BRPI0408752A - processo para o preparo de um polimorfo de maleato de rosiglitazona - Google Patents
processo para o preparo de um polimorfo de maleato de rosiglitazonaInfo
- Publication number
- BRPI0408752A BRPI0408752A BRPI0408752-6A BRPI0408752A BRPI0408752A BR PI0408752 A BRPI0408752 A BR PI0408752A BR PI0408752 A BRPI0408752 A BR PI0408752A BR PI0408752 A BRPI0408752 A BR PI0408752A
- Authority
- BR
- Brazil
- Prior art keywords
- preparing
- rosiglitazone maleate
- maleate polymorph
- compound
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
"PROCESSO PARA O PREPARO DE UM POLIMORFO DE MALEATO DE ROSIGLITAZONA". Um processo de cristalização para o preparo de maleato de rosiglitazona (Composto 1) , e um processo para o preparo do Composto 1 com uma pureza polimórfica que seja adequado para o uso como um material de semeadura em um processo de cristalização para o preparo do Composto 1.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0307259.2A GB0307259D0 (en) | 2003-03-28 | 2003-03-28 | Process |
PCT/GB2004/001306 WO2004085435A1 (en) | 2003-03-28 | 2004-03-25 | Process for preparing a polymorph of rosiglitazone maleate |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0408752A true BRPI0408752A (pt) | 2006-03-28 |
Family
ID=9955778
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0408752-6A BRPI0408752A (pt) | 2003-03-28 | 2004-03-25 | processo para o preparo de um polimorfo de maleato de rosiglitazona |
Country Status (18)
Country | Link |
---|---|
US (1) | US20070167494A1 (pt) |
EP (1) | EP1615918A1 (pt) |
JP (1) | JP2006521340A (pt) |
KR (1) | KR20050120670A (pt) |
CN (1) | CN1768057A (pt) |
AU (2) | AU2004224068A1 (pt) |
BR (1) | BRPI0408752A (pt) |
CA (1) | CA2520249A1 (pt) |
EA (1) | EA009331B1 (pt) |
EC (1) | ECSP056038A (pt) |
GB (1) | GB0307259D0 (pt) |
IS (1) | IS8087A (pt) |
MA (1) | MA27727A1 (pt) |
MX (1) | MXPA05010413A (pt) |
NO (1) | NO20054911L (pt) |
OA (1) | OA13042A (pt) |
WO (1) | WO2004085435A1 (pt) |
ZA (1) | ZA200507100B (pt) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20020137940A1 (en) | 1997-12-16 | 2002-09-26 | Smithkline Beecham P.L.C. | 5-[4-[2-(N-methyl-N-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2, 4-dione, maleic acid salt, hydrate as pharmaceutical |
US20040248945A1 (en) | 1999-04-23 | 2004-12-09 | Smithkline Beecham P.L.C. | Thiazolidinedione derivative and its use as antidiabetic |
GB2405403A (en) * | 2003-08-29 | 2005-03-02 | Cipla Ltd | Rosiglitazone maleate of particular polymorphic forms and methods of preparing rosiglitazone free base |
ITMI20041537A1 (it) * | 2004-07-28 | 2004-10-28 | Chemi Spa | Nuova forma polimorfa del rosiglitazone maleato |
CZ298424B6 (cs) * | 2005-05-24 | 2007-09-26 | Zentiva, A. S. | Zpusob krystalizace rosiglitazonu a jeho derivátuze smesných rozpouštedel |
KR20230170135A (ko) | 2017-01-27 | 2023-12-18 | 뉴로크린 바이오사이언시즈 인코퍼레이티드 | 특정 vmat2 억제제의 투여 방법 |
IL309802A (en) | 2017-09-21 | 2024-02-01 | Neurocrine Biosciences Inc | High dose valbenazine formulation and related preparations, methods and kits |
CN116492340A (zh) | 2017-10-10 | 2023-07-28 | 纽罗克里生物科学有限公司 | 施用某些vmat2抑制剂的方法 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9218830D0 (en) * | 1992-09-05 | 1992-10-21 | Smithkline Beecham Plc | Novel compounds |
GB9723295D0 (en) * | 1997-11-04 | 1998-01-07 | Smithkline Beecham Plc | Novel process |
JP2002543076A (ja) * | 1999-04-23 | 2002-12-17 | スミスクライン ビーチャム パブリック リミテッド カンパニー | チアゾリジンジオン誘導体および抗糖尿病薬としてのその使用 |
ES2203453T3 (es) * | 1999-04-23 | 2004-04-16 | Smithkline Beecham Plc | Polimorfo de sal del acido maleico de 5-(4-(2-(n-metil-n-(2-piridil)amino)etoxi)bentil)tiazolidina-2,4-diona. |
PT1173434E (pt) * | 1999-04-23 | 2003-12-31 | Smithkline Beecham Plc | Novo produto farmaceutico |
IL155036A0 (en) * | 2000-09-26 | 2003-10-31 | Reddy Research Foundation | Polymorphic forms of 5-[4-[2-[n-methyl-n-(2-pyridyl) amino] ethoxy] benzyl] thiazolidine-2,4-dione maleate and pharmaceutical compositions containing the same |
-
2003
- 2003-03-28 GB GBGB0307259.2A patent/GB0307259D0/en not_active Ceased
-
2004
- 2004-03-25 US US10/551,021 patent/US20070167494A1/en not_active Abandoned
- 2004-03-25 EP EP04723254A patent/EP1615918A1/en not_active Withdrawn
- 2004-03-25 JP JP2006506028A patent/JP2006521340A/ja not_active Withdrawn
- 2004-03-25 MX MXPA05010413A patent/MXPA05010413A/es unknown
- 2004-03-25 KR KR1020057018143A patent/KR20050120670A/ko not_active Application Discontinuation
- 2004-03-25 BR BRPI0408752-6A patent/BRPI0408752A/pt not_active IP Right Cessation
- 2004-03-25 WO PCT/GB2004/001306 patent/WO2004085435A1/en active Application Filing
- 2004-03-25 EA EA200501527A patent/EA009331B1/ru unknown
- 2004-03-25 CA CA002520249A patent/CA2520249A1/en not_active Abandoned
- 2004-03-25 AU AU2004224068A patent/AU2004224068A1/en not_active Abandoned
- 2004-03-25 CN CNA2004800083916A patent/CN1768057A/zh active Pending
- 2004-03-25 OA OA1200500267A patent/OA13042A/en unknown
-
2005
- 2005-09-05 ZA ZA200507100A patent/ZA200507100B/en unknown
- 2005-09-26 EC EC2005006038A patent/ECSP056038A/es unknown
- 2005-10-11 MA MA28549A patent/MA27727A1/fr unknown
- 2005-10-24 NO NO20054911A patent/NO20054911L/no not_active Application Discontinuation
- 2005-10-24 IS IS8087A patent/IS8087A/is unknown
-
2008
- 2008-10-30 AU AU2008237610A patent/AU2008237610A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CN1768057A (zh) | 2006-05-03 |
EP1615918A1 (en) | 2006-01-18 |
ZA200507100B (en) | 2006-07-26 |
OA13042A (en) | 2006-11-10 |
GB0307259D0 (en) | 2003-05-07 |
CA2520249A1 (en) | 2004-10-07 |
JP2006521340A (ja) | 2006-09-21 |
MA27727A1 (fr) | 2006-01-02 |
KR20050120670A (ko) | 2005-12-22 |
EA009331B1 (ru) | 2007-12-28 |
WO2004085435A1 (en) | 2004-10-07 |
EA200501527A1 (ru) | 2006-02-24 |
AU2008237610A1 (en) | 2008-11-27 |
IS8087A (is) | 2005-10-24 |
MXPA05010413A (es) | 2005-11-04 |
ECSP056038A (es) | 2006-01-27 |
AU2004224068A1 (en) | 2004-10-07 |
US20070167494A1 (en) | 2007-07-19 |
NO20054911L (no) | 2005-10-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A ANUIDADE. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2137 DE 20/12/2011. |