CA1041498A - Benzodiazepine derivatives - Google Patents

Benzodiazepine derivatives

Info

Publication number
CA1041498A
CA1041498A CA063,875A CA63875A CA1041498A CA 1041498 A CA1041498 A CA 1041498A CA 63875 A CA63875 A CA 63875A CA 1041498 A CA1041498 A CA 1041498A
Authority
CA
Canada
Prior art keywords
hydrogen
chloro
lower alkyl
phenyl
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA063,875A
Other languages
English (en)
French (fr)
Inventor
Leo H. Sternbach
Michael E. Derieg
James V. Earley
Rodney I. Fryer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Priority to CA180,793A priority Critical patent/CA974236A/en
Application granted granted Critical
Publication of CA1041498A publication Critical patent/CA1041498A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61H—PHYSICAL THERAPY APPARATUS, e.g. DEVICES FOR LOCATING OR STIMULATING REFLEX POINTS IN THE BODY; ARTIFICIAL RESPIRATION; MASSAGE; BATHING DEVICES FOR SPECIAL THERAPEUTIC OR HYGIENIC PURPOSES OR SPECIFIC PARTS OF THE BODY
    • A61H23/00—Percussion or vibration massage, e.g. using supersonic vibration; Suction-vibration massage; Massage with moving diaphragms
    • A61H23/02—Percussion or vibration massage, e.g. using supersonic vibration; Suction-vibration massage; Massage with moving diaphragms with electric or magnetic drive
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Rehabilitation Therapy (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Harvester Elements (AREA)
CA063,875A 1968-10-18 1969-09-30 Benzodiazepine derivatives Expired CA1041498A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CA180,793A CA974236A (en) 1968-10-18 1973-09-11 Benzodiazepine derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US76890968A 1968-10-18 1968-10-18

Publications (1)

Publication Number Publication Date
CA1041498A true CA1041498A (en) 1978-10-31

Family

ID=25083843

Family Applications (1)

Application Number Title Priority Date Filing Date
CA063,875A Expired CA1041498A (en) 1968-10-18 1969-09-30 Benzodiazepine derivatives

Country Status (20)

Country Link
JP (2) JPS4925278B1 (enExample)
AT (3) AT303747B (enExample)
BE (1) BE740347A (enExample)
BR (1) BR6913309D0 (enExample)
CA (1) CA1041498A (enExample)
CH (2) CH554361A (enExample)
DE (1) DE1952486A1 (enExample)
DK (1) DK149817C (enExample)
ES (1) ES372620A1 (enExample)
FI (1) FI50984C (enExample)
FR (1) FR2021010B1 (enExample)
GB (1) GB1233489A (enExample)
HU (1) HU166865B (enExample)
IE (1) IE34252B1 (enExample)
IL (1) IL33103A (enExample)
MY (1) MY7500083A (enExample)
NL (1) NL156141B (enExample)
NO (1) NO127504B (enExample)
SE (3) SE382983B (enExample)
YU (1) YU34205B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1812252C2 (de) * 1968-11-26 1981-09-24 Sankyo Co., Ltd., Tokyo Benzodiazepinderivate, Verfahren zu ihrer Herstellung und Arzneimittel
CH565180A5 (enExample) * 1970-12-23 1975-08-15 Hoffmann La Roche
FR2403330A1 (fr) * 1977-06-16 1979-04-13 Fabre Sa Pierre Nouveaux derives de benzoyl-2-chloro-4-glycinanilides substitues, leur procede de preparation et leur application en tant que medicaments
AU538998B2 (en) * 1980-06-27 1984-09-06 Wahl Clipper Corp. Cushioned massager

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1812252C2 (de) * 1968-11-26 1981-09-24 Sankyo Co., Ltd., Tokyo Benzodiazepinderivate, Verfahren zu ihrer Herstellung und Arzneimittel

Also Published As

Publication number Publication date
AT303747B (de) 1972-11-15
AT306037B (de) 1973-02-15
CH554361A (de) 1974-09-30
ES372620A1 (es) 1972-03-16
YU34205B (en) 1979-02-28
HU166865B (enExample) 1975-06-28
GB1233489A (enExample) 1971-05-26
JPS4927199B1 (enExample) 1974-07-16
FI50984B (enExample) 1976-05-31
BR6913309D0 (pt) 1973-01-04
DK149817B (da) 1986-10-06
DE1952486C2 (enExample) 1988-06-23
MY7500083A (en) 1975-12-31
DK149817C (da) 1987-04-06
FR2021010B1 (enExample) 1973-07-13
SE7508208L (sv) 1975-07-17
SE420409B (sv) 1981-10-05
IL33103A (en) 1974-06-30
CH562247A5 (enExample) 1975-05-30
IE34252L (en) 1970-04-18
NL156141B (nl) 1978-03-15
SE382983B (sv) 1976-02-23
AT302305B (de) 1972-10-10
DE1952486A1 (de) 1970-04-30
NL6915750A (enExample) 1970-04-21
IE34252B1 (en) 1975-03-19
FI50984C (fi) 1976-09-10
SE398232B (sv) 1977-12-12
YU260469A (en) 1978-06-30
JPS4925278B1 (enExample) 1974-06-28
FR2021010A1 (enExample) 1970-07-17
IL33103A0 (en) 1969-11-30
NO127504B (enExample) 1973-07-02
BE740347A (enExample) 1970-04-16

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