CA2540460A1 - Composes heterocycliques, leurs procedes de fabrication et leur utilisation - Google Patents
Composes heterocycliques, leurs procedes de fabrication et leur utilisation Download PDFInfo
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- CA2540460A1 CA2540460A1 CA002540460A CA2540460A CA2540460A1 CA 2540460 A1 CA2540460 A1 CA 2540460A1 CA 002540460 A CA002540460 A CA 002540460A CA 2540460 A CA2540460 A CA 2540460A CA 2540460 A1 CA2540460 A1 CA 2540460A1
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- halogen
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-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
- C07D239/90—Oxygen atoms with acyclic radicals attached in position 2 or 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/22—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
- C07D311/26—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4 with aromatic rings attached in position 2 or 3
- C07D311/28—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4 with aromatic rings attached in position 2 or 3 with aromatic rings attached in position 2 only
- C07D311/30—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4 with aromatic rings attached in position 2 or 3 with aromatic rings attached in position 2 only not hydrogenated in the hetero ring, e.g. flavones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Cardiology (AREA)
- Immunology (AREA)
- Neurology (AREA)
- Pulmonology (AREA)
- Physical Education & Sports Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
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- Obesity (AREA)
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- Urology & Nephrology (AREA)
- Emergency Medicine (AREA)
- Oncology (AREA)
- Transplantation (AREA)
- Ophthalmology & Optometry (AREA)
- Gastroenterology & Hepatology (AREA)
- Psychiatry (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN861/CHE/2003 | 2003-10-28 | ||
| IN861CH2003 | 2003-10-28 | ||
| US61016304P | 2004-09-15 | 2004-09-15 | |
| US60/610,163 | 2004-09-15 | ||
| PCT/US2004/035939 WO2005042712A2 (fr) | 2003-10-28 | 2004-10-28 | Composes heterocycliques, leurs procedes de fabrication et leur utilisation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2540460A1 true CA2540460A1 (fr) | 2005-05-12 |
Family
ID=34553826
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002540460A Abandoned CA2540460A1 (fr) | 2003-10-28 | 2004-10-28 | Composes heterocycliques, leurs procedes de fabrication et leur utilisation |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP1678157A4 (fr) |
| JP (2) | JP2007509966A (fr) |
| KR (1) | KR20070026306A (fr) |
| AU (1) | AU2004286277A1 (fr) |
| CA (1) | CA2540460A1 (fr) |
| IL (1) | IL174249A0 (fr) |
| NO (1) | NO20061292L (fr) |
| RU (1) | RU2006112343A (fr) |
| WO (1) | WO2005042712A2 (fr) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2007509966A (ja) * | 2003-10-28 | 2007-04-19 | レディ ユーエス セラピューティックス， インコーポレイテッド | 複素環化合物およびそれらを製造し使用する方法 |
| AU2006275514B2 (en) | 2005-07-29 | 2012-04-05 | Resverlogix Corp. | Pharmaceutical compositions for the prevention and treatment of complex diseases and their delivery by insertable medical devices |
| CA2676984C (fr) | 2007-02-01 | 2015-03-17 | Resverlogix Corp. | Composes destines a la prevention et au traitement de maladies cardiovasculaires |
| ES2542835T3 (es) | 2009-01-08 | 2015-08-12 | Resverlogix Corporation | Compuestos para la prevención y el tratamiento de enfermedades cardiovasculares |
| JP5795304B2 (ja) | 2009-03-18 | 2015-10-14 | レスバーロジックス コーポレイション | 新規抗炎症剤 |
| KR101892987B1 (ko) | 2009-04-22 | 2018-08-30 | 리스버로직스 코퍼레이션 | 신규한 소염제 |
| CZ2009358A3 (cs) * | 2009-06-03 | 2010-12-15 | C3 Bio Gmbh | 5,7-Disubstituované 3-isopropylpyrazolo[4,3-d]pyrimidiny pro použití jako lécivo a farmaceutické prípravky tyto látky obsahující |
| US9101564B2 (en) | 2009-09-30 | 2015-08-11 | Shiseido Company, Ltd. | Heparanase activity inhibitor, wrinkle improving agent containing same, and pharmaceutical composition |
| CA2851996C (fr) | 2011-11-01 | 2020-01-07 | Resverlogix Corp. | Compositions pharmaceutiques pour des quinazolinones substituees |
| WO2014080290A2 (fr) | 2012-11-21 | 2014-05-30 | Rvx Therapeutics Inc. | Amines cycliques servant d'inhibiteurs de bromodomaines |
