CA2438210A1 - Steroid compounds, use of these compounds for the preparation of meiosis-regulating medicaments and method for the preparation of these compounds - Google Patents

Steroid compounds, use of these compounds for the preparation of meiosis-regulating medicaments and method for the preparation of these compounds Download PDF

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Publication number
CA2438210A1
CA2438210A1 CA002438210A CA2438210A CA2438210A1 CA 2438210 A1 CA2438210 A1 CA 2438210A1 CA 002438210 A CA002438210 A CA 002438210A CA 2438210 A CA2438210 A CA 2438210A CA 2438210 A1 CA2438210 A1 CA 2438210A1
Authority
CA
Canada
Prior art keywords
pregna
methyl
beta
cndot
dien
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002438210A
Other languages
English (en)
French (fr)
Inventor
Thorsten Blume
Peter Esperling
Christa Hegele-Hartung
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Schering AG
Novo Nordisk AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering AG, Novo Nordisk AS filed Critical Schering AG
Publication of CA2438210A1 publication Critical patent/CA2438210A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of only two carbon atoms, e.g. pregnane derivatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA002438210A 2001-03-26 2002-03-20 Steroid compounds, use of these compounds for the preparation of meiosis-regulating medicaments and method for the preparation of these compounds Abandoned CA2438210A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP01250108A EP1245572A1 (en) 2001-03-26 2001-03-26 Aminosterol compounds, their use in the preparation of meiosis-regulating medicaments and method for their preparation
EP01250108.6 2001-03-26
PCT/EP2002/003148 WO2002079220A2 (en) 2001-03-26 2002-03-20 Aminosterol compounds, their use in the preparation of meiosis-regulating medicaments and method for their preparation

Publications (1)

Publication Number Publication Date
CA2438210A1 true CA2438210A1 (en) 2002-10-10

Family

ID=8181575

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002438210A Abandoned CA2438210A1 (en) 2001-03-26 2002-03-20 Steroid compounds, use of these compounds for the preparation of meiosis-regulating medicaments and method for the preparation of these compounds

Country Status (18)

Country Link
US (1) US6916921B2 (https=)
EP (2) EP1245572A1 (https=)
JP (1) JP2004534011A (https=)
KR (1) KR20030088043A (https=)
CN (1) CN1332975C (https=)
AU (1) AU2002315260B2 (https=)
BR (1) BR0208381A (https=)
CA (1) CA2438210A1 (https=)
CZ (1) CZ20032578A3 (https=)
HU (1) HUP0303643A2 (https=)
IL (1) IL157272A0 (https=)
MX (1) MXPA03008199A (https=)
NO (1) NO20034273L (https=)
PL (1) PL369576A1 (https=)
RU (1) RU2289587C2 (https=)
UA (1) UA75130C2 (https=)
WO (1) WO2002079220A2 (https=)
ZA (1) ZA200308271B (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1514874A1 (en) * 2003-07-28 2005-03-16 Schering Aktiengesellschaft Thiomorpholino steroid compounds, the use thereof for the preparation of meiosis regulating medicaments and method for the preparation thereof
KR100689260B1 (ko) * 2005-05-24 2007-03-02 삼원산업주식회사 항산화성 스틸벤계 형광증백제 및 이의 합성방법

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1095167A (en) * 1963-12-05 1967-12-13 Shalom Sarel Amino-steroids
US3419661A (en) * 1964-01-13 1968-12-31 Univ Missouri Oral contraceptive for birds
DE1643004A1 (de) * 1967-02-07 1971-04-08 Schering Ag Bisnorcholenderivate und Verfahren zu ihrer Herstellung
DE1930473A1 (de) * 1969-06-14 1970-12-17 Schering Ag 22-N-substituierte (20R)-23,24-dinor-cholanderivate
US5716777A (en) 1994-06-23 1998-02-10 Novo Nordisk A/S Regulation of meiosis using sterols
HUP9800731A3 (en) * 1995-03-06 2000-03-28 Novo Nordisk As Stimulation of meiosis
CA2224866A1 (en) 1995-06-23 1997-01-09 Novo Nordisk A/S Meiosis regulating compounds
JP2001506656A (ja) 1996-12-20 2001-05-22 ノボ ノルディスク アクティーゼルスカブ 減数分裂調節化合物
WO1999058549A1 (en) * 1998-05-13 1999-11-18 Novo Nordisk A/S Meiosis regulating compounds
EP1098652A2 (en) 1998-05-26 2001-05-16 Schering Aktiengesellschaft Treatment of infertility with camp-increasing compounds alone or in combination with at least one meiosis-stimulating compound
CN1353617A (zh) 1999-02-24 2002-06-12 诺沃挪第克公司 不孕症的治疗
AU2794000A (en) 1999-02-24 2000-09-14 Novo Nordisk A/S Treatment of infertility
CZ20012671A3 (cs) 1999-02-26 2002-01-16 Novo Nordisk A/S Způsob in vitro oplodnění s pouľitím kultivačního média obsahujícího sterol aktivující meiosu
CA2382908A1 (en) 1999-09-16 2001-03-22 Novo Nordisk A/S Composition for ivf
WO2001062260A2 (en) 2000-02-25 2001-08-30 Schering Aktiengesellschaft Improvement of implantation rate
ATE386495T1 (de) * 2001-02-06 2008-03-15 Novo Nordisk As Behältnis mit niedrigem sauerstoffgehalt, das ff- mas enthält
US6988613B2 (en) * 2001-02-06 2006-01-24 Novo Nordisk A/S Composition for IVF

Also Published As

Publication number Publication date
RU2003130228A (ru) 2005-04-10
ZA200308271B (en) 2005-01-24
PL369576A1 (en) 2005-05-02
IL157272A0 (en) 2004-02-19
JP2004534011A (ja) 2004-11-11
WO2002079220A2 (en) 2002-10-10
NO20034273L (no) 2003-11-25
NO20034273D0 (no) 2003-09-25
CZ20032578A3 (cs) 2003-12-17
UA75130C2 (en) 2006-03-15
CN1332975C (zh) 2007-08-22
US6916921B2 (en) 2005-07-12
EP1245572A1 (en) 2002-10-02
AU2002315260B2 (en) 2008-04-03
HUP0303643A2 (hu) 2004-03-01
WO2002079220A3 (en) 2003-10-16
CN1543473A (zh) 2004-11-03
MXPA03008199A (es) 2004-01-29
US20020188143A1 (en) 2002-12-12
KR20030088043A (ko) 2003-11-15
HK1070900A1 (en) 2005-06-30
RU2289587C2 (ru) 2006-12-20
EP1401856A2 (en) 2004-03-31
BR0208381A (pt) 2004-06-15

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued