CA1032938A - Pyrido (1,2a)-pyrimidine-derivatives and process for the preparation thereof - Google Patents

Pyrido (1,2a)-pyrimidine-derivatives and process for the preparation thereof

Info

Publication number
CA1032938A
CA1032938A CA196,195A CA196195A CA1032938A CA 1032938 A CA1032938 A CA 1032938A CA 196195 A CA196195 A CA 196195A CA 1032938 A CA1032938 A CA 1032938A
Authority
CA
Canada
Prior art keywords
pyrido
pyrimidine
derivatives
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA196,195A
Other languages
English (en)
French (fr)
Other versions
CA196195S (en
Inventor
Zoltan Meszaros
Istvan Hermecz
Lelle Vasvari
Agnes Horvath
Jozsef Knoll
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Chinoin Private Co Ltd
Original Assignee
Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt filed Critical Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Zrt
Application granted granted Critical
Publication of CA1032938A publication Critical patent/CA1032938A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA196,195A 1973-03-30 1974-03-28 Pyrido (1,2a)-pyrimidine-derivatives and process for the preparation thereof Expired CA1032938A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HUCI1361A HU168014B (fi) 1973-03-30 1973-03-30

Publications (1)

Publication Number Publication Date
CA1032938A true CA1032938A (en) 1978-06-13

Family

ID=10994473

Family Applications (1)

Application Number Title Priority Date Filing Date
CA196,195A Expired CA1032938A (en) 1973-03-30 1974-03-28 Pyrido (1,2a)-pyrimidine-derivatives and process for the preparation thereof

Country Status (20)

Country Link
JP (1) JPS505396A (fi)
AT (1) AT336624B (fi)
BE (1) BE813021A (fi)
CA (1) CA1032938A (fi)
CH (1) CH605940A5 (fi)
CS (1) CS189872B1 (fi)
DD (1) DD110661A1 (fi)
DE (1) DE2414751A1 (fi)
DK (1) DK138327B (fi)
ES (1) ES424758A1 (fi)
FI (1) FI57949C (fi)
FR (1) FR2223036B1 (fi)
GB (1) GB1454312A (fi)
HU (1) HU168014B (fi)
IL (1) IL44417A (fi)
NL (1) NL7403901A (fi)
NO (1) NO140821C (fi)
PL (1) PL93755B1 (fi)
SE (1) SE418087B (fi)
SU (1) SU566524A3 (fi)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU173438B (hu) * 1975-11-27 1979-05-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija novykh proizvodnykh 4-okso-1,6,7,8-/tetragidro-4h-pirido/1,2/pirimidina s zaderzhivajuhhejj vozgoranie aktivnot'ju i protivosvertivajuhhem effektom
HU174693B (hu) * 1976-02-12 1980-03-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija kondensirovannykh proizvodnykh pirimidina
HU174901B (hu) * 1976-06-25 1980-04-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija novykh proizvodnykh pirido/1,2-a/pirimidina
HU178910B (en) * 1977-08-19 1982-07-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines
HU180701B (en) * 1977-12-29 1983-04-29 Chinoin Gyogyszer Es Vegyeszet Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering
HU185925B (en) * 1977-12-29 1985-04-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing compounds with nitrogen bridge head
HU178496B (en) * 1977-12-29 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity
HU179143B (en) * 1977-12-29 1982-08-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydroxy-groops-containing 6,7-dihydro-pyrido-square bracket-1,2-a-square bracket closed-pyrimidin derivatives and esters thereof
AT376675B (de) * 1979-05-08 1984-12-27 Erba Farmitalia Verfahren zum herstellen von neuen substituierten pyrido(1,2-a)pyrimidinen
US4661592A (en) * 1984-06-27 1987-04-28 G. D. Searle & Co. 4H-pyrimido[2,1-a]isoquinolin-4-one derivatives
HU201551B (en) * 1988-02-03 1990-11-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 4-oxo-4h-pyrido(1,2-a)pyrimidine-3-carboxylic acid amide derivatives and pharmaceutical compositions comprising same
JP5419894B2 (ja) * 2008-01-11 2014-02-19 グレンマーク ファーマシューティカルズ， エセ．アー． Ｔｒｐｖ３モジュレーターとしての縮合ピリミジン誘導体

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT286990B (de) * 1966-11-02 1971-01-11 Chinoin Gyogyszer Es Vegyeszet Verfahren zur Herstellung von neuen Homopyrimidazol-Derivaten sowie von deren Salzen

Also Published As

Publication number Publication date
SE418087B (sv) 1981-05-04
DE2414751A1 (de) 1974-10-10
AT336624B (de) 1977-05-10
DD110661A1 (fi) 1975-01-05
ES424758A1 (es) 1976-06-16
GB1454312A (en) 1976-11-03
FR2223036B1 (fi) 1977-05-06
AU6670474A (en) 1975-09-18
IL44417A0 (en) 1974-06-30
FR2223036A1 (fi) 1974-10-25
DK138327B (da) 1978-08-14
PL93755B1 (en) 1977-06-30
NO140821C (no) 1979-11-21
DK138327C (fi) 1979-01-22
NO140821B (no) 1979-08-13
NL7403901A (fi) 1974-10-02
BE813021A (fr) 1974-07-15
NO741125A (no) 1974-10-01
CH605940A5 (fi) 1978-10-13
CS189872B1 (en) 1979-05-31
FI57949B (fi) 1980-07-31
SU566524A3 (ru) 1977-07-25
FI57949C (fi) 1980-11-10
IL44417A (en) 1978-01-31
HU168014B (fi) 1976-02-28
JPS505396A (fi) 1975-01-21
ATA252674A (de) 1976-09-15

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