CA2860810A1 - (3,4-dichloro-phenyl)-((s)-3-propyl-pyrrolidin-3-yl)-methanone hydrochloride and manufacturing processes - Google Patents
(3,4-dichloro-phenyl)-((s)-3-propyl-pyrrolidin-3-yl)-methanone hydrochloride and manufacturing processes Download PDFInfo
- Publication number
- CA2860810A1 CA2860810A1 CA2860810A CA2860810A CA2860810A1 CA 2860810 A1 CA2860810 A1 CA 2860810A1 CA 2860810 A CA2860810 A CA 2860810A CA 2860810 A CA2860810 A CA 2860810A CA 2860810 A1 CA2860810 A1 CA 2860810A1
- Authority
- CA
- Canada
- Prior art keywords
- compound
- formula
- mmol
- certain embodiment
- added
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP12165529 | 2012-04-25 | ||
EP12165527 | 2012-04-25 | ||
EP12165529.4 | 2012-04-25 | ||
EP12165527.8 | 2012-04-25 | ||
PCT/EP2013/058344 WO2013160273A1 (en) | 2012-04-25 | 2013-04-23 | (3,4-dichloro-phenyl)-((s)-3-propyl-pyrrolidin-3-yl)-methanone hydrochloride and manufacturing processes |
Publications (1)
Publication Number | Publication Date |
---|---|
CA2860810A1 true CA2860810A1 (en) | 2013-10-31 |
Family
ID=48170481
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA2860810A Abandoned CA2860810A1 (en) | 2012-04-25 | 2013-04-23 | (3,4-dichloro-phenyl)-((s)-3-propyl-pyrrolidin-3-yl)-methanone hydrochloride and manufacturing processes |
Country Status (10)
Country | Link |
---|---|
US (1) | US9527810B2 (ja) |
EP (1) | EP2841418B1 (ja) |
JP (1) | JP6235560B2 (ja) |
KR (1) | KR20150013137A (ja) |
CN (1) | CN104203915B (ja) |
CA (1) | CA2860810A1 (ja) |
HK (1) | HK1200818A1 (ja) |
MX (1) | MX2014011419A (ja) |
RU (1) | RU2014145806A (ja) |
WO (1) | WO2013160273A1 (ja) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN108689904B (zh) * | 2017-04-12 | 2022-06-17 | 轩竹生物科技股份有限公司 | 手性杂环叔醇中间体的制备方法及其应用 |
WO2023161533A1 (en) | 2022-02-28 | 2023-08-31 | Noema Pharma Ag | Triple uptake inhibitor for the treatment of atypical depression |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1599032A (en) | 1977-03-04 | 1981-09-30 | May & Baker Ltd | Imidazole derivatives having herbicidal activity |
JP2006505531A (ja) * | 2002-09-11 | 2006-02-16 | メルク エンド カムパニー インコーポレーテッド | メラノコルチン−4受容体作働薬としてのピペラジン尿素誘導体 |
GB0325745D0 (en) * | 2003-11-05 | 2003-12-10 | Astrazeneca Ab | Chemical compounds |
KR20050045927A (ko) * | 2003-11-12 | 2005-05-17 | 주식회사 엘지생명과학 | 멜라노코틴 수용체의 항진제 |
ATE513808T1 (de) * | 2006-12-19 | 2011-07-15 | Hoffmann La Roche | Heteroarylpyrrolidinyl- und piperidinylketonderivate |
UA107652C2 (en) | 2008-10-06 | 2015-02-10 | Incuron Llc | Carbazole compounds and therapeutic uses of the compounds |
UA99555C2 (en) | 2008-11-12 | 2012-08-27 | Элджи Лайф Саенсез Лтд. | Melanocortin receptor agonists |
WO2010121022A1 (en) | 2009-04-15 | 2010-10-21 | Research Triangle Institute | Monoamine reuptake inhibitors |
MX339899B (es) * | 2011-02-25 | 2016-06-16 | Array Biopharma Inc | Compuestos de triazolopiridina como inhibidores de pim cinasa. |
-
2013
- 2013-04-23 MX MX2014011419A patent/MX2014011419A/es unknown
- 2013-04-23 JP JP2015507491A patent/JP6235560B2/ja active Active
- 2013-04-23 CN CN201380012619.8A patent/CN104203915B/zh active Active
- 2013-04-23 RU RU2014145806A patent/RU2014145806A/ru not_active Application Discontinuation
- 2013-04-23 KR KR1020147029811A patent/KR20150013137A/ko not_active Application Discontinuation
- 2013-04-23 EP EP13718188.9A patent/EP2841418B1/en active Active
- 2013-04-23 WO PCT/EP2013/058344 patent/WO2013160273A1/en active Application Filing
- 2013-04-23 CA CA2860810A patent/CA2860810A1/en not_active Abandoned
-
2014
- 2014-10-24 US US14/522,775 patent/US9527810B2/en active Active
-
2015
- 2015-02-05 HK HK15101246.3A patent/HK1200818A1/xx unknown
Also Published As
Publication number | Publication date |
---|---|
HK1200818A1 (en) | 2015-08-14 |
CN104203915A (zh) | 2014-12-10 |
MX2014011419A (es) | 2014-11-25 |
KR20150013137A (ko) | 2015-02-04 |
JP6235560B2 (ja) | 2017-11-22 |
EP2841418B1 (en) | 2017-03-08 |
CN104203915B (zh) | 2017-03-08 |
JP2015515484A (ja) | 2015-05-28 |
US9527810B2 (en) | 2016-12-27 |
WO2013160273A1 (en) | 2013-10-31 |
EP2841418A1 (en) | 2015-03-04 |
US20150045408A1 (en) | 2015-02-12 |
RU2014145806A (ru) | 2016-06-10 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FZDE | Dead |
Effective date: 20190423 |