BRPI0508969A - compostos orgánicos - Google Patents
compostos orgánicosInfo
- Publication number
- BRPI0508969A BRPI0508969A BRPI0508969-7A BRPI0508969A BRPI0508969A BR PI0508969 A BRPI0508969 A BR PI0508969A BR PI0508969 A BRPI0508969 A BR PI0508969A BR PI0508969 A BRPI0508969 A BR PI0508969A
- Authority
- BR
- Brazil
- Prior art keywords
- organic compounds
- compounds
- remedies
- formula
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/12—Radicals substituted by oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Abstract
COMPOSTOS ORGáNICOS. A invenção refere-se novos amino ácooios de fórmula geral (I) onde X, R¬ 1¬, R¬ 2¬, R¬ 3¬, R¬ 4¬, R¬ 5¬ e R¬ 6¬ são, cada um,como definidos em detalhes na descrição, a um processo para sua preparação e ao uso destes compostos como remédios, particularmente como inibidores de renina.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH4792004 | 2004-03-19 | ||
PCT/EP2005/051241 WO2005090304A1 (en) | 2004-03-19 | 2005-03-17 | Organic compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0508969A true BRPI0508969A (pt) | 2007-08-21 |
Family
ID=34961967
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0508969-7A BRPI0508969A (pt) | 2004-03-19 | 2005-03-17 | compostos orgánicos |
Country Status (10)
Country | Link |
---|---|
US (1) | US7868036B2 (pt) |
EP (1) | EP1725530A1 (pt) |
JP (1) | JP4927704B2 (pt) |
CN (1) | CN1934082A (pt) |
AR (1) | AR048107A1 (pt) |
BR (1) | BRPI0508969A (pt) |
CA (1) | CA2560195A1 (pt) |
IL (1) | IL178099A0 (pt) |
TW (1) | TW200609215A (pt) |
WO (1) | WO2005090304A1 (pt) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0505969D0 (en) | 2005-03-23 | 2005-04-27 | Novartis Ag | Organic compounds |
EP1764099A3 (en) * | 2005-09-17 | 2007-05-09 | Speedel Experimenta AG | Diaminoalcohol derivatives for the treatment of Alzheimer, malaria, HIV |
EP1968940B1 (en) | 2005-12-30 | 2014-04-02 | Novartis AG | 3 , 5-substitued piperidine compounds as renin inhibitors |
TW200815324A (en) * | 2006-06-23 | 2008-04-01 | Daiichi Sankyo Co Ltd | Straight chain amine compound |
NZ573720A (en) | 2006-06-23 | 2011-01-28 | Daiichi Sankyo Co Ltd | Cyclic amine compound |
EP2181105B1 (en) | 2007-06-25 | 2015-04-29 | Novartis AG | N5-(2-ethoxyethyl)-n3-(2-pyridinyl)-3,5-piperidinedicarboxamide derivatives for use as renin inhibitors |
DK2975024T3 (en) | 2009-06-10 | 2018-04-23 | Chugai Pharmaceutical Co Ltd | Tetracyclic compounds |
AR077428A1 (es) * | 2009-07-29 | 2011-08-24 | Sanofi Aventis | (aza) indolizinacarboxamidas ciclicas su preparacion y su uso como agentes farmaceuticos |
EP2606886B1 (en) | 2010-08-20 | 2020-01-08 | Chugai Seiyaku Kabushiki Kaisha | Composition comprising tetracyclic compound |
CN111388478A (zh) | 2012-09-25 | 2020-07-10 | 中外制药株式会社 | Ret抑制剂 |
CN104418835A (zh) * | 2013-09-02 | 2015-03-18 | 上海龙翔生物医药开发有限公司 | 一种甲磺酸伊马替尼的制备方法 |
AR100187A1 (es) | 2014-04-25 | 2016-09-14 | Chugai Pharmaceutical Co Ltd | Composición farmacéutica que contiene un inhibidor de alk (quinasa de linfoma anaplásico) |
US9714229B2 (en) | 2014-04-25 | 2017-07-25 | Chugai Seiyaku Kabushiki Kaisha | Crystal of tetracyclic compound |
TWI765410B (zh) | 2014-08-08 | 2022-05-21 | 日商中外製藥股份有限公司 | 4環性化合物的非晶質體的用途 |
WO2016114375A1 (ja) | 2015-01-16 | 2016-07-21 | 中外製薬株式会社 | 併用医薬 |
CN112585126B (zh) | 2018-09-04 | 2024-05-07 | 中外制药株式会社 | 四环化合物的制备方法 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY119161A (en) | 1994-04-18 | 2005-04-30 | Novartis Ag | Delta-amino-gamma-hydroxy-omega-aryl-alkanoic acid amides with enzyme especially renin inhibiting activities |
US5659065A (en) | 1994-04-18 | 1997-08-19 | Novartis Corporation | Alpha-aminoalkanoic acids and reduction products |
US5606078A (en) | 1994-04-18 | 1997-02-25 | Ciba-Geigy Corporation | 3,5-Disubstituted tetrahydrofuran-2-ones |
US8168616B1 (en) * | 2000-11-17 | 2012-05-01 | Novartis Ag | Combination comprising a renin inhibitor and an angiotensin receptor inhibitor for hypertension |
US7312360B2 (en) | 2001-12-06 | 2007-12-25 | Elan Pharmaceuticals, Inc. | Substituted hydroxyethylamines |
-
2005
- 2005-03-17 EP EP05717092A patent/EP1725530A1/en not_active Withdrawn
- 2005-03-17 CN CNA2005800087339A patent/CN1934082A/zh active Pending
- 2005-03-17 CA CA002560195A patent/CA2560195A1/en not_active Abandoned
- 2005-03-17 TW TW094108180A patent/TW200609215A/zh unknown
- 2005-03-17 BR BRPI0508969-7A patent/BRPI0508969A/pt not_active IP Right Cessation
- 2005-03-17 JP JP2007503351A patent/JP4927704B2/ja not_active Expired - Fee Related
- 2005-03-17 US US10/593,461 patent/US7868036B2/en not_active Expired - Fee Related
- 2005-03-17 WO PCT/EP2005/051241 patent/WO2005090304A1/en not_active Application Discontinuation
- 2005-03-18 AR ARP050101072A patent/AR048107A1/es unknown
-
2006
- 2006-09-14 IL IL178099A patent/IL178099A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
US7868036B2 (en) | 2011-01-11 |
JP4927704B2 (ja) | 2012-05-09 |
US20080058320A1 (en) | 2008-03-06 |
EP1725530A1 (en) | 2006-11-29 |
AR048107A1 (es) | 2006-03-29 |
IL178099A0 (en) | 2006-12-31 |
JP2007529473A (ja) | 2007-10-25 |
CN1934082A (zh) | 2007-03-21 |
WO2005090304A1 (en) | 2005-09-29 |
CA2560195A1 (en) | 2005-09-29 |
TW200609215A (en) | 2006-03-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 8A ANUIDADE |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2204 DE 02/04/2013. |