| WO2014080291A2 (fr) | 2012-11-21 | 2014-05-30 | Rvx Therapeutics Inc. | Dérivés biaryle servant d'inhibiteurs de bromodomaines |
| EP2935253B1 (fr) | 2012-12-21 | 2018-08-01 | Zenith Epigenetics Ltd. | Nouveaux composés hétérocycliques en tant qu'inhibiteurs de bromodomaine |
| CA2977308A1 (fr) | 2015-03-13 | 2016-09-22 | Resverlogix Corp. | Compositions et procedes therapeutiques pour le traitement de maladies associees au complement |
| JP7116422B2 (ja) | 2016-04-05 | 2022-08-10 | イミューン センサー リミテッド ライアビリティ カンパニー | ｃＧＡＳアンタゴニスト化合物 |
| RU2635112C1 (ru) * | 2016-12-12 | 2017-11-09 | федеральное государственное автономное образовательное учреждение высшего образования "Южный федеральный университет" | Галогениды 1-(4-трет-бутилфенил)-2-{ 3-[2-(4-фторфенокси)этил]-2-метил-3Н-бензимидазол-1-ил} этанона, обладающие свойством разрывателей поперечных сшивок гликированных белков |
| EP3897645A4 (fr) * | 2018-12-21 | 2022-08-31 | Acurx Pharmaceuticals, LLC | Inhibiteurs d'adn polymérase iiic et leur utilisation |
| CN112300141B (zh) * | 2020-10-12 | 2023-04-18 | 贵州大学 | 含喹唑啉的杨梅素衍生物、其制备方法及用途 |
| WO2022255765A1 (fr) * | 2021-06-01 | 2022-12-08 | 주식회사 에즈큐리스 | Nouveau dérivé de flavonoïde substitué par du fluor, et composition pharmaceutique pour prévenir ou traiter des maladies allergiques le comprenant |
| EP4426434A1 (fr) | 2021-11-02 | 2024-09-11 | Flare Therapeutics, Inc. | Agonistes inverses de pparg et leurs utilisations |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0739203A4 (fr) * | 1994-01-14 | 2000-12-20 | Cell Therapeutics Inc | Methode de traitement d'affections dues a la proliferation cellulaire en reponse aux pdgf, egf, fgf et vegf |
| JPH09268189A (ja) * | 1996-01-31 | 1997-10-14 | Ss Pharmaceut Co Ltd | ベンゾアジン誘導体又はその塩及びこれを含有する医薬 |
| TW399051B (en) * | 1996-01-31 | 2000-07-21 | Ssp Co Ltd | A novel benzoazine thiazolidinedione derivative and pharmaceutical composition for reducing blood glucose |
| US5885997A (en) * | 1996-07-01 | 1999-03-23 | Dr. Reddy's Research Foundation | Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases |
| BR9711098B1 (pt) * | 1996-07-01 | 2011-10-04 | compostos heterocìclicos, processo para sua preparação e composições farmacêuticas contendo os mesmos e seu uso no tratamento de diabetes e doenças relacionadas. | |
| DK0958296T3 (da) * | 1996-12-31 | 2003-08-18 | Reddys Lab Ltd Dr | Heterocykliske forbindelser, fremgangsmåde til deres fremstilling og farmaceutiske præparater, der indeholder dem, og deres anvendelse i behandlingen af diabetes og beslægtede sygdomme |
| DE69815008T2 (de) * | 1997-09-19 | 2004-04-01 | Ssp Co., Ltd. | Alfa-substituierte Phenylpropionsäurederivate und diese enthaltende Arzneimittel |
| US6028088A (en) * | 1998-10-30 | 2000-02-22 | The University Of Mississippi | Flavonoid derivatives |
| US6608038B2 (en) * | 2000-03-15 | 2003-08-19 | Novartis Ag | Methods and compositions for treatment of diabetes and related conditions via gene therapy |
| JP2007509966A (ja) * | 2003-10-28 | 2007-04-19 | レディ ユーエス セラピューティックス， インコーポレイテッド | 複素環化合物およびそれらを製造し使用する方法 |
-
2004
- 2004-10-28 JP JP2006538290A patent/JP2007509966A/ja active Pending
- 2004-10-28 KR KR1020067005607A patent/KR20070026306A/ko not_active Application Discontinuation
- 2004-10-28 WO PCT/US2004/035939 patent/WO2005042712A2/fr active Application Filing
- 2004-10-28 AU AU2004286277A patent/AU2004286277A1/en not_active Abandoned
- 2004-10-28 EP EP04817481A patent/EP1678157A4/fr not_active Withdrawn
- 2004-10-28 CA CA002540460A patent/CA2540460A1/fr not_active Abandoned
- 2004-10-28 RU RU2006112343/04A patent/RU2006112343A/ru not_active Application Discontinuation
-
2006
- 2006-03-12 IL IL174249A patent/IL174249A0/en unknown
- 2006-03-21 NO NO20061292A patent/NO20061292L/no not_active Application Discontinuation
-
2007
- 2007-10-11 JP JP2007265960A patent/JP2008074858A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| EP1678157A2 (fr) | 2006-07-12 |
| RU2006112343A (ru) | 2007-12-10 |
| WO2005042712A2 (fr) | 2005-05-12 |
| KR20070026306A (ko) | 2007-03-08 |
| JP2008074858A (ja) | 2008-04-03 |
| JP2007509966A (ja) | 2007-04-19 |
| AU2004286277A1 (en) | 2005-05-12 |
| WO2005042712A3 (fr) | 2005-07-21 |
| IL174249A0 (en) | 2006-08-01 |
| NO20061292L (no) | 2006-07-28 |
| EP1678157A4 (fr) | 2009-03-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request | ||
| FZDE | Discontinued |