CA2733265A1 - Transdermal extended-delivery donepezil compositions and methods for using the same - Google Patents

Transdermal extended-delivery donepezil compositions and methods for using the same Download PDF

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Publication number
CA2733265A1
CA2733265A1 CA2733265A CA2733265A CA2733265A1 CA 2733265 A1 CA2733265 A1 CA 2733265A1 CA 2733265 A CA2733265 A CA 2733265A CA 2733265 A CA2733265 A CA 2733265A CA 2733265 A1 CA2733265 A1 CA 2733265A1
Authority
CA
Canada
Prior art keywords
active agent
donepezil active
donepezil
composition according
extended delivery
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2733265A
Other languages
English (en)
French (fr)
Inventor
Jianye Wen
Yoshiko Katori
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Teikoku Pharma USA Inc
Original Assignee
Teikoku Pharma USA Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teikoku Pharma USA Inc filed Critical Teikoku Pharma USA Inc
Publication of CA2733265A1 publication Critical patent/CA2733265A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A61K9/7061—Polyacrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA2733265A 2008-09-30 2009-08-31 Transdermal extended-delivery donepezil compositions and methods for using the same Abandoned CA2733265A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10141208P 2008-09-30 2008-09-30
US61/101,412 2008-09-30
PCT/US2009/055542 WO2010039381A1 (en) 2008-09-30 2009-08-31 Transdermal extended-delivery donepezil compositions and methods for using the same

Publications (1)

Publication Number Publication Date
CA2733265A1 true CA2733265A1 (en) 2010-04-08

Family

ID=42057739

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2733265A Abandoned CA2733265A1 (en) 2008-09-30 2009-08-31 Transdermal extended-delivery donepezil compositions and methods for using the same

Country Status (12)

Country Link
US (1) US20100080842A1 (enExample)
EP (1) EP2328582A4 (enExample)
JP (1) JP2012504163A (enExample)
CN (1) CN102164601A (enExample)
AR (1) AR073696A1 (enExample)
AU (1) AU2009300184A1 (enExample)
BR (1) BRPI0917862A2 (enExample)
CA (1) CA2733265A1 (enExample)
IL (1) IL210970A0 (enExample)
MX (1) MX2011002260A (enExample)
TW (1) TW201029653A (enExample)
WO (1) WO2010039381A1 (enExample)

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WO2013078608A1 (en) 2011-11-29 2013-06-06 Ziqiang Gu Donepezil pamoate and methods of making and using the same
KR101485822B1 (ko) 2014-01-22 2015-01-23 주식회사 대웅제약 도네페질 또는 그의 염을 함유하는 경피흡수제제
ES2829807T3 (es) 2014-02-20 2021-06-02 Nal Pharmaceutical Group Ltd Sistema de administración transdérmica de fármacos que contiene donepezilo
JP6793648B2 (ja) * 2014-12-18 2020-12-02 アイキュア ファーマスーティカル インク． ドネペジルを有効成分として含有する経皮吸収製剤
KR102033686B1 (ko) 2017-05-19 2019-10-18 보령제약 주식회사 도네페질을 함유하는 마이크로니들 경피 패치
US20190175520A1 (en) * 2017-12-13 2019-06-13 Corium International, Inc. Method for depot creation during transdermal drug delivery
KR102024996B1 (ko) 2017-12-27 2019-09-25 동아에스티 주식회사 도네페질을 함유하는 치매 치료용 경피흡수제제
KR102372630B1 (ko) 2019-05-15 2022-03-14 주식회사 대웅제약 고함량의 도네페질 또는 그의 염을 포함하는 경피흡수제제
CN112823793A (zh) * 2019-11-20 2021-05-21 成都康弘药业集团股份有限公司 一种含有多奈哌齐的透皮贴剂及其制备方法
WO2024127805A1 (ja) * 2022-12-16 2024-06-20 帝國製薬株式会社 ドネペジル含有経皮吸収製剤

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Also Published As

Publication number Publication date
CN102164601A (zh) 2011-08-24
TW201029653A (en) 2010-08-16
EP2328582A1 (en) 2011-06-08
BRPI0917862A2 (pt) 2015-11-24
JP2012504163A (ja) 2012-02-16
AR073696A1 (es) 2010-11-24
EP2328582A4 (en) 2012-02-22
MX2011002260A (es) 2011-04-07
WO2010039381A1 (en) 2010-04-08
IL210970A0 (en) 2011-04-28
US20100080842A1 (en) 2010-04-01
AU2009300184A1 (en) 2010-04-08

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Legal Events

Date Code Title Description
FZDE Discontinued