CA2535953C - Treating bone-related disorders with selective androgen receptor modulators - Google Patents
Treating bone-related disorders with selective androgen receptor modulators Download PDFInfo
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- CA2535953C CA2535953C CA2535953A CA2535953A CA2535953C CA 2535953 C CA2535953 C CA 2535953C CA 2535953 A CA2535953 A CA 2535953A CA 2535953 A CA2535953 A CA 2535953A CA 2535953 C CA2535953 C CA 2535953C
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US61320604P | 2004-09-28 | 2004-09-28 | |
| US60/613,206 | 2004-09-28 | ||
| PCT/US2004/033395 WO2005037201A2 (en) | 2003-10-14 | 2004-10-12 | Treating bone-related disorders with selective androgen receptor modulators |
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| US (1) | US20060019931A1 (enExample) |
| EP (2) | EP1673376A4 (enExample) |
| JP (2) | JP2007508386A (enExample) |
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| AU (1) | AU2004281708B2 (enExample) |
| CA (1) | CA2535953C (enExample) |
| EA (1) | EA013738B1 (enExample) |
| IL (1) | IL172043A0 (enExample) |
| MX (1) | MXPA06002462A (enExample) |
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| US8853266B2 (en) | 2001-12-06 | 2014-10-07 | University Of Tennessee Research Foundation | Selective androgen receptor modulators for treating diabetes |
| US20070161608A1 (en) * | 2001-12-06 | 2007-07-12 | Dalton James T | Selective androgen receptor modulators for treating muscle wasting |
| WO2004035739A2 (en) * | 2002-10-16 | 2004-04-29 | Gtx, Inc. | Treating androgen decline in aging male (adam)-associated conditions with sarms |
| US20060276539A1 (en) * | 2002-10-16 | 2006-12-07 | Dalton James T | Treating Androgen Decline in Aging Male (ADAM)- associated conditions with SARMS |
| US8309603B2 (en) | 2004-06-07 | 2012-11-13 | University Of Tennessee Research Foundation | SARMs and method of use thereof |
| CA2543827C (en) * | 2004-06-07 | 2010-03-09 | James T. Dalton | Selective androgen receptor modulators and methods of use thereof |
| US20110237664A1 (en) * | 2004-06-07 | 2011-09-29 | Dalton James T | Selective androgen receptor modulators for treating diabetes |
| US9889110B2 (en) | 2004-06-07 | 2018-02-13 | University Of Tennessee Research Foundation | Selective androgen receptor modulator for treating hormone-related conditions |
| US9884038B2 (en) | 2004-06-07 | 2018-02-06 | University Of Tennessee Research Foundation | Selective androgen receptor modulator and methods of use thereof |
| CA2658394C (en) * | 2006-07-12 | 2016-08-16 | University Of Tennessee Research Foundation | Substituted acylanilides and methods of use thereof |
| PT2054049E (pt) | 2006-08-24 | 2016-06-02 | Univ Tennessee Res Found | Acilanilidas substituídas e métodos de utilização das mesmas |
| US10010521B2 (en) | 2006-08-24 | 2018-07-03 | University Of Tennessee Research Foundation | SARMs and method of use thereof |
| US9730908B2 (en) | 2006-08-24 | 2017-08-15 | University Of Tennessee Research Foundation | SARMs and method of use thereof |
| US9844528B2 (en) | 2006-08-24 | 2017-12-19 | University Of Tennessee Research Foundation | SARMs and method of use thereof |
| EP2205552B1 (en) * | 2007-09-11 | 2018-02-28 | GTx, Inc. | Crystalline polymorph of the selective androgen modulators (r) or (s)-n-(4-cyano-3-(trifluoromethyl)phenyl)-3-(4-cyanophenoxy)-2-hydroxy-2-methylpropanamide |
| US7968603B2 (en) | 2007-09-11 | 2011-06-28 | University Of Tennessee Research Foundation | Solid forms of selective androgen receptor modulators |
| US8395552B2 (en) | 2010-11-23 | 2013-03-12 | Metamagnetics, Inc. | Antenna module having reduced size, high gain, and increased power efficiency |
| WO2013152170A1 (en) * | 2012-04-04 | 2013-10-10 | Catylix, Inc. | Selective androgen receptor modulators |
| IN2015DN01046A (enExample) | 2012-07-13 | 2015-06-26 | Gtx Inc | |
| US9969683B2 (en) | 2012-07-13 | 2018-05-15 | Gtx, Inc. | Method of treating estrogen receptor (ER)-positive breast cancers with selective androgen receptor modulator (SARMS) |
| US10987334B2 (en) | 2012-07-13 | 2021-04-27 | University Of Tennessee Research Foundation | Method of treating ER mutant expressing breast cancers with selective androgen receptor modulators (SARMs) |
| US10258596B2 (en) | 2012-07-13 | 2019-04-16 | Gtx, Inc. | Method of treating HER2-positive breast cancers with selective androgen receptor modulators (SARMS) |
| US9622992B2 (en) | 2012-07-13 | 2017-04-18 | Gtx, Inc. | Method of treating androgen receptor (AR)-positive breast cancers with selective androgen receptor modulator (SARMs) |
| US10314807B2 (en) | 2012-07-13 | 2019-06-11 | Gtx, Inc. | Method of treating HER2-positive breast cancers with selective androgen receptor modulators (SARMS) |
| US9744149B2 (en) | 2012-07-13 | 2017-08-29 | Gtx, Inc. | Method of treating androgen receptor (AR)-positive breast cancers with selective androgen receptor modulator (SARMs) |
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| LU88769I2 (fr) * | 1982-07-23 | 1996-11-05 | Zeneca Ltd | Bicalutamide et ses sels et esters pharmaceutiquement acceptables (Casodex (R)) |
| US6995284B2 (en) * | 2000-08-24 | 2006-02-07 | The University Of Tennessee Research Foundation | Synthesis of selective androgen receptor modulators |
| WO1998053826A1 (en) * | 1997-05-30 | 1998-12-03 | The University Of Tennessee Research Corporation | Non-steroidal agonist compounds and their use in male hormone therapy |
| US20020022026A1 (en) * | 1998-05-11 | 2002-02-21 | Paz Einat | Genes associated with mechanical stress, expression products therefrom, and uses thereof |
| AU8821301A (en) * | 2000-06-28 | 2002-01-08 | Bristol Myers Squibb Co | Selective androgen receptor modulators and methods for their identification, design and use |
| US20030232792A1 (en) * | 2000-08-24 | 2003-12-18 | Dalton James T. | Selective androgen receptor modulators and methods of use thereof |
| US7026500B2 (en) * | 2000-08-24 | 2006-04-11 | University Of Tennessee Research Foundation | Halogenated selective androgen receptor modulators and methods of use thereof |
| IL154425A0 (en) * | 2000-08-24 | 2003-09-17 | Univ Tennessee Res H Corp | Selective androgen receptor modulators and methods of use thereof |
| AU2001285230C1 (en) * | 2000-08-24 | 2008-03-13 | University Of Tennessee Research Foundation | Selective androgen receptor modulators and methods of use thereof |
| US6838484B2 (en) * | 2000-08-24 | 2005-01-04 | University Of Tennessee Research Foundation | Formulations comprising selective androgen receptor modulators |
| US6777427B2 (en) * | 2000-09-14 | 2004-08-17 | Kaken Pharmaceutical Co., Ltd. | Tetrahydroquinoline compounds |
| US20030022868A1 (en) * | 2001-06-25 | 2003-01-30 | Dalton James T. | Selective androgen receptor modulators and methods of use thereof |
| EP1429779A2 (en) * | 2001-09-21 | 2004-06-23 | Merck & Co., Inc. | Androstanes as androgen receptor modulators |
| IL162340A0 (en) * | 2001-12-06 | 2005-11-20 | Gtx Inc | Treating muscle wasting with selective androgen receptor modulators |
| DK1480634T3 (da) * | 2002-02-07 | 2011-11-14 | Univ Tennessee Res Foundation | Selektive androgenreceptormodulatorer (SARM) til behandling af benign prostatahyperplasi |
| CA2478186C (en) * | 2002-03-13 | 2011-08-23 | Merck & Co., Inc. | Fluorinated 4-azasteroid derivatives as androgen receptor modulators |
| WO2004034978A2 (en) * | 2002-10-15 | 2004-04-29 | Gtx, Inc. | Treating obesity with selective androgen receptor modulators |
| WO2004035739A2 (en) * | 2002-10-16 | 2004-04-29 | Gtx, Inc. | Treating androgen decline in aging male (adam)-associated conditions with sarms |
| PT1592658E (pt) * | 2003-01-13 | 2013-06-25 | Univ Tennessee Res Foundation | Síntese em larga escala de modulador selectivo de receptor de androgénio |
| CA2514024A1 (en) * | 2003-01-22 | 2004-08-05 | Gtx Inc. | Treating androgen deficiency in female (adif)-associated conditions with sarms |
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| CN101721402B (zh) | 2013-03-13 |
| WO2005037201A2 (en) | 2005-04-28 |
| EP1673376A2 (en) | 2006-06-28 |
| CN101721402A (zh) | 2010-06-09 |
| EP2476415A3 (en) | 2012-08-29 |
| JP2010280733A (ja) | 2010-12-16 |
| IL172043A0 (en) | 2009-02-11 |
| JP2007508386A (ja) | 2007-04-05 |
| EP2476415A2 (en) | 2012-07-18 |
| AU2004281708B2 (en) | 2011-02-17 |
| WO2005037201A3 (en) | 2005-10-06 |
| AU2004281708A1 (en) | 2005-04-28 |
| EA200600228A1 (ru) | 2006-08-25 |
| MXPA06002462A (es) | 2006-06-20 |
| CA2535953A1 (en) | 2005-04-28 |
| EP1673376A4 (en) | 2010-06-23 |
| US20060019931A1 (en) | 2006-01-26 |
| EA013738B1 (ru) | 2010-06-30 |
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| EEER | Examination request | ||
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