BRPI0916692A2 - processo para a preparação de um composto, e, composto - Google Patents

processo para a preparação de um composto, e, composto

Info

Publication number
BRPI0916692A2
BRPI0916692A2 BRPI0916692A BRPI0916692A BRPI0916692A2 BR PI0916692 A2 BRPI0916692 A2 BR PI0916692A2 BR PI0916692 A BRPI0916692 A BR PI0916692A BR PI0916692 A BRPI0916692 A BR PI0916692A BR PI0916692 A2 BRPI0916692 A2 BR PI0916692A2
Authority
BR
Brazil
Prior art keywords
compound
preparing
Prior art date
Application number
BRPI0916692A
Other languages
English (en)
Inventor
Hans J Sanders
Jeroen Van Rheenen
Josephus H M Lange
Original Assignee
Abbott Healthcare Products Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Healthcare Products Bv filed Critical Abbott Healthcare Products Bv
Publication of BRPI0916692A2 publication Critical patent/BRPI0916692A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BRPI0916692A 2008-08-01 2009-07-30 processo para a preparação de um composto, e, composto BRPI0916692A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08161619 2008-08-01
PCT/EP2009/059844 WO2010012797A2 (en) 2008-08-01 2009-07-30 Synthesis of 3,4-diaryl-4,5-dihydro-(1h)-pyrazole-1- carboxamidine derivatives

Publications (1)

Publication Number Publication Date
BRPI0916692A2 true BRPI0916692A2 (pt) 2016-05-17

Family

ID=40380031

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0916692A BRPI0916692A2 (pt) 2008-08-01 2009-07-30 processo para a preparação de um composto, e, composto

Country Status (12)

Country Link
EP (1) EP2321280A2 (pt)
JP (1) JP2011529868A (pt)
KR (1) KR20110042095A (pt)
CN (1) CN102089284A (pt)
AR (1) AR072539A1 (pt)
AU (1) AU2009275838A1 (pt)
BR (1) BRPI0916692A2 (pt)
CA (1) CA2729969A1 (pt)
EA (1) EA201170284A1 (pt)
MX (1) MX2011001211A (pt)
TW (1) TW201010981A (pt)
WO (1) WO2010012797A2 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR079935A1 (es) * 2010-01-29 2012-02-29 Abbott Healthcare Products Bv Sintesis de derivados de pirazolin carboxamidina sustituida
US20220227714A1 (en) * 2019-05-17 2022-07-21 The United States Of America,As Represented By The Secretary,Department Of Health And Human Services A scalable synthesis of dual-target inhibitor of cannabinoid-1 receptor and inducible nitric oxide synthase
CN111686806B (zh) * 2020-05-29 2022-09-30 黑龙江大学 一种聚[2-(3-噻吩基)乙醇]/石墨相氮化碳复合可见光催化剂的制备方法及应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5369121A (en) * 1990-01-31 1994-11-29 E. I. Du Pont De Nemours And Company Arthropodicidal pyrazolines, pyrazolidines and hydrazines
DE4005114A1 (de) * 1990-02-17 1991-08-22 Bayer Ag Substituierte pyrazolinderivate
ATE346047T1 (de) * 2000-03-23 2006-12-15 Solvay Pharm Bv 4,5-dihydro-1h-pyrazolderivate mit cb1- antagonistischer aktivität
UA77441C2 (en) * 2001-09-21 2006-12-15 4,5-dihydro-1h-pyrazole derivatives as potent cb1 receptor antagonists, methods for their preparation (variants), intermediate, pharmaceutical composition and method for its preparation

Also Published As

Publication number Publication date
EA201170284A1 (ru) 2011-06-30
WO2010012797A2 (en) 2010-02-04
EP2321280A2 (en) 2011-05-18
JP2011529868A (ja) 2011-12-15
CN102089284A (zh) 2011-06-08
WO2010012797A3 (en) 2010-04-22
MX2011001211A (es) 2011-03-29
TW201010981A (en) 2010-03-16
AR072539A1 (es) 2010-09-01
AU2009275838A1 (en) 2010-02-04
KR20110042095A (ko) 2011-04-22
CA2729969A1 (en) 2010-02-04

Similar Documents

Publication Publication Date Title
BRPI0910910A2 (pt) processo para preparar um composto
BRPI0910911A2 (pt) processo para preparar um composto
BRPI1014547A2 (pt) composto, e, processo para preparar um composto.
BRPI0911254A2 (pt) processo para a preparação de um composto
BRPI0812054A2 (pt) Processo para preparar compostos, e, compostos.
BRPI0908252A2 (pt) Processo para preparar um composto, e, uso de um composto
BRPI0814980A2 (pt) Processo para produzir um composto, e, composto.
BRPI0911898A2 (pt) processo para preparar compostos, e, composto.
BRPI1011888A2 (pt) processo para preparar um composto, e, composição.
BRPI1012018A2 (pt) processo para preparar um composto
BRPI0810067A2 (pt) Processo para a preparação de capecitabina
BRPI0816911A2 (pt) Processo para preparação de 4-aminobut-2-enolidas
BRPI0812422A2 (pt) Processo de preparação de um aldeído hidroxiaromático
BRPI0914674A2 (pt) processo para preparação de um pó
BRPI0911897A2 (pt) Processo para a preparação de compostos, e, composto
BRPI0813772A2 (pt) Composto, processo para a preparação de um composto, e, conjugado
BRPI0815784A2 (pt) Processo para a preparação de 1,2-propanodiol
BRPI0921882A2 (pt) processo para fabricar um composto.
BRPI0810216A2 (pt) Processo para a preparação de composto, composto, e, método de tratamento de distúrbio bipolar
BRPI0909280A2 (pt) processo para preparar uretanos.
BRPI1014691A2 (pt) Composto, e, processo para a preparação de um composto.
BRPI0912558A2 (pt) Processo para a preparação de amidas
BRPI0921420A2 (pt) processo para preparar compostos
BRPI0811315A2 (pt) Processo para a preparação de um composto
BRPI0911992A2 (pt) processo para preparação de bifenilanilidas substituídas

Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired