CA1202969A - Imidazobenzodiazepines - Google Patents
ImidazobenzodiazepinesInfo
- Publication number
- CA1202969A CA1202969A CA000431129A CA431129A CA1202969A CA 1202969 A CA1202969 A CA 1202969A CA 000431129 A CA000431129 A CA 000431129A CA 431129 A CA431129 A CA 431129A CA 1202969 A CA1202969 A CA 1202969A
- Authority
- CA
- Canada
- Prior art keywords
- oxo
- imidazo
- benzodiazepine
- carboxylate
- signifies
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
- C07D265/26—Two oxygen atoms, e.g. isatoic anhydride
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/32—Oxygen atoms
- C07D209/38—Oxygen atoms in positions 2 and 3, e.g. isatin
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pyrrole Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH446082 | 1982-07-21 | ||
CH4460/82 | 1982-07-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
CA1202969A true CA1202969A (en) | 1986-04-08 |
Family
ID=4276529
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA000431129A Expired CA1202969A (en) | 1982-07-21 | 1983-06-24 | Imidazobenzodiazepines |
Country Status (25)
Country | Link |
---|---|
US (1) | US4489003A (no) |
EP (1) | EP0100906B1 (no) |
JP (1) | JPS5933286A (no) |
KR (1) | KR840005836A (no) |
AT (1) | ATE27160T1 (no) |
AU (1) | AU560286B2 (no) |
BR (1) | BR8303898A (no) |
CA (1) | CA1202969A (no) |
CS (1) | CS246063B2 (no) |
CU (1) | CU21554A3 (no) |
DE (1) | DE3371516D1 (no) |
DK (1) | DK335083A (no) |
ES (4) | ES524280A0 (no) |
FI (1) | FI832654A (no) |
GR (1) | GR79322B (no) |
HU (1) | HU189719B (no) |
IE (1) | IE56121B1 (no) |
IL (1) | IL69242A (no) |
MC (1) | MC1528A1 (no) |
NO (1) | NO832633L (no) |
NZ (1) | NZ204912A (no) |
PH (1) | PH18980A (no) |
PT (1) | PT77063B (no) |
ZA (1) | ZA835147B (no) |
ZW (1) | ZW14383A1 (no) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3587913D1 (de) * | 1984-01-19 | 1994-10-06 | Hoffmann La Roche | Imidazodiazepin-Derivate. |
CA1259612A (en) * | 1985-02-28 | 1989-09-19 | Emilio Kyburz | Imidazodiazepine derivatives |
DK174086D0 (da) * | 1986-04-16 | 1986-04-16 | Ferrosan As | Nye benzodiazepinderivater samt fremgangsmaade til fremstilling af samme |
GB8720414D0 (en) * | 1987-08-28 | 1987-10-07 | Roussel Lab Ltd | Chemical compounds |
CA2015336A1 (en) * | 1989-05-19 | 1990-11-19 | F. Hoffmann-La Roche Ag | Imidazodiazepines for the treatment of neurological symptoms |
IE910939A1 (en) * | 1990-04-13 | 1991-10-23 | Neurosearch As | Use of benzodiazepine compounds |
GB9911152D0 (en) * | 1999-05-14 | 1999-07-14 | Glaxo Group Ltd | Short-acting benzodiazepines |
US7160880B1 (en) | 1999-05-14 | 2007-01-09 | Cenes Limited | Short-acting benzodiazepines |
AU2006276998A1 (en) * | 2005-05-16 | 2007-02-15 | Wisys Technology Foundation, Inc. | Gabaergic agents to treat memory deficits |
KR20150081370A (ko) | 2006-07-10 | 2015-07-13 | 파이온 유케이 리미티드 | 속효형 벤조디아제핀 염 및 이의 중합체 형태 |
KR101589314B1 (ko) | 2007-08-20 | 2016-01-28 | 에보텍 인터내셔널 게엠베하 | 수면 장애의 치료 |
US20090054412A1 (en) * | 2007-08-20 | 2009-02-26 | John Alan Kemp | Treatment of Sleep Disorders |
EP2450039A1 (en) | 2010-11-08 | 2012-05-09 | PAION UK Ltd. | Dosing regimen for sedation with CNS 7056 (Remimazolam) |
AR094963A1 (es) | 2013-03-04 | 2015-09-09 | Ono Pharmaceutical Co | Reacción de oxidación excelente en el índice de conversión |
US20230101747A1 (en) * | 2019-12-06 | 2023-03-30 | Schrödinger, Inc. | Cyclic compounds and methods of using same |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1143728A (en) * | 1979-10-04 | 1983-03-29 | Max Gerecke | Imidazodiazepine derivatives |
CA1173441A (en) * | 1981-02-27 | 1984-08-28 | Hoffmann-La Roche Limited | Imidazodiazepines |
CA1184175A (en) * | 1981-02-27 | 1985-03-19 | Walter Hunkeler | Imidazodiazepines |
CA1185602A (en) * | 1981-02-27 | 1985-04-16 | Emilio Kyburz | Imidazodiazepines |
US4352817A (en) * | 1981-02-27 | 1982-10-05 | Hoffmann-La Roche Inc. | Imidazo-diazepines and their use |
-
1983
- 1983-06-19 MC MC@@@@1648A patent/MC1528A1/xx unknown
- 1983-06-24 CA CA000431129A patent/CA1202969A/en not_active Expired
- 1983-06-24 ZW ZW143/83A patent/ZW14383A1/xx unknown
- 1983-07-14 DE DE8383106920T patent/DE3371516D1/de not_active Expired
- 1983-07-14 US US06/513,571 patent/US4489003A/en not_active Expired - Fee Related
- 1983-07-14 AT AT83106920T patent/ATE27160T1/de not_active IP Right Cessation
- 1983-07-14 ZA ZA835147A patent/ZA835147B/xx unknown
- 1983-07-14 EP EP83106920A patent/EP0100906B1/de not_active Expired
- 1983-07-15 NZ NZ204912A patent/NZ204912A/en unknown
- 1983-07-15 AU AU16888/83A patent/AU560286B2/en not_active Ceased
- 1983-07-15 IL IL69242A patent/IL69242A/xx unknown
- 1983-07-18 HU HU832533A patent/HU189719B/hu unknown
- 1983-07-19 GR GR71965A patent/GR79322B/el unknown
- 1983-07-19 CS CS835419A patent/CS246063B2/cs unknown
- 1983-07-19 KR KR1019830003325A patent/KR840005836A/ko not_active Application Discontinuation
- 1983-07-19 NO NO832633A patent/NO832633L/no unknown
- 1983-07-20 BR BR8303898A patent/BR8303898A/pt unknown
- 1983-07-20 JP JP58131150A patent/JPS5933286A/ja active Pending
- 1983-07-20 IE IE1696/83A patent/IE56121B1/xx unknown
- 1983-07-20 ES ES524280A patent/ES524280A0/es active Granted
- 1983-07-20 PT PT77063A patent/PT77063B/pt unknown
- 1983-07-20 PH PH29251A patent/PH18980A/en unknown
- 1983-07-20 DK DK335083A patent/DK335083A/da not_active Application Discontinuation
- 1983-07-21 CU CU8335935A patent/CU21554A3/es unknown
- 1983-07-21 FI FI832654A patent/FI832654A/fi not_active Application Discontinuation
-
1984
- 1984-03-16 ES ES530673A patent/ES8504805A1/es not_active Expired
- 1984-03-16 ES ES530672A patent/ES530672A0/es active Granted
- 1984-03-16 ES ES530671A patent/ES530671A0/es active Granted
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MKEX | Expiry |