BRPI0917862A2 - composições transdérmicas de donepezil com distribuição prolongada e métodos para usar as mesmas - Google Patents
composições transdérmicas de donepezil com distribuição prolongada e métodos para usar as mesmasInfo
- Publication number
- BRPI0917862A2 BRPI0917862A2 BRPI0917862A BRPI0917862A BRPI0917862A2 BR PI0917862 A2 BRPI0917862 A2 BR PI0917862A2 BR PI0917862 A BRPI0917862 A BR PI0917862A BR PI0917862 A BRPI0917862 A BR PI0917862A BR PI0917862 A2 BRPI0917862 A2 BR PI0917862A2
- Authority
- BR
- Brazil
- Prior art keywords
- methods
- compositions
- prolonged distribution
- transdermal donepezil
- transdermal
- Prior art date
Links
- ADEBPBSSDYVVLD-UHFFFAOYSA-N donepezil Chemical compound O=C1C=2C=C(OC)C(OC)=CC=2CC1CC(CC1)CCN1CC1=CC=CC=C1 ADEBPBSSDYVVLD-UHFFFAOYSA-N 0.000 title 2
- 229960003530 donepezil Drugs 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 230000002035 prolonged effect Effects 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
- A61K9/7061—Polyacrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10141208P | 2008-09-30 | 2008-09-30 | |
PCT/US2009/055542 WO2010039381A1 (en) | 2008-09-30 | 2009-08-31 | Transdermal extended-delivery donepezil compositions and methods for using the same |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0917862A2 true BRPI0917862A2 (pt) | 2015-11-24 |
Family
ID=42057739
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0917862A BRPI0917862A2 (pt) | 2008-09-30 | 2009-08-31 | composições transdérmicas de donepezil com distribuição prolongada e métodos para usar as mesmas |
Country Status (12)
Country | Link |
---|---|
US (1) | US20100080842A1 (pt) |
EP (1) | EP2328582A4 (pt) |
JP (1) | JP2012504163A (pt) |
CN (1) | CN102164601A (pt) |
AR (1) | AR073696A1 (pt) |
AU (1) | AU2009300184A1 (pt) |
BR (1) | BRPI0917862A2 (pt) |
CA (1) | CA2733265A1 (pt) |
IL (1) | IL210970A0 (pt) |
MX (1) | MX2011002260A (pt) |
TW (1) | TW201029653A (pt) |
WO (1) | WO2010039381A1 (pt) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ605352A (en) | 2010-06-30 | 2013-10-25 | Nal Pharmaceuticals Ltd | Process for producing glycosaminoglycans |
JP5850371B2 (ja) * | 2010-09-30 | 2016-02-03 | 積水メディカル株式会社 | 貼付剤 |
TWI433904B (zh) * | 2011-01-12 | 2014-04-11 | Taiwan Biotech Co Ltd | 多奈哌齊經皮貼片 |
WO2013078608A1 (en) * | 2011-11-29 | 2013-06-06 | Ziqiang Gu | Donepezil pamoate and methods of making and using the same |
KR101485822B1 (ko) | 2014-01-22 | 2015-01-23 | 주식회사 대웅제약 | 도네페질 또는 그의 염을 함유하는 경피흡수제제 |
US10195408B2 (en) | 2014-02-20 | 2019-02-05 | Nal Pharmaceutical Group Limited | Transdermal drug delivery system containing donepezil |
KR101796771B1 (ko) * | 2014-12-18 | 2017-11-10 | 아이큐어 주식회사 | 도네페질을 유효성분으로 함유하는 경피흡수제제 |
KR102033686B1 (ko) | 2017-05-19 | 2019-10-18 | 보령제약 주식회사 | 도네페질을 함유하는 마이크로니들 경피 패치 |
CN111818914A (zh) * | 2017-12-13 | 2020-10-23 | 考里安公司 | 透皮药物递送期间创建储库的方法 |
KR102024996B1 (ko) | 2017-12-27 | 2019-09-25 | 동아에스티 주식회사 | 도네페질을 함유하는 치매 치료용 경피흡수제제 |
KR102372630B1 (ko) | 2019-05-15 | 2022-03-14 | 주식회사 대웅제약 | 고함량의 도네페질 또는 그의 염을 포함하는 경피흡수제제 |
CN112823793A (zh) * | 2019-11-20 | 2021-05-21 | 成都康弘药业集团股份有限公司 | 一种含有多奈哌齐的透皮贴剂及其制备方法 |
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DE4341444C2 (de) * | 1993-12-04 | 1996-03-14 | Lohmann Therapie Syst Lts | Wirkstoffhaltiges Pflaster und Verfahren zu seiner Herstellung |
US5536263A (en) * | 1994-03-30 | 1996-07-16 | Lectec Corporation | Non-occulusive adhesive patch for applying medication to the skin |
US5635203A (en) * | 1994-09-29 | 1997-06-03 | Alza Corporation | Transdermal device having decreased delamination |
US5759560A (en) * | 1995-07-27 | 1998-06-02 | Bio Med Sciences, Inc. | Silicone thermoplastic sheeting for scar treatment and useful article thereof; process of manufacture and use |
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US6512010B1 (en) * | 1996-07-15 | 2003-01-28 | Alza Corporation | Formulations for the administration of fluoxetine |
JP2001502693A (ja) * | 1996-10-24 | 2001-02-27 | アルザ コーポレイション | 経皮薬物投与組成物、装置、および方法に適した透過促進剤 |
US7150881B2 (en) * | 1997-06-26 | 2006-12-19 | Mylan Technologies, Inc. | Adhesive mixture for transdermal delivery of highly plasticizing drugs |
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-
2009
- 2009-08-31 BR BRPI0917862A patent/BRPI0917862A2/pt not_active Application Discontinuation
- 2009-08-31 US US12/551,231 patent/US20100080842A1/en not_active Abandoned
- 2009-08-31 WO PCT/US2009/055542 patent/WO2010039381A1/en active Application Filing
- 2009-08-31 EP EP09818191A patent/EP2328582A4/en not_active Withdrawn
- 2009-08-31 AU AU2009300184A patent/AU2009300184A1/en not_active Abandoned
- 2009-08-31 CA CA2733265A patent/CA2733265A1/en not_active Abandoned
- 2009-08-31 MX MX2011002260A patent/MX2011002260A/es not_active Application Discontinuation
- 2009-08-31 JP JP2011530087A patent/JP2012504163A/ja active Pending
- 2009-08-31 CN CN200980138160XA patent/CN102164601A/zh active Pending
- 2009-09-28 AR ARP090103720A patent/AR073696A1/es not_active Application Discontinuation
- 2009-09-29 TW TW098132814A patent/TW201029653A/zh unknown
-
2011
- 2011-01-31 IL IL210970A patent/IL210970A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
AR073696A1 (es) | 2010-11-24 |
CN102164601A (zh) | 2011-08-24 |
US20100080842A1 (en) | 2010-04-01 |
TW201029653A (en) | 2010-08-16 |
JP2012504163A (ja) | 2012-02-16 |
MX2011002260A (es) | 2011-04-07 |
WO2010039381A1 (en) | 2010-04-08 |
IL210970A0 (en) | 2011-04-28 |
EP2328582A1 (en) | 2011-06-08 |
CA2733265A1 (en) | 2010-04-08 |
EP2328582A4 (en) | 2012-02-22 |
AU2009300184A1 (en) | 2010-04-08 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |