CA2913313A1 - Dinuceloside polyphosphates for the treatment of pain - Google Patents
Dinuceloside polyphosphates for the treatment of pain Download PDFInfo
- Publication number
- CA2913313A1 CA2913313A1 CA2913313A CA2913313A CA2913313A1 CA 2913313 A1 CA2913313 A1 CA 2913313A1 CA 2913313 A CA2913313 A CA 2913313A CA 2913313 A CA2913313 A CA 2913313A CA 2913313 A1 CA2913313 A1 CA 2913313A1
- Authority
- CA
- Canada
- Prior art keywords
- pain
- dinucleoside polyphosphate
- polyphosphate analogue
- analogue
- use according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
- C07F9/65616—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings containing the ring system having three or more than three double bonds between ring members or between ring members and non-ring members, e.g. purine or analogs
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
- C07H21/02—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids with ribosyl as saccharide radical
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Biochemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Endocrinology (AREA)
- Pain & Pain Management (AREA)
- Reproductive Health (AREA)
- Rheumatology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB201209244A GB201209244D0 (en) | 2012-05-25 | 2012-05-25 | Compositions |
| GB1209244.1 | 2012-05-25 | ||
| PCT/GB2013/051377 WO2013175231A1 (en) | 2012-05-25 | 2013-05-24 | Dinuceloside polyphosphates for the treatment of pain |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2913313A1 true CA2913313A1 (en) | 2013-11-28 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2913313A Abandoned CA2913313A1 (en) | 2012-05-25 | 2013-05-24 | Dinuceloside polyphosphates for the treatment of pain |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20150119352A1 (enExample) |
| EP (1) | EP2854821A1 (enExample) |
| JP (1) | JP2015517565A (enExample) |
| AU (1) | AU2013264966A1 (enExample) |
| CA (1) | CA2913313A1 (enExample) |
| GB (1) | GB201209244D0 (enExample) |
| HK (1) | HK1203054A1 (enExample) |
| WO (1) | WO2013175231A1 (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN107312039B (zh) | 2012-08-30 | 2019-06-25 | 江苏豪森药业集团有限公司 | 一种替诺福韦前药的制备方法 |
| GB201320962D0 (en) * | 2013-11-27 | 2014-01-08 | Globalacorn Ltd | Compositions |
| WO2017209267A1 (ja) * | 2016-06-03 | 2017-12-07 | 塩野義製薬株式会社 | プリン誘導体 |
| CN112004551A (zh) | 2018-03-15 | 2020-11-27 | 丹米尔治疗有限责任公司 | 3”,5”-二烷氧基苯甲酰基-3’-氨基-3’-脱氧腺苷-5’-三磷酸及其药物用途 |
| WO2021117874A1 (ja) * | 2019-12-13 | 2021-06-17 | 中外製薬株式会社 | 細胞外プリン受容体リガンドを検出するシステムおよび当該システムを導入した非ヒト動物 |
| US20230032473A1 (en) * | 2021-07-23 | 2023-02-02 | Wisconsin Alumni Research Foundation | Nad(h) nanoparticles and methods of use |
| CN114685588B (zh) * | 2022-05-05 | 2024-03-29 | 江苏申基生物科技有限公司 | 一种含开环核苷结构的起始加帽寡核苷酸引物 |
| WO2026014535A1 (ja) * | 2024-07-11 | 2026-01-15 | 国立大学法人旭川医科大学 | 子宮内膜症の予防又は治療用組成物 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5049550A (en) * | 1987-11-05 | 1991-09-17 | Worcester Foundation For Experimental Biology | Diadenosine 5', 5'"-p1, p4,-tetraphosphate analogs as antithrombotic agents |
| JP2783880B2 (ja) * | 1989-11-24 | 1998-08-06 | 富士レビオ株式会社 | 心臓病治療剤 |
| US5635160A (en) * | 1995-06-07 | 1997-06-03 | The University Of North Carolina At Chapel Hill | Dinucleotides useful for the treatment of cystic fibrosis and for hydrating mucus secretions |
| US5837861A (en) * | 1997-02-10 | 1998-11-17 | Inspire Pharmaceuticals, Inc. | Dinucleotides and their use as modulators of mucociliary clearance and ciliary beat frequency |
| US5681823A (en) * | 1996-05-02 | 1997-10-28 | Prp Inc. | P1, P4 -dithio-P2 -P3 -monochloromethylene 5', 5'"-diadenosine P1, P4 -tetraphosphate as antithrombotic agent |
| US6462028B2 (en) * | 1997-07-25 | 2002-10-08 | Inspire Pharmaceuticals, Inc. | Method of promoting cervical and vaginal secretions |
| WO2003000056A1 (en) * | 2001-06-25 | 2003-01-03 | Inspire Pharmaceuticals, Inc. | Joint lubrication with p2y purinergic receptor agonists |
| MXPA04004215A (es) * | 2001-11-06 | 2004-07-08 | Inspire Pharmaceuticals Inc | Metodo para el tratamiento o la prevencion de enfermedades inflamatorias. |
| EP1348466A3 (en) * | 2002-02-01 | 2003-10-29 | Inspire Pharmaceuticals, Inc. | Method for treating pain with adenosine-tetraphosphates |
| FR2842424A1 (fr) * | 2002-07-22 | 2004-01-23 | Univ Paris 7 Denis Diderot | Utilisation du nad ou de l'un de ses analogues, substrat des mono-adp-ribosyl tranferases, pour la preparation d'un medicament destine au traitement des pathologies liees aux recepteurs purinergiques |
| GB0502250D0 (en) * | 2005-02-03 | 2005-03-09 | Ic Vec Ltd | Use |
-
2012
- 2012-05-25 GB GB201209244A patent/GB201209244D0/en not_active Ceased
-
2013
- 2013-05-24 WO PCT/GB2013/051377 patent/WO2013175231A1/en not_active Ceased
- 2013-05-24 US US14/403,560 patent/US20150119352A1/en not_active Abandoned
- 2013-05-24 AU AU2013264966A patent/AU2013264966A1/en not_active Abandoned
- 2013-05-24 HK HK15103596.5A patent/HK1203054A1/xx unknown
- 2013-05-24 CA CA2913313A patent/CA2913313A1/en not_active Abandoned
- 2013-05-24 EP EP13725462.9A patent/EP2854821A1/en not_active Withdrawn
- 2013-05-24 JP JP2015513277A patent/JP2015517565A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| EP2854821A1 (en) | 2015-04-08 |
| JP2015517565A (ja) | 2015-06-22 |
| AU2013264966A1 (en) | 2015-01-22 |
| US20150119352A1 (en) | 2015-04-30 |
| WO2013175231A1 (en) | 2013-11-28 |
| GB201209244D0 (en) | 2012-07-04 |
| HK1203054A1 (en) | 2015-10-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |
Effective date: 20190524 |