CA2651811A1 - Method for increasing the bioavailability of benzhydryl piperazine containing compounds - Google Patents

Method for increasing the bioavailability of benzhydryl piperazine containing compounds Download PDF

Info

Publication number
CA2651811A1
CA2651811A1 CA002651811A CA2651811A CA2651811A1 CA 2651811 A1 CA2651811 A1 CA 2651811A1 CA 002651811 A CA002651811 A CA 002651811A CA 2651811 A CA2651811 A CA 2651811A CA 2651811 A1 CA2651811 A1 CA 2651811A1
Authority
CA
Canada
Prior art keywords
phenyl
compound
piperazine
food
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002651811A
Other languages
English (en)
French (fr)
Inventor
Terrance P. Snutch
Dennis M. Fisher
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Taro Pharmaceuticals Inc
Original Assignee
Neuromed Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neuromed Pharmaceuticals Ltd filed Critical Neuromed Pharmaceuticals Ltd
Publication of CA2651811A1 publication Critical patent/CA2651811A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA002651811A 2006-05-11 2007-05-04 Method for increasing the bioavailability of benzhydryl piperazine containing compounds Abandoned CA2651811A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US79933406P 2006-05-11 2006-05-11
US60/799,334 2006-05-11
PCT/US2007/010846 WO2007133481A2 (en) 2006-05-11 2007-05-04 Method for increasing the bioavailability of benzhydryl piperazine containing compounds

Publications (1)

Publication Number Publication Date
CA2651811A1 true CA2651811A1 (en) 2007-11-22

Family

ID=38694401

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002651811A Abandoned CA2651811A1 (en) 2006-05-11 2007-05-04 Method for increasing the bioavailability of benzhydryl piperazine containing compounds

Country Status (4)

Country Link
US (1) US8362021B2 (de)
EP (1) EP2019676A2 (de)
CA (1) CA2651811A1 (de)
WO (1) WO2007133481A2 (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9492439B2 (en) 2010-03-11 2016-11-15 New York University Amido compounds as RORγt modulators and uses thereof
US8409560B2 (en) 2011-03-08 2013-04-02 Zalicus Pharmaceuticals Ltd. Solid dispersion formulations and methods of use thereof
JP2014507424A (ja) * 2011-03-08 2014-03-27 ザリカス ファーマスーティカルズ リミテッド 固体分散物製剤およびその使用方法
JP6258867B2 (ja) * 2012-01-25 2018-01-10 ノバルティス アーゲー 複素環式化合物およびその使用方法
WO2017223231A1 (en) * 2016-06-21 2017-12-28 Alios Biopharma, Inc. (s)-8-(benzhydryl )-6-isopropyl-3,5-dioxo- 5, 6,7,8,-tetrahydro-3h-pyrazino-[1,2-b]pyridazin-yl-isobutyrate antiviral agent for use in treating influenza
CN111100097A (zh) * 2019-12-04 2020-05-05 中国科学院高能物理研究所 二芳基甲烷类化合物及其制备方法

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Also Published As

Publication number Publication date
WO2007133481A3 (en) 2008-01-24
US20090312346A1 (en) 2009-12-17
EP2019676A2 (de) 2009-02-04
WO2007133481A2 (en) 2007-11-22
US8362021B2 (en) 2013-01-29

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Legal Events

Date Code Title Description
FZDE Discontinued