CA2834528A1 - Protein kinase inhibitors - Google Patents
Protein kinase inhibitors Download PDFInfo
- Publication number
- CA2834528A1 CA2834528A1 CA2834528A CA2834528A CA2834528A1 CA 2834528 A1 CA2834528 A1 CA 2834528A1 CA 2834528 A CA2834528 A CA 2834528A CA 2834528 A CA2834528 A CA 2834528A CA 2834528 A1 CA2834528 A1 CA 2834528A1
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- CA
- Canada
- Prior art keywords
- compound
- kinase
- protein kinase
- formula
- activity
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Classifications
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- G01N33/58—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving labelled substances
- G01N33/582—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving labelled substances with fluorescent label
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Landscapes
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Priority Applications (10)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CA2834528A CA2834528A1 (en) | 2013-11-26 | 2013-11-26 | Protein kinase inhibitors |
| CA2929889A CA2929889A1 (en) | 2013-11-26 | 2014-11-26 | Protein kinase inhibitors |
| CN201480064253.3A CN105764906A (zh) | 2013-11-26 | 2014-11-26 | 蛋白激酶抑制剂 |
| JP2016554766A JP2017503006A (ja) | 2013-11-26 | 2014-11-26 | プロテインキナーゼ阻害剤 |
| EP14865858.6A EP3074401A4 (en) | 2013-11-26 | 2014-11-26 | Protein kinase inhibitors |
| KR1020167014057A KR20160089378A (ko) | 2013-11-26 | 2014-11-26 | 단백질 키나제 저해제 |
| US15/039,127 US20170158697A1 (en) | 2013-11-26 | 2014-11-26 | Protein Kinase Inhibitors |
| TW103141063A TW201602112A (zh) | 2013-11-26 | 2014-11-26 | 蛋白質激酶抑制劑 |
| RU2016124366A RU2016124366A (ru) | 2013-11-26 | 2014-11-26 | Ингибиторы протеинкиназы |
| PCT/CA2014/000848 WO2015077866A1 (en) | 2013-11-26 | 2014-11-26 | Protein kinase inhibitors |
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| CA2834528A CA2834528A1 (en) | 2013-11-26 | 2013-11-26 | Protein kinase inhibitors |
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| CA2929889A Abandoned CA2929889A1 (en) | 2013-11-26 | 2014-11-26 | Protein kinase inhibitors |
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| CA2929889A Abandoned CA2929889A1 (en) | 2013-11-26 | 2014-11-26 | Protein kinase inhibitors |
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| EP (1) | EP3074401A4 (enExample) |
| JP (1) | JP2017503006A (enExample) |
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| CN (1) | CN105764906A (enExample) |
| CA (2) | CA2834528A1 (enExample) |
| RU (1) | RU2016124366A (enExample) |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2016187723A1 (en) * | 2015-05-27 | 2016-12-01 | Pharmascience Inc. | Inhibitors of the tec kinase enzyme family |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN108794483B (zh) * | 2018-04-27 | 2021-04-23 | 四川大学华西医院 | 一种7-脱氮嘌呤衍生物及其六元环超分子结构 |
| KR20230064355A (ko) | 2021-11-03 | 2023-05-10 | 고려대학교 산학협력단 | Ｎ아세틸ｌ트립토판 ３，５비스（트리플루오로메틸）벤질 에스테르 화합물을 유효성분으로 포함하는 통증의 예방 또는 치료용 약학적 조성물 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7863444B2 (en) * | 1997-03-19 | 2011-01-04 | Abbott Laboratories | 4-aminopyrrolopyrimidines as kinase inhibitors |
| US6713474B2 (en) * | 1998-09-18 | 2004-03-30 | Abbott Gmbh & Co. Kg | Pyrrolopyrimidines as therapeutic agents |
| DE69928414T2 (de) * | 1998-09-18 | 2006-08-03 | Abbott Gmbh & Co. Kg | 4-aminopyrrolopyrimidine als kinaseinhibitoren |
| TR200101186T2 (tr) * | 1998-09-18 | 2001-10-22 | Basf Aktiengesellschaft | Protein kinaz engelleyiciler olarak pyrrolopyrimidin'ler |
| AU2000240570A1 (en) * | 2000-03-29 | 2001-10-08 | Knoll Gesellschaft Mit Beschraenkter Haftung | Pyrrolopyrimidines as tyrosine kinase inhibitors |
| US9796716B2 (en) * | 2012-05-31 | 2017-10-24 | Pharmascience, Inc. | Selective inhibitors of Tec and Src protein kinase families |
| CA2813299A1 (en) * | 2013-04-17 | 2014-10-17 | Pharmascience Inc. | Protein kinase inhibitors |
| CA2779184A1 (en) * | 2012-05-31 | 2013-11-30 | Pharmascience Inc. | Protein kinase inhibitors |
| CA2782774A1 (en) * | 2012-07-06 | 2014-01-06 | Pharmascience Inc. | Protein kinase inhibitors |
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2013
- 2013-11-26 CA CA2834528A patent/CA2834528A1/en not_active Abandoned
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2014
- 2014-11-26 CA CA2929889A patent/CA2929889A1/en not_active Abandoned
- 2014-11-26 RU RU2016124366A patent/RU2016124366A/ru unknown
- 2014-11-26 CN CN201480064253.3A patent/CN105764906A/zh active Pending
- 2014-11-26 EP EP14865858.6A patent/EP3074401A4/en not_active Withdrawn
- 2014-11-26 WO PCT/CA2014/000848 patent/WO2015077866A1/en not_active Ceased
- 2014-11-26 US US15/039,127 patent/US20170158697A1/en not_active Abandoned
- 2014-11-26 TW TW103141063A patent/TW201602112A/zh unknown
- 2014-11-26 KR KR1020167014057A patent/KR20160089378A/ko not_active Withdrawn
- 2014-11-26 JP JP2016554766A patent/JP2017503006A/ja not_active Withdrawn
Cited By (1)
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| WO2016187723A1 (en) * | 2015-05-27 | 2016-12-01 | Pharmascience Inc. | Inhibitors of the tec kinase enzyme family |
Also Published As
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|---|---|
| WO2015077866A1 (en) | 2015-06-04 |
| CA2929889A1 (en) | 2015-06-04 |
| TW201602112A (zh) | 2016-01-16 |
| JP2017503006A (ja) | 2017-01-26 |
| CN105764906A (zh) | 2016-07-13 |
| KR20160089378A (ko) | 2016-07-27 |
| RU2016124366A (ru) | 2018-01-09 |
| US20170158697A1 (en) | 2017-06-08 |
| EP3074401A1 (en) | 2016-10-05 |
| EP3074401A4 (en) | 2017-05-10 |
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| FZDE | Discontinued |
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