CA2977367A1 - Methods and compositions for decreasing gastric emptying - Google Patents
Methods and compositions for decreasing gastric emptying Download PDFInfo
- Publication number
- CA2977367A1 CA2977367A1 CA2977367A CA2977367A CA2977367A1 CA 2977367 A1 CA2977367 A1 CA 2977367A1 CA 2977367 A CA2977367 A CA 2977367A CA 2977367 A CA2977367 A CA 2977367A CA 2977367 A1 CA2977367 A1 CA 2977367A1
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- alkyl
- group
- agent
- optionally substituted
- treating
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| US9656959B2 (en) | 2010-12-22 | 2017-05-23 | Purdue Pharma L.P. | Substituted pyridines as sodium channel blockers |
| US9163008B2 (en) | 2011-09-02 | 2015-10-20 | Purdue Pharma, L.P. | Pyrimidines as sodium channel blockers |
| EP2935257B1 (en) | 2012-12-20 | 2018-02-07 | Purdue Pharma LP | Cyclic sulfonamides as sodium channel blockers |
| US9120786B2 (en) | 2013-03-04 | 2015-09-01 | Purdue Pharma, L.P. | Triazine carboxamides as sodium channel blockers |
| JP6426694B2 (ja) | 2013-03-15 | 2018-11-21 | グローバル ブラッド セラピューティクス インコーポレイテッド | ヘモグロビンの修飾のための化合物及びその使用 |
| WO2015031036A1 (en) | 2013-08-26 | 2015-03-05 | Purdue Pharma L.P. | Azaspiro[4.5] decane derivatives and use thereof |
| US9828348B2 (en) | 2013-11-08 | 2017-11-28 | Purdue Pharma L.P. | Benzimidazole derivatives and use thereof |
| EA201992707A1 (ru) | 2013-11-18 | 2020-06-30 | Глобал Блад Терапьютикс, Инк. | Соединения и их применения для модуляции гемоглобина |
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| WO2015097547A1 (en) | 2013-12-26 | 2015-07-02 | Purdue Pharma L.P. | 10-substituted morphinan hydantoins |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2017490C1 (ru) | 1990-01-18 | 1994-08-15 | Назаренко Петр Михайлович | Способ лечения демпин-синдрома после резекции желудка по способу бильрот-1 |
| ATE301457T1 (de) | 1995-06-12 | 2005-08-15 | Searle & Co | Mittel, enthaltend einen cyclooxygenase-2 inhibitor und einen 5-lipoxygenase inhibitor |
| US20040038970A1 (en) * | 1998-06-12 | 2004-02-26 | Societe De Conseils De Recherches Etd' Application Scientifiques, S.A.S. A Paris, France Corp. | Beta-carboline compounds |
| AR029489A1 (es) | 2000-03-10 | 2003-07-02 | Euro Celtique Sa | Piridinas, pirimidinas, pirazinas, triazinas sustituidas por arilo, composiciones farmaceuticas y el uso de las mismas para la manufactura de un medicamento |
| EP1292577B1 (en) | 2000-03-24 | 2012-10-24 | Euro-Celtique S.A. | Aryl substituted pyrazoles, triazoles and tetrazoles as sodium channel blocker |
| JP2003529589A (ja) | 2000-03-31 | 2003-10-07 | ユーロ−セルティック エス． ア． | アミノピリジンならびにこれらの鎮痙薬およびナトリウムチャンネル遮断薬としての使用 |
| IL159765A0 (en) | 2001-07-16 | 2004-06-20 | Euro Celtique Sa | Aryl substituted thiazolidinone derivatives and pharmaceutical compositions containing the same |
| AR036873A1 (es) | 2001-09-07 | 2004-10-13 | Euro Celtique Sa | Piridinas aril sustituidas a, composiciones farmaceuticas y el uso de las mismas para la preparacion de un medicamento |
| CA2479036A1 (en) | 2002-03-13 | 2003-09-18 | Euro-Celtique S.A. | Aryl substituted pyrimidines and the use thereof |
| JP2006504660A (ja) | 2002-07-31 | 2006-02-09 | ユーロ−セルティーク エス．エイ． | アリール置換ベンゾイミダゾール類およびナトリウムチャネルブロッカーとしてのそれらの使用 |
| CA2514574A1 (en) * | 2003-01-30 | 2004-08-12 | Dynogen Pharmaceuticals, Inc. | Use of sodium channel modulators for treating gastrointestinal tract disorders |
| EP1533298A1 (en) * | 2003-11-21 | 2005-05-25 | Newron Pharmaceuticals S.p.A. | 3-aminopyrrolidone derivatives |
| AU2006206274A1 (en) * | 2005-01-20 | 2006-07-27 | Sirtris Pharmaceuticals, Inc. | Use of sirtuin-activating compounds for treating flushing and drug induced weight gain |
| US20070020194A1 (en) * | 2005-06-08 | 2007-01-25 | Greenway Frank L Iii | Nasally administered appetite suppressant |
| EP1984339A1 (en) | 2006-01-23 | 2008-10-29 | Pfizer Limited | Pyridine derivatives as sodium channel modulators |
| WO2008044770A1 (en) * | 2006-10-13 | 2008-04-17 | Ajinomoto Co., Inc. | Agent for suppression of gastric emptying comprising 4-hydroxyisoleucine |
| ES2389456T3 (es) | 2006-11-01 | 2012-10-26 | Purdue Pharma Lp | Compuestos de fenilpropionamida y uso de los mismos |
| US8853250B2 (en) | 2007-07-13 | 2014-10-07 | Icagen, Inc. | Sodium channel inhibitors |
| JP5460589B2 (ja) | 2007-07-13 | 2014-04-02 | アイカジェン， インコーポレイテッド | ナトリウムチャネル阻害物質 |
| EP2582666B1 (en) | 2010-06-16 | 2014-08-13 | Purdue Pharma L.P. | Aryl substituted indoles and their use as blockers of sodium channels |
| WO2012004664A2 (en) | 2010-07-07 | 2012-01-12 | Purdue Pharma L.P. | Analogs of sodium channel peptide toxin |
| JP2013531687A (ja) | 2010-07-16 | 2013-08-08 | パーデュー、ファーマ、リミテッド、パートナーシップ | ナトリウムチャネル遮断剤としてのピリジン化合物 |
| EP2616441B1 (en) | 2010-09-17 | 2019-08-07 | Purdue Pharma L.P. | Pyridine compounds and the uses thereof |
| KR20130095772A (ko) | 2010-10-05 | 2013-08-28 | 퍼듀 퍼머 엘피 | 나트륨 채널 차단제로서 퀴나졸린 화합물 |
| US9656959B2 (en) | 2010-12-22 | 2017-05-23 | Purdue Pharma L.P. | Substituted pyridines as sodium channel blockers |
| US9163008B2 (en) | 2011-09-02 | 2015-10-20 | Purdue Pharma, L.P. | Pyrimidines as sodium channel blockers |
| BR112014009102A2 (pt) | 2011-10-26 | 2017-04-18 | Pfizer Ltd | compostos químicos |
| AU2012321111A1 (en) | 2011-10-31 | 2013-05-16 | Purdue Pharma L.P. | Quaternized amines as sodium channel blockers |
| WO2013072758A1 (en) | 2011-11-15 | 2013-05-23 | Purdue Pharma L.P. | Pyrimidine diol amides as sodium channel blockers |
| JP5938219B2 (ja) * | 2012-01-23 | 2016-06-22 | 株式会社明治 | 胃排出遅延のための食品用の剤または医療用の剤 |
| WO2013136170A1 (en) | 2012-03-16 | 2013-09-19 | Purdue Pharma L.P. | Substituted pyridines as sodium channel blockers |
| US9718865B2 (en) | 2012-07-27 | 2017-08-01 | Purdue Pharma L.P. | Sodium channel blocking peptides and the use thereof |
| JP6110516B2 (ja) * | 2013-03-04 | 2017-04-05 | パーデュー、ファーマ、リミテッド、パートナーシップ | ナトリウムチャネル遮断剤としてのピリミジンカルボキサミド |
| EP3666274A1 (en) | 2013-03-15 | 2020-06-17 | Purdue Pharma LP | Carboxamide derivatives and use thereof |
| AU2016219879A1 (en) * | 2015-02-19 | 2017-08-24 | Purdue Pharma L.P. | Methods and compositions for decreasing gastric emptying |
-
2016
- 2016-02-19 AU AU2016219879A patent/AU2016219879A1/en not_active Abandoned
- 2016-02-19 KR KR1020177025621A patent/KR20170117170A/ko not_active Withdrawn
- 2016-02-19 BR BR112017017619A patent/BR112017017619A2/pt not_active Application Discontinuation
- 2016-02-19 CA CA2977367A patent/CA2977367A1/en not_active Abandoned
- 2016-02-19 MX MX2017010682A patent/MX2017010682A/es unknown
- 2016-02-19 WO PCT/US2016/018715 patent/WO2016134283A1/en not_active Ceased
- 2016-02-19 EP EP16753165.6A patent/EP3258925B1/en active Active
- 2016-02-19 US US15/048,530 patent/US9763955B2/en active Active
- 2016-02-19 JP JP2017543916A patent/JP6762308B2/ja active Active
- 2016-02-19 CN CN201680021578.2A patent/CN107613965A/zh active Pending
-
2017
- 2017-08-03 PH PH12017501393A patent/PH12017501393A1/en unknown
- 2017-08-10 IL IL253949A patent/IL253949A0/en unknown
- 2017-08-18 US US15/680,737 patent/US10143696B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| US10143696B2 (en) | 2018-12-04 |
| JP2018509397A (ja) | 2018-04-05 |
| KR20170117170A (ko) | 2017-10-20 |
| US9763955B2 (en) | 2017-09-19 |
| JP6762308B2 (ja) | 2020-09-30 |
| EP3258925B1 (en) | 2023-03-29 |
| US20170340646A1 (en) | 2017-11-30 |
| BR112017017619A2 (pt) | 2018-05-08 |
| PH12017501393A1 (en) | 2018-01-08 |
| CN107613965A (zh) | 2018-01-19 |
| AU2016219879A1 (en) | 2017-08-24 |
| MX2017010682A (es) | 2018-04-24 |
| IL253949A0 (en) | 2017-10-31 |
| US20160243129A1 (en) | 2016-08-25 |
| EP3258925A1 (en) | 2017-12-27 |
| WO2016134283A1 (en) | 2016-08-25 |
| EP3258925A4 (en) | 2019-01-09 |
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Legal Events
| Date | Code | Title | Description |
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| EEER | Examination request |
Effective date: 20170821 |
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| FZDE | Discontinued |
Effective date: 20191206 |