CA2908815A1 - Drug combinations to treat cancer - Google Patents
Drug combinations to treat cancerInfo
- Publication number
- CA2908815A1 CA2908815A1 CA2908815A CA2908815A CA2908815A1 CA 2908815 A1 CA2908815 A1 CA 2908815A1 CA 2908815 A CA2908815 A CA 2908815A CA 2908815 A CA2908815 A CA 2908815A CA 2908815 A1 CA2908815 A1 CA 2908815A1
- Authority
- CA
- Canada
- Prior art keywords
- compound
- administered
- dose
- fasting
- once daily
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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| JP6158705B2 (ja) | 2010-09-27 | 2017-07-05 | エクセリクシス， インク． | 去勢抵抗性前立腺癌および造骨性転移の治療のためのｍｅｔおよびｖｅｇｆの二元阻害薬 |
| KR20210147117A (ko) | 2011-02-10 | 2021-12-06 | 엑셀리시스, 인코포레이티드 | 퀴놀린 화합물들의 제조 방법들 및 상기 화합물들을 함유하는 약학 조성물들 |
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| ES2927651T3 (es) | 2013-04-04 | 2022-11-10 | Exelixis Inc | Forma de dosificación de cabozantinib y uso en el tratamiento del cáncer |
| UA123534C2 (uk) | 2014-02-14 | 2021-04-21 | Екселіксис, Інк. | Кристалічні тверді форми n-{4-[(6,7-диметоксихінолін-4-іл)окси]феніл}-n'-(4-флуорофеніл)циклопропан-1,1-дикарбоксаміду, способи отримання і способи застосування |
| JP6666849B2 (ja) | 2014-03-17 | 2020-03-18 | エグゼリクシス， インコーポレイテッド | カボザンチニブ製剤の投与 |
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| CN109069499A (zh) | 2016-04-15 | 2018-12-21 | 埃克塞里艾克西斯公司 | 使用 n-(4-(6,7-二甲氧基喹啉-4-基氧基)苯基)-n’-(4-氟苯基)环丙烷-1,1-二甲酰胺,(2s)-羟基丁二酸盐治疗肾细胞癌的方法 |
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| TW201118072A (en) * | 2009-07-17 | 2011-06-01 | Exelixis Inc | Crystalline forms of N-[3-fluoro-4-({6-(methyloxy)-7-[(3-morpholin-4-ylpropyl)oxy]-quinolin-4-yl}oxy)phenyl]-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide |
| UA108618C2 (uk) * | 2009-08-07 | 2015-05-25 | Застосування c-met-модуляторів в комбінації з темозоломідом та/або променевою терапією для лікування раку | |
| JP6158705B2 (ja) * | 2010-09-27 | 2017-07-05 | エクセリクシス， インク． | 去勢抵抗性前立腺癌および造骨性転移の治療のためのｍｅｔおよびｖｅｇｆの二元阻害薬 |
| CN103664778B (zh) * | 2013-11-27 | 2017-04-05 | 苏州摩尔医药有限公司 | 一种抗肿瘤治疗药物卡博替尼的合成方法 |
-
2014
- 2014-04-04 CN CN201480029297.2A patent/CN108472242A/zh active Pending
- 2014-04-04 AU AU2014248001A patent/AU2014248001A1/en not_active Abandoned
- 2014-04-04 KR KR1020157030445A patent/KR20150138268A/ko not_active Withdrawn
- 2014-04-04 CA CA2908815A patent/CA2908815A1/en not_active Abandoned
- 2014-04-04 EP EP14724594.8A patent/EP2983639A1/en not_active Withdrawn
- 2014-04-04 WO PCT/US2014/033008 patent/WO2014165779A1/en not_active Ceased
- 2014-04-04 MX MX2015014046A patent/MX2015014046A/es unknown
- 2014-04-04 JP JP2016506653A patent/JP2016515628A/ja active Pending
- 2014-04-04 BR BR112015025408A patent/BR112015025408A8/pt not_active IP Right Cessation
- 2014-04-04 HK HK16109729.1A patent/HK1221424A1/zh unknown
- 2014-04-04 US US14/782,493 patent/US20160082019A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2014165779A1 (en) | 2014-10-09 |
| CN108472242A (zh) | 2018-08-31 |
| HK1221424A1 (zh) | 2017-06-02 |
| EP2983639A1 (en) | 2016-02-17 |
| JP2016515628A (ja) | 2016-05-30 |
| BR112015025408A2 (pt) | 2017-07-18 |
| AU2014248001A1 (en) | 2015-11-19 |
| MX2015014046A (es) | 2016-05-16 |
| BR112015025408A8 (pt) | 2018-07-10 |
| US20160082019A1 (en) | 2016-03-24 |
| KR20150138268A (ko) | 2015-12-09 |
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