BRPI0606724A2 - preparação farmacêutica para contracepção - Google Patents

preparação farmacêutica para contracepção

Info

Publication number
BRPI0606724A2
BRPI0606724A2 BRPI0606724-7A BRPI0606724A BRPI0606724A2 BR PI0606724 A2 BRPI0606724 A2 BR PI0606724A2 BR PI0606724 A BRPI0606724 A BR PI0606724A BR PI0606724 A2 BRPI0606724 A2 BR PI0606724A2
Authority
BR
Brazil
Prior art keywords
daily dose
contraception
dienogest
pharmaceutical preparation
ethinyl estradiol
Prior art date
Application number
BRPI0606724-7A
Other languages
English (en)
Inventor
Thomas Graeser
Claus Claussen
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of BRPI0606724A2 publication Critical patent/BRPI0606724A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/567Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Endocrinology (AREA)
  • Organic Chemistry (AREA)
  • Reproductive Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

PREPARAçãO FARMACêUTICA PARA CONTRACEPçãO. A presente invenção refere-se a uma composição farmacêutica contendo dienogest em uma quantidade que na administração da composição corresponde a uma unidade de dose diária de 1,5 mg ou 2,0 mg e contendo etinilestradiol em uma quantidade que na administração da composição corresponde a uma unidade de dose diária de 0,015 mg ou 0,020 mg, juntamente com um ou mais veículos farmaceuticamente aceitáveis para pelo menos 21 unidades de doses diárias. Além disso, a invenção refere-se a um preparado farmacêutico para contracepção oral, contendo 1,5 mg de 17<244>-cianometil-17-<225>-hidroxiestra-4,9-dien-3-ona (dienogest) e 0,015 ou 0,020 mg de 17<244>-etinilestradiol (etinilestradiol) ou 2,0 mg de dienogest e 0,015 mg de etinilestradiol, juntamente com um ou mais veículos farmaceuticamente aceitáveis para pelo menos 21 unidades de doses diárias de um ciclo menstrual de 28 dias.
BRPI0606724-7A 2005-02-15 2006-02-15 preparação farmacêutica para contracepção BRPI0606724A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05003179A EP1690543A1 (de) 2005-02-15 2005-02-15 Pharmazeutisches Präparat zur Kontrazeption
PCT/EP2006/001354 WO2006087173A1 (de) 2005-02-15 2006-02-15 Pharmazeutisches präparat zur kontrazeption

Publications (1)

Publication Number Publication Date
BRPI0606724A2 true BRPI0606724A2 (pt) 2009-07-14

Family

ID=34933759

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0606724-7A BRPI0606724A2 (pt) 2005-02-15 2006-02-15 preparação farmacêutica para contracepção

Country Status (20)

Country Link
EP (2) EP1690543A1 (pt)
JP (1) JP2008527018A (pt)
KR (1) KR20070086380A (pt)
CN (1) CN101119732A (pt)
AR (1) AR053545A1 (pt)
AU (1) AU2006215818A1 (pt)
BR (1) BRPI0606724A2 (pt)
CA (1) CA2590004A1 (pt)
CR (1) CR9324A (pt)
DO (1) DOP2006000035A (pt)
EA (1) EA200701091A1 (pt)
IL (1) IL183635A0 (pt)
MX (1) MX2007009061A (pt)
NO (1) NO20072687L (pt)
PA (1) PA8663401A1 (pt)
PE (1) PE20061291A1 (pt)
TW (1) TW200640468A (pt)
UA (1) UA85003C2 (pt)
WO (1) WO2006087173A1 (pt)
ZA (1) ZA200707910B (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1774970A1 (de) * 2005-10-13 2007-04-18 Bayer Schering Pharma AG Verfahren zur Herstellung eines einphasigen pharmazeutischen Präparates zur Therapie der dysfunktionellen uterinen Blutung, enthaltend Ethinylestradiol und Dienogest
US20090099144A1 (en) * 2007-10-11 2009-04-16 Katrin Mittmann Oral contraception (long-cycle regimen and 21-days-regimen with 30 mg ethinylestradiol and 2 mg dienogest) without treatment of thrombosis/hemostasis
EP2055306A1 (de) * 2007-11-05 2009-05-06 Bayer Schering Pharma AG Verwendung eines Gestagens in Kombination mit einem Estrogen und einem oder mehreren pharmazeutisch annehmbaren hilfsstoffen/Trägern zur laktosefreien oralen Kontrazeption

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2000515890A (ja) * 1996-07-26 2000-11-28 アメリカン・ホーム・プロダクツ・コーポレイション プロゲスチンとエストロゲンとの混合剤からなる一相性避妊法およびキット

Also Published As

Publication number Publication date
IL183635A0 (en) 2007-10-31
TW200640468A (en) 2006-12-01
CR9324A (es) 2007-10-11
MX2007009061A (es) 2007-09-11
EP1853273A1 (de) 2007-11-14
AR053545A1 (es) 2007-05-09
EA200701091A1 (ru) 2008-02-28
CN101119732A (zh) 2008-02-06
PE20061291A1 (es) 2006-12-07
KR20070086380A (ko) 2007-08-27
NO20072687L (no) 2007-11-13
WO2006087173A1 (de) 2006-08-24
EP1690543A1 (de) 2006-08-16
DOP2006000035A (es) 2006-09-15
PA8663401A1 (es) 2006-12-07
UA85003C2 (ru) 2008-12-10
ZA200707910B (en) 2009-08-26
AU2006215818A1 (en) 2006-08-24
JP2008527018A (ja) 2008-07-24
CA2590004A1 (en) 2006-08-24

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 5A E 6A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2161 DE 05/06/2012.