BRPI0718351A2 - "processo para a preparação do enantiômero s ou r, processo para formar um composto r ou s, uso de um catalisador quiral, composto, sal tartrato do enantiômero s ou r de um composto, complexo de metal de transição e catalisador" - Google Patents
"processo para a preparação do enantiômero s ou r, processo para formar um composto r ou s, uso de um catalisador quiral, composto, sal tartrato do enantiômero s ou r de um composto, complexo de metal de transição e catalisador"Info
- Publication number
- BRPI0718351A2 BRPI0718351A2 BRPI0718351A BRPI0718351A BRPI0718351A2 BR PI0718351 A2 BRPI0718351 A2 BR PI0718351A2 BR PI0718351 A BRPI0718351 A BR PI0718351A BR PI0718351 A BRPI0718351 A BR PI0718351A BR PI0718351 A2 BRPI0718351 A2 BR PI0718351A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- enantiomer
- catalyst
- preparing
- forming
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 3
- 239000003054 catalyst Substances 0.000 title 2
- 238000004519 manufacturing process Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 150000003892 tartrate salts Chemical class 0.000 title 1
- 229910052723 transition metal Inorganic materials 0.000 title 1
- 150000003624 transition metals Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Catalysts (AREA)
- Pyrane Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US86960506P | 2006-12-12 | 2006-12-12 | |
PCT/GB2007/004756 WO2008071951A2 (en) | 2006-12-12 | 2007-12-12 | Catalytic process for asymmetric hydrogenation |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0718351A2 true BRPI0718351A2 (pt) | 2019-09-24 |
Family
ID=39247380
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0718351A BRPI0718351A2 (pt) | 2006-12-12 | 2007-12-12 | "processo para a preparação do enantiômero s ou r, processo para formar um composto r ou s, uso de um catalisador quiral, composto, sal tartrato do enantiômero s ou r de um composto, complexo de metal de transição e catalisador" |
Country Status (15)
Country | Link |
---|---|
US (1) | US8546571B2 (pt) |
EP (1) | EP2102182B1 (pt) |
JP (1) | JP5372771B2 (pt) |
KR (1) | KR20090091326A (pt) |
CN (1) | CN101627023A (pt) |
AR (1) | AR064308A1 (pt) |
AU (1) | AU2007331340A1 (pt) |
BR (1) | BRPI0718351A2 (pt) |
CA (1) | CA2671830C (pt) |
ES (1) | ES2483718T3 (pt) |
MX (1) | MX2009006113A (pt) |
NO (1) | NO20092259L (pt) |
PT (1) | PT103901B (pt) |
RU (1) | RU2009126571A (pt) |
WO (1) | WO2008071951A2 (pt) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MX2009006113A (es) | 2006-12-12 | 2009-07-17 | Bial Portela & Ca Sa | Proceso catalitico para hidrogenacion asimetrica. |
GB0709695D0 (en) * | 2007-05-21 | 2007-06-27 | Portela & Ca Sa | Process |
TW200927740A (en) * | 2007-11-13 | 2009-07-01 | Bial Portela & Ca Sa | Process |
AR070841A1 (es) * | 2008-03-13 | 2010-05-05 | Bial Portela & Ca Sa | Proceso de hidrogenacion catalitica asimetrica |
WO2009116883A2 (en) * | 2008-03-19 | 2009-09-24 | Bial - Portela & Ca., S. A, | Catalytic asymetric hydrogenation |
AR071632A1 (es) | 2008-05-06 | 2010-06-30 | Bial Portela & Ca Sa | Proceso catalitico para hidrogenacion asimetrica en la sintesis de inhibidores de la dopamina-beta-hidroxilasa" |
CN111196759B (zh) * | 2018-11-16 | 2023-03-24 | 上海博志研新药物技术有限公司 | 盐酸西那卡塞及其中间体的制备方法 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5202474A (en) | 1989-06-22 | 1993-04-13 | Monsanto Company | Asymmetric catalytic hydrogenation of α-arylpropenoic acids |
US5420151A (en) | 1989-12-22 | 1995-05-30 | Aktiebolaget Astra | Chroman derivatives |
EP0757677B1 (en) | 1994-04-26 | 2003-06-18 | Syntex (U.S.A.) LLC | Benzocyclohexylimidazolethione derivatives |
US5886182A (en) * | 1997-12-10 | 1999-03-23 | The Hong Kong Polytechnic University | Chiral pyridylphosphines and their application in asymmetric catalytic hydrogenation of 2-arylpropenoic acids |
US7125904B2 (en) * | 2002-10-11 | 2006-10-24 | Portela & C.A., S.A. | Peripherally-selective inhibitors of dopamine-β-hydroxylase and method of their preparation |
GB0316439D0 (en) * | 2003-07-15 | 2003-08-20 | Johnson Matthey Plc | Catalysts |
MX2009006113A (es) | 2006-12-12 | 2009-07-17 | Bial Portela & Ca Sa | Proceso catalitico para hidrogenacion asimetrica. |
-
2007
- 2007-12-12 MX MX2009006113A patent/MX2009006113A/es not_active Application Discontinuation
- 2007-12-12 CN CN200780051168A patent/CN101627023A/zh active Pending
- 2007-12-12 AR ARP070105572A patent/AR064308A1/es unknown
- 2007-12-12 JP JP2009540851A patent/JP5372771B2/ja not_active Expired - Fee Related
- 2007-12-12 PT PT103901A patent/PT103901B/pt active IP Right Grant
- 2007-12-12 US US12/518,416 patent/US8546571B2/en active Active
- 2007-12-12 ES ES07848500.0T patent/ES2483718T3/es active Active
- 2007-12-12 EP EP07848500.0A patent/EP2102182B1/en not_active Not-in-force
- 2007-12-12 CA CA2671830A patent/CA2671830C/en active Active
- 2007-12-12 WO PCT/GB2007/004756 patent/WO2008071951A2/en active Application Filing
- 2007-12-12 AU AU2007331340A patent/AU2007331340A1/en not_active Abandoned
- 2007-12-12 RU RU2009126571/04A patent/RU2009126571A/ru not_active Application Discontinuation
- 2007-12-12 KR KR1020097014315A patent/KR20090091326A/ko not_active Application Discontinuation
- 2007-12-12 BR BRPI0718351A patent/BRPI0718351A2/pt not_active IP Right Cessation
-
2009
- 2009-06-11 NO NO20092259A patent/NO20092259L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EP2102182B1 (en) | 2014-04-23 |
NO20092259L (no) | 2009-06-25 |
RU2009126571A (ru) | 2011-01-20 |
CN101627023A (zh) | 2010-01-13 |
KR20090091326A (ko) | 2009-08-27 |
WO2008071951A3 (en) | 2008-10-02 |
ES2483718T3 (es) | 2014-08-07 |
EP2102182A2 (en) | 2009-09-23 |
PT103901B (pt) | 2012-03-01 |
CA2671830C (en) | 2019-03-19 |
JP2010512379A (ja) | 2010-04-22 |
CA2671830A1 (en) | 2008-06-19 |
MX2009006113A (es) | 2009-07-17 |
AU2007331340A1 (en) | 2008-06-19 |
US20100036127A1 (en) | 2010-02-11 |
US8546571B2 (en) | 2013-10-01 |
AR064308A1 (es) | 2009-03-25 |
JP5372771B2 (ja) | 2013-12-18 |
PT103901A (pt) | 2008-06-12 |
WO2008071951A2 (en) | 2008-06-19 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application fees: application dismissed [chapter 8.6 patent gazette] | ||
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2543 DE 01-10-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |