BRPI0607407A2 - derivados de mentano carboxamida tendo propriedades de refrescáncia - Google Patents

derivados de mentano carboxamida tendo propriedades de refrescáncia

Info

Publication number
BRPI0607407A2
BRPI0607407A2 BRPI0607407-3A BRPI0607407A BRPI0607407A2 BR PI0607407 A2 BRPI0607407 A2 BR PI0607407A2 BR PI0607407 A BRPI0607407 A BR PI0607407A BR PI0607407 A2 BRPI0607407 A2 BR PI0607407A2
Authority
BR
Brazil
Prior art keywords
carboxamide
menthane derivatives
refreshing properties
properties
group
Prior art date
Application number
BRPI0607407-3A
Other languages
English (en)
Inventor
Lucienne Cole
Stefan Michael Furrer
Christophe Galopin
Pablo Victor Krawec
Adam Masur
Jay Patrick Slack
Original Assignee
Givaudan Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Givaudan Sa filed Critical Givaudan Sa
Publication of BRPI0607407A2 publication Critical patent/BRPI0607407A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/40—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
    • A61K8/42—Amides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q11/00—Preparations for care of the teeth, of the oral cavity or of dentures; Dentifrices, e.g. toothpastes; Mouth rinses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/135—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/20—Chemical, physico-chemical or functional or structural properties of the composition as a whole
    • A61K2800/24—Thermal properties
    • A61K2800/244—Endothermic; Cooling; Cooling sensation

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Birds (AREA)
  • Oral & Maxillofacial Surgery (AREA)
  • Dermatology (AREA)
  • Cosmetics (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Seasonings (AREA)

Abstract

DERIVADOS DE MENTANO CARBOXAMIDA TENDO PROPRIEDADES DE REFRESCáNCIA. Um composto da Fórmula (I) onde X e Y são selecionados conforme definido na descrição. Os compostos têm propriedades de refrescância e são úteis em, por exemplo, alimentos, dentifrícios e cosméticos.
BRPI0607407-3A 2005-03-01 2006-02-23 derivados de mentano carboxamida tendo propriedades de refrescáncia BRPI0607407A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US65756205P 2005-03-01 2005-03-01
PCT/CH2006/000116 WO2006092074A1 (en) 2005-03-01 2006-02-23 Menthane carboxamide derivatives having cooling properties

Publications (1)

Publication Number Publication Date
BRPI0607407A2 true BRPI0607407A2 (pt) 2009-09-01

Family

ID=36127379

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0607407-3A BRPI0607407A2 (pt) 2005-03-01 2006-02-23 derivados de mentano carboxamida tendo propriedades de refrescáncia

Country Status (12)

Country Link
US (1) US7868004B2 (pt)
EP (1) EP1853565B1 (pt)
JP (1) JP2008531606A (pt)
KR (1) KR20070107083A (pt)
CN (1) CN101133030B (pt)
AT (1) ATE482199T1 (pt)
BR (1) BRPI0607407A2 (pt)
CA (1) CA2597415A1 (pt)
DE (1) DE602006017038D1 (pt)
ES (1) ES2352563T3 (pt)
MX (1) MX2007010040A (pt)
WO (1) WO2006092074A1 (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE602004026619D1 (en) 2003-11-21 2010-05-27 Givaudan Sa N-substituierte p-menthancarbonsäureamide
ATE443046T1 (de) 2005-10-25 2009-10-15 Givaudan Sa Organische verbindungen
EP2104436A1 (en) * 2006-12-20 2009-09-30 Givaudan Nederland Services B.V. N-substituted-p-menthane-3-carboxamide and uses thereof
WO2009076792A1 (en) * 2007-12-19 2009-06-25 Givaudan Sa Cooling compounds
US20100297038A1 (en) * 2008-01-17 2010-11-25 Givaudan S.A. Benzimidazole Derivatives And Their Use As Cooling Agents
GB0902849D0 (en) * 2009-02-19 2009-04-08 Givaudan Sa Organic compounds
GB201103103D0 (en) 2011-02-23 2011-04-06 Givaudan Sa Organic compounds
EP2497458A1 (en) 2011-03-08 2012-09-12 B.R.A.I.N. Biotechnology Research And Information Network AG Small molecule modulators of the cold and menthol receptor TRPM8
US9492411B2 (en) 2014-04-23 2016-11-15 The Procter & Gamble Company Medications for deposition on biological surfaces

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1351761A (en) * 1971-02-04 1974-05-01 Wilkinson Sword Ltd Substituted p-menthane carboxamides and compositions containing them
US5918309A (en) * 1997-10-14 1999-07-06 Second Chance Body Armor, Inc. Blunt force resistant structure for a protective garment
EP1556332B1 (en) * 2002-10-28 2016-10-05 Givaudan SA Coolant solutions and compositions comprising the same
JP5105873B2 (ja) 2003-07-02 2012-12-26 ジェネンテック， インコーポレイテッド Ｔｒｐ−ｐ８活性化合物と治療的処置方法
CA2535265C (en) 2003-08-22 2014-01-28 Dendreon Corporation Compositions and methods for the treatment of disease associated with trp-p8 expression
DE602004026619D1 (en) * 2003-11-21 2010-05-27 Givaudan Sa N-substituierte p-menthancarbonsäureamide
GB0425661D0 (en) 2004-11-23 2004-12-22 Givaudan Sa Organic compounds
US8673198B2 (en) * 2006-02-18 2014-03-18 Honeywell International Inc Method of making improved ballistic products

Also Published As

Publication number Publication date
EP1853565B1 (en) 2010-09-22
US20080305051A1 (en) 2008-12-11
ATE482199T1 (de) 2010-10-15
CN101133030A (zh) 2008-02-27
KR20070107083A (ko) 2007-11-06
US7868004B2 (en) 2011-01-11
EP1853565A1 (en) 2007-11-14
JP2008531606A (ja) 2008-08-14
CA2597415A1 (en) 2006-09-08
ES2352563T3 (es) 2011-02-21
WO2006092074A1 (en) 2006-09-08
DE602006017038D1 (de) 2010-11-04
MX2007010040A (es) 2007-09-21
CN101133030B (zh) 2010-07-28

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Legal Events

Date Code Title Description
B15K Others concerning applications: alteration of classification

Free format text: AS CLASSIFICACOES ANTERIORES ERAM: C07D 231/12 , C07D 249/08 , C07D 263/32 , C07D 295/135 , A61K 8/49

Ipc: A61K 8/42 (2006.01), A61K 8/49 (2006.01), A61Q 11/

B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements