BRPI0418973A - composições de risedronato e seus métodos de uso - Google Patents
composições de risedronato e seus métodos de usoInfo
- Publication number
- BRPI0418973A BRPI0418973A BRPI0418973-6A BRPI0418973A BRPI0418973A BR PI0418973 A BRPI0418973 A BR PI0418973A BR PI0418973 A BRPI0418973 A BR PI0418973A BR PI0418973 A BRPI0418973 A BR PI0418973A
- Authority
- BR
- Brazil
- Prior art keywords
- risedronate
- compositions
- methods
- polymorph
- solvate
- Prior art date
Links
- IIDJRNMFWXDHID-UHFFFAOYSA-N Risedronic acid Chemical compound OP(=O)(O)C(P(O)(O)=O)(O)CC1=CC=CN=C1 IIDJRNMFWXDHID-UHFFFAOYSA-N 0.000 title abstract 3
- 229940089617 risedronate Drugs 0.000 title abstract 3
- 239000000203 mixture Substances 0.000 title abstract 2
- 241000124008 Mammalia Species 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 210000000988 bone and bone Anatomy 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 208000030159 metabolic disease Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/662—Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
- A61K31/663—Compounds having two or more phosphorus acid groups or esters thereof, e.g. clodronic acid, pamidronic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Physical Education & Sports Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/897,897 US20050070504A1 (en) | 2001-12-21 | 2004-07-23 | Risedronate compositions and their methods of use |
| PCT/US2004/031975 WO2006022755A1 (en) | 2004-07-23 | 2004-09-25 | Risedronate compositions and their methods of use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0418973A true BRPI0418973A (pt) | 2007-12-04 |
Family
ID=34958880
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0418973-6A BRPI0418973A (pt) | 2004-07-23 | 2004-09-25 | composições de risedronato e seus métodos de uso |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US20050070504A1 (enExample) |
| EP (1) | EP1776123A1 (enExample) |
| JP (3) | JP5377852B2 (enExample) |
| KR (2) | KR20070038115A (enExample) |
| CN (1) | CN101146542A (enExample) |
| AR (1) | AR046036A1 (enExample) |
| AU (2) | AU2004322703B2 (enExample) |
| BR (1) | BRPI0418973A (enExample) |
| CA (1) | CA2564898A1 (enExample) |
| IL (1) | IL180907A0 (enExample) |
| IS (1) | IS8597A (enExample) |
| MA (1) | MA28778B1 (enExample) |
| MX (1) | MX2007000967A (enExample) |
| NO (1) | NO20071058L (enExample) |
| NZ (1) | NZ552799A (enExample) |
| PE (1) | PE20060144A1 (enExample) |
| RU (1) | RU2007103306A (enExample) |
| TW (1) | TWI351286B (enExample) |
| WO (1) | WO2006022755A1 (enExample) |
| ZA (1) | ZA200701308B (enExample) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL162053A0 (en) * | 2001-12-21 | 2005-11-20 | Procter & Gamble | Method for the treatment of bone disorders |
| EP2851105A1 (en) * | 2002-05-10 | 2015-03-25 | F. Hoffmann-La Roche AG | Bisphosphonic acids for treatment and prevention of osteoporosis |
| WO2004056373A1 (en) * | 2002-12-20 | 2004-07-08 | F. Hoffmann-La Roche Ag | High dose ibandronate formulation |
| US7645459B2 (en) | 2004-05-24 | 2010-01-12 | The Procter & Gamble Company | Dosage forms of bisphosphonates |
| US20080287400A1 (en) * | 2004-05-24 | 2008-11-20 | Richard John Dansereau | Low Dosage Forms Of Risedronate Or Its Salts |
| AU2011218625B2 (en) * | 2004-05-24 | 2014-03-20 | Theramex HQ UK Limited | Dosage forms of risedronate |
| US20080286359A1 (en) * | 2004-05-24 | 2008-11-20 | Richard John Dansereau | Low Dosage Forms Of Risedronate Or Its Salts |
| US8071574B2 (en) * | 2005-02-22 | 2011-12-06 | John Dennis Bobyn | Implant improving local bone formation |
| US7473684B2 (en) | 2005-09-16 | 2009-01-06 | Selamine Limited | Bisphosphonate formulation |
| ES2567595T3 (es) * | 2005-10-12 | 2016-04-25 | Opko Renal, Llc | Métodos y artículos para tratar la insuficiencia y la deficiencia de 25-hidroxivitamina D |
| GB0624090D0 (en) * | 2006-12-01 | 2007-01-10 | Selamine Ltd | Ramipril amine salts |
| GB0624084D0 (en) * | 2006-12-01 | 2007-01-10 | Selamine Ltd | Ramipril amino acid salts |
| GB0624087D0 (en) * | 2006-12-01 | 2007-01-10 | Selamine Ltd | Ramipril combination salt |
| KR100844256B1 (ko) | 2007-03-23 | 2008-07-07 | 코오롱제약주식회사 | 리세드로네이트와 비타민 d를 포함하는 대사성 골질환치료용 약제조성물 및 이의 제조방법 |
| JP2011529901A (ja) * | 2008-07-31 | 2011-12-15 | 味の素株式会社 | リセドロネートまたはその塩の低投与量形態 |
| KR101379664B1 (ko) * | 2008-09-23 | 2014-04-02 | 한림제약(주) | 리세드론산 또는 그의 염 및 비타민 d를 포함하는 약학 조성물 |
| KR101102364B1 (ko) | 2009-09-18 | 2012-01-03 | 한림제약(주) | 비스포스포네이트 유도체 및 고용량의 콜레칼시페롤을 포함하는 약학 조성물 |
| PT106978A (pt) * | 2013-05-31 | 2014-12-02 | Tecnimede Sociedade Tecnico Medicinal S A | Composição sólida oral contendo ácido ibandrónico e vitamina d |
Family Cites Families (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA777769A (en) * | 1963-03-18 | 1968-02-06 | H. Roy Clarence | Substituted methylene diphosphonic acid compounds and detergent compositions |
| IT1201087B (it) * | 1982-04-15 | 1989-01-27 | Gentili Ist Spa | Bifosfonati farmacologicamente attivi,procedimento per la loro preparazione e relative composizioni farmaceutiche |
| FR2531088B1 (fr) * | 1982-07-29 | 1987-08-28 | Sanofi Sa | Produits anti-inflammatoires derives de l'acide methylenediphosphonique et leur procede de preparation |
| IL77243A (en) * | 1984-12-21 | 1996-11-14 | Procter & Gamble | Pharmaceutical compositions containing geminal diphosphonic acid compounds and certain such novel compounds |
| US4761406A (en) * | 1985-06-06 | 1988-08-02 | The Procter & Gamble Company | Regimen for treating osteoporosis |
| DE3623397A1 (de) * | 1986-07-11 | 1988-01-14 | Boehringer Mannheim Gmbh | Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
| CA1339805C (en) * | 1988-01-20 | 1998-04-07 | Yasuo Isomura | (cycloalkylamino)methylenebis(phosphonic acid) and medicines containing the same as an active |
| GB2217988B (en) * | 1988-04-11 | 1992-04-01 | Gould Leonard W | Regimen for increasing bone density in humans |
| US4922007A (en) * | 1989-06-09 | 1990-05-01 | Merck & Co., Inc. | Process for preparing 4-amino-1-hydroxybutylidene-1,1-bisphosphonic acid or salts thereof |
| US5227506A (en) * | 1989-09-06 | 1993-07-13 | Merck & Co., Inc. | Acyloxymethyl esters of bisphosphonic acids as bone resorption inhibitors |
| NL8902727A (nl) * | 1989-11-06 | 1991-06-03 | Philips Nv | Objecthouder voor ondersteuning van een object in een geladen deeltjesbundelsysteem. |
| EP0650361B1 (en) * | 1992-06-30 | 1999-04-28 | PROCTER & GAMBLE PHARMACEUTICALS, INC. | Compositions for the treatment of arthritis containing phosphonates and nsaids |
| US5646134A (en) * | 1994-04-21 | 1997-07-08 | Merck & Co., Inc. | Alendronate therapy to prevent loosening of, or pain associated with, orthopedic implant devices |
| US6008206A (en) * | 1994-09-21 | 1999-12-28 | Merck & Co., Inc. | Sodium alendronate preparation for local administration |
| US6750216B2 (en) * | 1996-03-08 | 2004-06-15 | Adolor Corporation | Kappa agonist compounds and pharmaceutical formulations thereof |
| US5730715A (en) * | 1996-06-14 | 1998-03-24 | Becton Dickinson And Company | Method for the iontophoretic administration of bisphosphonates |
| GB2324726A (en) * | 1997-05-01 | 1998-11-04 | Merck & Co Inc | Combination Therapy for the Treatment of Osteoporosis |
| SK284690B6 (sk) * | 1997-06-11 | 2005-09-08 | The Procter And Gamble Company | Ústna dávkovacia forma na zvýšenie ochrany horného tráviaceho traktu |
| US6015801A (en) * | 1997-07-22 | 2000-01-18 | Merck & Co., Inc. | Method for inhibiting bone resorption |
| US5994329A (en) * | 1997-07-22 | 1999-11-30 | Merck & Co., Inc. | Method for inhibiting bone resorption |
| US6432932B1 (en) * | 1997-07-22 | 2002-08-13 | Merck & Co., Inc. | Method for inhibiting bone resorption |
| US6331533B1 (en) * | 1998-11-16 | 2001-12-18 | Merck & Co., Inc. | Method for inhibiting dental resorptive lesions |
| US6225801B1 (en) * | 1999-01-14 | 2001-05-01 | Lucent Technologies Inc. | Article comprising electronic circuits and devices with magnetically programmable electrical resistance |
| JP2001253827A (ja) * | 2000-02-15 | 2001-09-18 | Pfizer Prod Inc | 骨粗鬆症を治療するための組成物および方法 |
| US6468559B1 (en) * | 2000-04-28 | 2002-10-22 | Lipocine, Inc. | Enteric coated formulation of bishosphonic acid compounds and associated therapeutic methods |
| KR100864743B1 (ko) * | 2000-06-20 | 2008-10-22 | 노파르티스 아게 | 비스포스포네이트의 투여 방법 |
| US6593310B1 (en) * | 2000-11-21 | 2003-07-15 | Arthropharm Pty. Ltd. | Treatment of osteoporosis |
| WO2003051373A1 (en) * | 2001-12-13 | 2003-06-26 | Merck & Co., Inc. | Liquid bisphosphonate formulations for bone disorders |
| EP2851105A1 (en) * | 2002-05-10 | 2015-03-25 | F. Hoffmann-La Roche AG | Bisphosphonic acids for treatment and prevention of osteoporosis |
| US20040188316A1 (en) * | 2003-03-26 | 2004-09-30 | The Procter & Gamble Company | Kit for pharmaceutical use |
-
2004
- 2004-07-23 US US10/897,897 patent/US20050070504A1/en not_active Abandoned
- 2004-09-25 NZ NZ552799A patent/NZ552799A/en not_active IP Right Cessation
- 2004-09-25 MX MX2007000967A patent/MX2007000967A/es unknown
- 2004-09-25 AU AU2004322703A patent/AU2004322703B2/en not_active Withdrawn - After Issue
- 2004-09-25 CN CNA2004800436570A patent/CN101146542A/zh active Pending
- 2004-09-25 CA CA002564898A patent/CA2564898A1/en not_active Abandoned
- 2004-09-25 KR KR1020077001602A patent/KR20070038115A/ko not_active Ceased
- 2004-09-25 KR KR1020087021196A patent/KR20080083219A/ko not_active Ceased
- 2004-09-25 RU RU2007103306/14A patent/RU2007103306A/ru unknown
- 2004-09-25 EP EP04789250A patent/EP1776123A1/en not_active Ceased
- 2004-09-25 WO PCT/US2004/031975 patent/WO2006022755A1/en not_active Ceased
- 2004-09-25 JP JP2007522476A patent/JP5377852B2/ja not_active Expired - Lifetime
- 2004-09-25 BR BRPI0418973-6A patent/BRPI0418973A/pt not_active Application Discontinuation
- 2004-09-29 AR ARP040103537A patent/AR046036A1/es unknown
- 2004-09-30 PE PE2004000960A patent/PE20060144A1/es not_active Application Discontinuation
- 2004-11-30 TW TW093136901A patent/TWI351286B/zh not_active IP Right Cessation
-
2007
- 2007-01-23 IL IL180907A patent/IL180907A0/en unknown
- 2007-01-24 IS IS8597A patent/IS8597A/is unknown
- 2007-02-01 MA MA29645A patent/MA28778B1/fr unknown
- 2007-02-14 ZA ZA200701308A patent/ZA200701308B/en unknown
- 2007-02-22 NO NO20071058A patent/NO20071058L/no not_active Application Discontinuation
-
2011
- 2011-03-02 AU AU2011200905A patent/AU2011200905A1/en not_active Abandoned
-
2013
- 2013-08-16 JP JP2013169220A patent/JP5761274B2/ja not_active Expired - Lifetime
-
2014
- 2014-10-21 JP JP2014214604A patent/JP5910698B2/ja not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| AR046036A1 (es) | 2005-11-23 |
| ZA200701308B (en) | 2008-07-30 |
| PE20060144A1 (es) | 2006-04-17 |
| CN101146542A (zh) | 2008-03-19 |
| AU2004322703B2 (en) | 2010-12-02 |
| US20050070504A1 (en) | 2005-03-31 |
| JP5910698B2 (ja) | 2016-04-27 |
| WO2006022755A1 (en) | 2006-03-02 |
| IS8597A (is) | 2007-01-24 |
| MX2007000967A (es) | 2007-07-11 |
| CA2564898A1 (en) | 2006-03-02 |
| AU2004322703A1 (en) | 2006-03-02 |
| JP2008507513A (ja) | 2008-03-13 |
| TW200603816A (en) | 2006-02-01 |
| IL180907A0 (en) | 2007-07-04 |
| JP5761274B2 (ja) | 2015-08-12 |
| AU2011200905A1 (en) | 2011-03-24 |
| KR20080083219A (ko) | 2008-09-16 |
| JP2013231087A (ja) | 2013-11-14 |
| NZ552799A (en) | 2010-04-30 |
| RU2007103306A (ru) | 2008-09-10 |
| JP2015038135A (ja) | 2015-02-26 |
| KR20070038115A (ko) | 2007-04-09 |
| JP5377852B2 (ja) | 2013-12-25 |
| NO20071058L (no) | 2007-02-22 |
| TWI351286B (en) | 2011-11-01 |
| EP1776123A1 (en) | 2007-04-25 |
| MA28778B1 (fr) | 2007-08-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B25A | Requested transfer of rights approved |
Owner name: WARNER CHILCOTT COMPANY, LLC (PR) |
|
| B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
| B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] |
Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI |
|
| B15K | Others concerning applications: alteration of classification |
Free format text: AS CLASSIFICACOES ANTERIORES ERAM: A61K 31/675 , A61P 19/10 Ipc: A61K 31/663 (2006.01), A61K 31/675 (2006.01), A61P |
|
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8 E 13 DA LPI |
|
| B12B | Appeal against refusal [chapter 12.2 patent gazette] | ||
| B25E | Requested change of name of applicant rejected |
Owner name: WARNER CHILCOTT COMPANY, LLC (PR) |