivatives and pharmaceutical compositions containing the same |
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| CA2492305A1 (en) | 2002-07-31 | 2004-02-05 | Euro-Celtique S.A. | Aryl substituted benzimidazoles and their use as sodium channel blockers |
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| EP1533298A1 (en) * | 2003-11-21 | 2005-05-25 | Newron Pharmaceuticals S.p.A. | 3-aminopyrrolidone derivatives |
| JP2008528510A (ja) | 2005-01-20 | 2008-07-31 | サートリス ファーマシューティカルズ， インコーポレイテッド | 紅潮および／または薬物誘発性体重増加を処置するためのサーチュイン活性化化合物の使用 |
| US20070020194A1 (en) * | 2005-06-08 | 2007-01-25 | Greenway Frank L Iii | Nasally administered appetite suppressant |
| WO2007083239A1 (en) | 2006-01-23 | 2007-07-26 | Pfizer Limited | Pyridine derivatives as sodium channel modulators |
| WO2008044770A1 (en) * | 2006-10-13 | 2008-04-17 | Ajinomoto Co., Inc. | Agent for suppression of gastric emptying comprising 4-hydroxyisoleucine |
| ES2433118T3 (es) | 2006-11-01 | 2013-12-09 | Purdue Pharma Lp | Compuestos de fenilpropionamida y uso de los mismos |
| WO2009012241A1 (en) | 2007-07-13 | 2009-01-22 | Icagen, Inc. | Sodium channel inhibitors |
| US8124610B2 (en) | 2007-07-13 | 2012-02-28 | Icagen Inc. | Sodium channel inhibitors |
| EP2582666B1 (en) | 2010-06-16 | 2014-08-13 | Purdue Pharma L.P. | Aryl substituted indoles and their use as blockers of sodium channels |
| US9279003B2 (en) | 2010-07-07 | 2016-03-08 | Purdue Pharma L.P. | Analogs of sodium channel peptide toxin |
| JP2013531687A (ja) | 2010-07-16 | 2013-08-08 | パーデュー、ファーマ、リミテッド、パートナーシップ | ナトリウムチャネル遮断剤としてのピリジン化合物 |
| AU2011303597A1 (en) | 2010-09-17 | 2013-04-11 | Purdue Pharma L.P. | Pyridine compounds and the uses thereof |
| KR20130095772A (ko) | 2010-10-05 | 2013-08-28 | 퍼듀 퍼머 엘피 | 나트륨 채널 차단제로서 퀴나졸린 화합물 |
| EP2655330B1 (en) | 2010-12-22 | 2016-02-10 | Purdue Pharma LP | Substituted pyridines as sodium channel blockers |
| EP3255041A1 (en) | 2011-09-02 | 2017-12-13 | Purdue Pharma L.P. | Pyrimidines as sodium channel blockers |
| CA2850925C (en) | 2011-10-26 | 2017-01-10 | Pfizer Limited | (4-phenylimidazol-2-yl) ethylamine derivatives useful as sodium channel modulators |
| WO2013064884A1 (en) | 2011-10-31 | 2013-05-10 | Purdue Pharma L.P. | Quaternized amines as sodium channel blockers |
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| JP5938219B2 (ja) * | 2012-01-23 | 2016-06-22 | 株式会社明治 | 胃排出遅延のための食品用の剤または医療用の剤 |
| WO2013136170A1 (en) | 2012-03-16 | 2013-09-19 | Purdue Pharma L.P. | Substituted pyridines as sodium channel blockers |
| US9718865B2 (en) | 2012-07-27 | 2017-08-01 | Purdue Pharma L.P. | Sodium channel blocking peptides and the use thereof |
| WO2014135955A1 (en) * | 2013-03-04 | 2014-09-12 | Purdue Pharma L.P. | Pyrimidine carboxamides as sodium channel blockers |
| CA2939549C (en) | 2013-03-15 | 2020-08-18 | Purdue Pharma L.P. | Carboxamide derivatives and use thereof |
| BR112017017619A2 (pt) * | 2015-02-19 | 2018-05-08 | Purdue Pharma Lp | métodos e composições para diminuir esvaziamento gástrico |
-
2016
- 2016-02-19 BR BR112017017619A patent/BR112017017619A2/pt not_active Application Discontinuation
- 2016-02-19 EP EP16753165.6A patent/EP3258925B1/en active Active
- 2016-02-19 JP JP2017543916A patent/JP6762308B2/ja active Active
- 2016-02-19 US US15/048,530 patent/US9763955B2/en active Active
- 2016-02-19 AU AU2016219879A patent/AU2016219879A1/en not_active Abandoned
- 2016-02-19 WO PCT/US2016/018715 patent/WO2016134283A1/en not_active Ceased
- 2016-02-19 MX MX2017010682A patent/MX2017010682A/es unknown
- 2016-02-19 KR KR1020177025621A patent/KR20170117170A/ko not_active Withdrawn
- 2016-02-19 CN CN201680021578.2A patent/CN107613965A/zh active Pending
- 2016-02-19 CA CA2977367A patent/CA2977367A1/en not_active Abandoned
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2017
- 2017-08-03 PH PH12017501393A patent/PH12017501393A1/en unknown
- 2017-08-10 IL IL253949A patent/IL253949A0/en unknown
- 2017-08-18 US US15/680,737 patent/US10143696B2/en active Active
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| US9763955B2 (en) | 2017-09-19 |
| MX2017010682A (es) | 2018-04-24 |
| EP3258925B1 (en) | 2023-03-29 |
| BR112017017619A2 (pt) | 2018-05-08 |
| EP3258925A4 (en) | 2019-01-09 |
| IL253949A0 (en) | 2017-10-31 |
| EP3258925A1 (en) | 2017-12-27 |
| WO2016134283A1 (en) | 2016-08-25 |
| JP2018509397A (ja) | 2018-04-05 |
| US20170340646A1 (en) | 2017-11-30 |
| US10143696B2 (en) | 2018-12-04 |
| PH12017501393A1 (en) | 2018-01-08 |
| JP6762308B2 (ja) | 2020-09-30 |
| CN107613965A (zh) | 2018-01-19 |
| AU2016219879A1 (en) | 2017-08-24 |
| KR20170117170A (ko) | 2017-10-20 |
| US20160243129A1 (en) | 2016-08-25 |
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Legal Events
| Date | Code | Title | Description |
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| EEER | Examination request |
Effective date: 20170821 |
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| FZDE | Discontinued |
Effective date: 20191206 |