CA2948175A1 - Pyrrolidine gpr40 modulators for the treatment of diseases such as diabetes - Google Patents
Pyrrolidine gpr40 modulators for the treatment of diseases such as diabetes Download PDFInfo
- Publication number
- CA2948175A1 CA2948175A1 CA2948175A CA2948175A CA2948175A1 CA 2948175 A1 CA2948175 A1 CA 2948175A1 CA 2948175 A CA2948175 A CA 2948175A CA 2948175 A CA2948175 A CA 2948175A CA 2948175 A1 CA2948175 A1 CA 2948175A1
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- Prior art keywords
- substituted
- alkyl
- occurrence
- independently selected
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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Classifications
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US201461989560P | 2014-05-07 | 2014-05-07 | |
| US61/989,560 | 2014-05-07 | ||
| PCT/US2015/029422 WO2015171733A1 (en) | 2014-05-07 | 2015-05-06 | Pyrrolidine gpr40 modulators for the treatment of diseases such as diabetes |
Publications (1)
| Publication Number | Publication Date |
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| CA2948175A1 true CA2948175A1 (en) | 2015-11-12 |
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| CA2948175A Abandoned CA2948175A1 (en) | 2014-05-07 | 2015-05-06 | Pyrrolidine gpr40 modulators for the treatment of diseases such as diabetes |
Country Status (14)
| Country | Link |
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| US (1) | US10017497B2 (OSRAM) |
| EP (1) | EP3140297B1 (OSRAM) |
| JP (1) | JP6488320B2 (OSRAM) |
| KR (1) | KR20170002543A (OSRAM) |
| CN (1) | CN106458987B (OSRAM) |
| AU (1) | AU2015256038B2 (OSRAM) |
| BR (1) | BR112016025188A2 (OSRAM) |
| CA (1) | CA2948175A1 (OSRAM) |
| EA (1) | EA032290B1 (OSRAM) |
| ES (1) | ES2671402T3 (OSRAM) |
| IL (1) | IL248670B (OSRAM) |
| MX (1) | MX2016014118A (OSRAM) |
| SG (1) | SG11201609167RA (OSRAM) |
| WO (1) | WO2015171733A1 (OSRAM) |
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| JP7062792B2 (ja) | 2018-02-13 | 2022-05-06 | ギリアード サイエンシーズ， インコーポレイテッド | Ｐｄ－１／ｐｄ－ｌ１阻害剤 |
| EP3781556B1 (en) | 2018-04-19 | 2025-06-18 | Gilead Sciences, Inc. | Pd-1/pd-l1 inhibitors |
| CN118221646A (zh) | 2018-07-13 | 2024-06-21 | 吉利德科学公司 | Pd-1/pd-l1抑制剂 |
| KR102635333B1 (ko) | 2018-10-24 | 2024-02-15 | 길리애드 사이언시즈, 인코포레이티드 | Pd-1/pd-l1 억제제 |
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| US5614492A (en) | 1986-05-05 | 1997-03-25 | The General Hospital Corporation | Insulinotropic hormone GLP-1 (7-36) and uses thereof |
| US6995183B2 (en) | 2003-08-01 | 2006-02-07 | Bristol Myers Squibb Company | Adamantylglycine-based inhibitors of dipeptidyl peptidase IV and methods |
| AU2010303670A1 (en) * | 2009-10-06 | 2012-03-29 | Bristol-Myers Squibb Company | Pyrrolidine GPR40 modulators |
| JP5864177B2 (ja) | 2011-09-15 | 2016-02-17 | 船井電機株式会社 | プロジェクタおよびプロジェクタシステム |
| CA2891569A1 (en) | 2012-11-16 | 2014-05-22 | Bristol-Myers Squibb Company | Pyrrolidine gpr40 modulators |
| ES2606685T3 (es) * | 2012-11-16 | 2017-03-27 | Bristol-Myers Squibb Company | Moduladores de dihidropirazol GPR40 |
| MX2015005720A (es) * | 2012-11-16 | 2015-09-08 | Bristol Myers Squibb Co | Moduladores de dihidropirazol de receptor acoplado a la proteina g (gpr40). |
| ES2605856T3 (es) * | 2012-11-16 | 2017-03-16 | Bristol-Myers Squibb Company | Moduladores GPR40 de dihidropirazol |
| BR112016024936A2 (pt) * | 2014-05-07 | 2017-08-15 | Bristol Myers Squibb Co | moduladores de gpr40 à base de pirrolidina para tratamento de doenças como diabetes |
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2015
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- 2015-05-06 AU AU2015256038A patent/AU2015256038B2/en not_active Ceased
- 2015-05-06 SG SG11201609167RA patent/SG11201609167RA/en unknown
- 2015-05-06 CN CN201580023783.8A patent/CN106458987B/zh not_active Expired - Fee Related
- 2015-05-06 CA CA2948175A patent/CA2948175A1/en not_active Abandoned
- 2015-05-06 BR BR112016025188A patent/BR112016025188A2/pt not_active Application Discontinuation
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- 2015-05-06 WO PCT/US2015/029422 patent/WO2015171733A1/en not_active Ceased
- 2015-05-06 KR KR1020167033864A patent/KR20170002543A/ko not_active Withdrawn
- 2015-05-06 JP JP2016566729A patent/JP6488320B2/ja not_active Expired - Fee Related
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- 2015-05-06 MX MX2016014118A patent/MX2016014118A/es unknown
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2016
- 2016-11-01 IL IL248670A patent/IL248670B/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| JP6488320B2 (ja) | 2019-03-20 |
| CN106458987A (zh) | 2017-02-22 |
| US10017497B2 (en) | 2018-07-10 |
| BR112016025188A2 (pt) | 2017-08-15 |
| US20170217930A1 (en) | 2017-08-03 |
| WO2015171733A1 (en) | 2015-11-12 |
| EA201692216A1 (ru) | 2017-04-28 |
| CN106458987B (zh) | 2019-09-24 |
| SG11201609167RA (en) | 2016-12-29 |
| IL248670A0 (en) | 2017-01-31 |
| EA032290B1 (ru) | 2019-05-31 |
| JP2017514865A (ja) | 2017-06-08 |
| EP3140297B1 (en) | 2018-04-11 |
| EP3140297A1 (en) | 2017-03-15 |
| AU2015256038A1 (en) | 2016-12-22 |
| AU2015256038B2 (en) | 2019-07-11 |
| MX2016014118A (es) | 2017-02-09 |
| KR20170002543A (ko) | 2017-01-06 |
| ES2671402T3 (es) | 2018-06-06 |
| IL248670B (en) | 2019-09-26 |
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