AT336624B - Verfahren zur herstellung von neuen 4h-pyrido (1,2-a)-pyrimidin-derivaten und deren salzen - Google Patents

Verfahren zur herstellung von neuen 4h-pyrido (1,2-a)-pyrimidin-derivaten und deren salzen

Info

Publication number
AT336624B
AT336624B AT252674A AT252674A AT336624B AT 336624 B AT336624 B AT 336624B AT 252674 A AT252674 A AT 252674A AT 252674 A AT252674 A AT 252674A AT 336624 B AT336624 B AT 336624B
Authority
AT
Austria
Prior art keywords
pyrido
salts
preparation
new
pyrimidine derivatives
Prior art date
Application number
AT252674A
Other languages
German (de)
English (en)
Other versions
ATA252674A (de
Inventor
Zoltan Chem Ing Dr Meszaros
Jozsef Dr Knoll
Istvan Chem Ing Hermecz
Lelle Vasvari
Agnes Chem Ing Horvath
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of ATA252674A publication Critical patent/ATA252674A/de
Application granted granted Critical
Publication of AT336624B publication Critical patent/AT336624B/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT252674A 1973-03-30 1974-03-27 Verfahren zur herstellung von neuen 4h-pyrido (1,2-a)-pyrimidin-derivaten und deren salzen AT336624B (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HUCI1361A HU168014B (fi) 1973-03-30 1973-03-30

Publications (2)

Publication Number Publication Date
ATA252674A ATA252674A (de) 1976-09-15
AT336624B true AT336624B (de) 1977-05-10

Family

ID=10994473

Family Applications (1)

Application Number Title Priority Date Filing Date
AT252674A AT336624B (de) 1973-03-30 1974-03-27 Verfahren zur herstellung von neuen 4h-pyrido (1,2-a)-pyrimidin-derivaten und deren salzen

Country Status (20)

Country Link
JP (1) JPS505396A (fi)
AT (1) AT336624B (fi)
BE (1) BE813021A (fi)
CA (1) CA1032938A (fi)
CH (1) CH605940A5 (fi)
CS (1) CS189872B1 (fi)
DD (1) DD110661A1 (fi)
DE (1) DE2414751A1 (fi)
DK (1) DK138327B (fi)
ES (1) ES424758A1 (fi)
FI (1) FI57949C (fi)
FR (1) FR2223036B1 (fi)
GB (1) GB1454312A (fi)
HU (1) HU168014B (fi)
IL (1) IL44417A (fi)
NL (1) NL7403901A (fi)
NO (1) NO140821C (fi)
PL (1) PL93755B1 (fi)
SE (1) SE418087B (fi)
SU (1) SU566524A3 (fi)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU173438B (hu) * 1975-11-27 1979-05-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija novykh proizvodnykh 4-okso-1,6,7,8-/tetragidro-4h-pirido/1,2/pirimidina s zaderzhivajuhhejj vozgoranie aktivnot'ju i protivosvertivajuhhem effektom
HU174693B (hu) * 1976-02-12 1980-03-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija kondensirovannykh proizvodnykh pirimidina
HU174901B (hu) * 1976-06-25 1980-04-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija novykh proizvodnykh pirido/1,2-a/pirimidina
HU178910B (en) * 1977-08-19 1982-07-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines
HU178496B (en) * 1977-12-29 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity
HU179143B (en) * 1977-12-29 1982-08-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydroxy-groops-containing 6,7-dihydro-pyrido-square bracket-1,2-a-square bracket closed-pyrimidin derivatives and esters thereof
HU185925B (en) * 1977-12-29 1985-04-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing compounds with nitrogen bridge head
HU180701B (en) * 1977-12-29 1983-04-29 Chinoin Gyogyszer Es Vegyeszet Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering
AT376675B (de) * 1979-05-08 1984-12-27 Erba Farmitalia Verfahren zum herstellen von neuen substituierten pyrido(1,2-a)pyrimidinen
US4661592A (en) * 1984-06-27 1987-04-28 G. D. Searle & Co. 4H-pyrimido[2,1-a]isoquinolin-4-one derivatives
HU201551B (en) * 1988-02-03 1990-11-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 4-oxo-4h-pyrido(1,2-a)pyrimidine-3-carboxylic acid amide derivatives and pharmaceutical compositions comprising same
EA018133B1 (ru) * 2008-01-11 2013-05-30 Гленмарк Фармасьютикалс, С.А. Конденсированные пиримидиновые производные как модуляторы trpv3

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT302311B (de) * 1966-11-02 1972-09-15 Chinoin Gyogyszer Es Vegyeszet Verfahren zur herstellung von homopyrimidazol-derivaten und deren saeureadditionssalzen und quaternaeren ammoniumsalzen

Also Published As

Publication number Publication date
DK138327C (fi) 1979-01-22
FR2223036B1 (fi) 1977-05-06
FR2223036A1 (fi) 1974-10-25
SE418087B (sv) 1981-05-04
NO140821C (no) 1979-11-21
FI57949C (fi) 1980-11-10
CH605940A5 (fi) 1978-10-13
DD110661A1 (fi) 1975-01-05
GB1454312A (en) 1976-11-03
PL93755B1 (en) 1977-06-30
SU566524A3 (ru) 1977-07-25
BE813021A (fr) 1974-07-15
IL44417A (en) 1978-01-31
ATA252674A (de) 1976-09-15
NO140821B (no) 1979-08-13
FI57949B (fi) 1980-07-31
IL44417A0 (en) 1974-06-30
CS189872B1 (en) 1979-05-31
HU168014B (fi) 1976-02-28
NO741125A (no) 1974-10-01
DK138327B (da) 1978-08-14
JPS505396A (fi) 1975-01-21
ES424758A1 (es) 1976-06-16
CA1032938A (en) 1978-06-13
NL7403901A (fi) 1974-10-02
AU6670474A (en) 1975-09-18
DE2414751A1 (de) 1974-10-10

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Legal Events

Date Code Title Description
ELJ Ceased due to non-payment of the annual fee