CA2269910A1 - New process for the preparation of morphinans - Google Patents
New process for the preparation of morphinans Download PDFInfo
- Publication number
- CA2269910A1 CA2269910A1 CA002269910A CA2269910A CA2269910A1 CA 2269910 A1 CA2269910 A1 CA 2269910A1 CA 002269910 A CA002269910 A CA 002269910A CA 2269910 A CA2269910 A CA 2269910A CA 2269910 A1 CA2269910 A1 CA 2269910A1
- Authority
- CA
- Canada
- Prior art keywords
- aryl
- compound
- formula
- cyclopropylmethyl
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/SE1996/001497 WO1998022467A1 (en) | 1996-11-19 | 1996-11-19 | New process for the preparation of morphinans |
Publications (1)
Publication Number | Publication Date |
---|---|
CA2269910A1 true CA2269910A1 (en) | 1998-05-28 |
Family
ID=20402270
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002269910A Abandoned CA2269910A1 (en) | 1996-11-19 | 1996-11-19 | New process for the preparation of morphinans |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP0946564A1 (ja) |
JP (1) | JP2001504829A (ja) |
AU (1) | AU1402497A (ja) |
CA (1) | CA2269910A1 (ja) |
WO (1) | WO1998022467A1 (ja) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE19939044A1 (de) * | 1999-08-18 | 2001-03-15 | Gruenenthal Gmbh | Verwendung von Morphinanderivaten als Arzneimittel |
WO2011154827A2 (en) * | 2010-06-11 | 2011-12-15 | Rhodes Technologies | Transition metal-catalyzed processes for the preparation of n-allyl compounds and use thereof |
US10800516B2 (en) | 2017-06-02 | 2020-10-13 | The Boeing Company | Semi-levered shrink landing gear |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3412727A1 (de) * | 1984-04-04 | 1985-10-17 | Helmut Dr. Innsbruck Schmidhammer | 14-alkoxy-n-methylmorphinan-6-one, verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel |
US5223507A (en) * | 1992-01-21 | 1993-06-29 | G. D. Searle & Co. | Method of using opioid compounds as delta opioid selective agonist analgesics |
US5225417A (en) * | 1992-01-21 | 1993-07-06 | G. D. Searle & Co. | Opioid agonist compounds |
US5354863A (en) * | 1992-01-21 | 1994-10-11 | G. D. Searle & Co. | Opioid agonist compounds |
SE9401728D0 (sv) * | 1994-05-18 | 1994-05-18 | Astra Ab | New compounds II |
-
1996
- 1996-11-19 WO PCT/SE1996/001497 patent/WO1998022467A1/en not_active Application Discontinuation
- 1996-11-19 CA CA002269910A patent/CA2269910A1/en not_active Abandoned
- 1996-11-19 AU AU14024/97A patent/AU1402497A/en not_active Abandoned
- 1996-11-19 EP EP96944151A patent/EP0946564A1/en not_active Withdrawn
- 1996-11-19 JP JP52353998A patent/JP2001504829A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
EP0946564A1 (en) | 1999-10-06 |
AU1402497A (en) | 1998-06-10 |
JP2001504829A (ja) | 2001-04-10 |
WO1998022467A1 (en) | 1998-05-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FZDE | Dead |