BRPI0408323A - processo para a preparação de compimidos de liberação prolongada - Google Patents

processo para a preparação de compimidos de liberação prolongada

Info

Publication number
BRPI0408323A
BRPI0408323A BRPI0408323-7A BRPI0408323A BRPI0408323A BR PI0408323 A BRPI0408323 A BR PI0408323A BR PI0408323 A BRPI0408323 A BR PI0408323A BR PI0408323 A BRPI0408323 A BR PI0408323A
Authority
BR
Brazil
Prior art keywords
present
release
pharmaceutical composition
preparation
sustained release
Prior art date
Application number
BRPI0408323-7A
Other languages
English (en)
Inventor
Nirmal Mulye
Original Assignee
Nirmal Mulye
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nirmal Mulye filed Critical Nirmal Mulye
Publication of BRPI0408323A publication Critical patent/BRPI0408323A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

"PROCESSO PARA A PREPARAçãO DE COMPRIMIDOS DE LIBERAçãO PROLONGADA". A presente invenção se refere a um novo processo para a preparação de comprimidos de liberação prolongada contendo compostos medicinais e aos produtos preparados por esse processo. A presente invenção se refere a um processo de preparação de uma composição farmacêutica de liberação prolongada com um perfil predeterminado de liberação de medicamento, mas que se desvie dele pela adição de uma quantidade eficaz para a formação de comprimidos de uma celulose insolúvel ou parcialmente insolúvel em água à composição farmacêutica, composta por um medicamento em uma quantidade terapeuticamente eficaz, um veículo de liberação prolongada, presente em quantidades eficaz para retardar a liberação do medicamento da composição farmacêutica, e a celulose, esta última estando presente em um sistema aquoso, o aperfeiçoamento compreendendo a adição à composição de uma quantidade eficaz de maltodextrina para retardar o aumento da taxa de liberação do medicamento pela adição da celulose a ele.
BRPI0408323-7A 2003-03-14 2004-03-15 processo para a preparação de compimidos de liberação prolongada BRPI0408323A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US45480303P 2003-03-14 2003-03-14
PCT/US2004/007826 WO2004082615A2 (en) 2003-03-14 2004-03-15 A process for preparing sustained release tablets

Publications (1)

Publication Number Publication Date
BRPI0408323A true BRPI0408323A (pt) 2006-03-07

Family

ID=33029912

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0408323-7A BRPI0408323A (pt) 2003-03-14 2004-03-15 processo para a preparação de compimidos de liberação prolongada

Country Status (9)

Country Link
US (2) US20040224017A1 (pt)
EP (1) EP1603540A2 (pt)
JP (1) JP2006520390A (pt)
AU (1) AU2004222339A1 (pt)
BR (1) BRPI0408323A (pt)
CA (1) CA2518734A1 (pt)
MX (1) MXPA05009886A (pt)
NZ (1) NZ542303A (pt)
WO (1) WO2004082615A2 (pt)

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CA2518734A1 (en) * 2003-03-14 2004-09-30 Nirmal Mulye A process for preparing sustained release tablets
AU2004289252C1 (en) 2003-11-08 2013-06-20 Prothera Biologics, Inc. Preparation and composition of Inter-alpha inhibitor proteins from human plasma for therapeutic use
US20070161711A1 (en) * 2003-12-23 2007-07-12 Temrel Limited Process for producing pellets for pharmaceutical compositions
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BRPI0610257A2 (pt) * 2005-04-25 2010-06-08 Teva Pharma formulações de liberação prolongada
US20080058408A1 (en) 2006-05-19 2008-03-06 Rogowski Roberta L Low-dose doxepin for treatment of sleep disorders in elderly patients
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WO2007136741A2 (en) * 2006-05-19 2007-11-29 Somaxon Pharmaceuticals, Inc. N-desmethyl-doxepin and methods of using the same to treat sleep disorders
CA2687118A1 (en) 2006-05-19 2007-12-13 Somaxon Pharmaceuticals, Inc. Methods of using low-dose doxepin for the improvement of sleep
US20100179214A1 (en) 2006-05-19 2010-07-15 Somaxon Pharmaceuticals, Inc. Doxepin trans isomers and isomeric mixtures and methods of using the same to treat sleep disorders
US20080069891A1 (en) * 2006-09-15 2008-03-20 Cima Labs, Inc. Abuse resistant drug formulation
CA2693992C (en) 2006-07-20 2017-01-31 Somaxon Pharmaceuticals, Inc. Methods of improving the pharmacokinetics of doxepin
US8445018B2 (en) * 2006-09-15 2013-05-21 Cima Labs Inc. Abuse resistant drug formulation
WO2008052139A2 (en) 2006-10-25 2008-05-02 Somaxon Pharmaceuticals, Inc. Ultra low dose doxepin and methods of using the same to treat sleep disorders
US20110077200A1 (en) 2006-12-06 2011-03-31 Somaxon Pharmaceuticals, Inc. Combination therapy using low-dose doxepin for the improvement of sleep
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WO2008128115A2 (en) 2007-04-13 2008-10-23 Somaxon Pharmaceuticals, Inc. Low-dose doxepin formulations
US20090036414A1 (en) * 2007-08-02 2009-02-05 Mutual Pharmaceutical Company, Inc. Mesalamine Formulations
EP2200613B1 (en) 2007-09-21 2018-09-05 The Johns Hopkins University Phenazine derivatives and uses thereof
WO2009042778A1 (en) * 2007-09-25 2009-04-02 Nirmal Mulye Controlled release pharmaceutical compositions
KR101569604B1 (ko) * 2007-12-28 2015-11-16 임팩스 라보라토리즈, 인코포레이티드 레보도파 방출 제어형 제제 및 이의 용도
PT2291654T (pt) 2008-05-28 2018-06-15 Prothera Biologics Inc Preparação e composição de proteínas inibidoras de interalfa do sangue
MX2012012991A (es) 2010-05-11 2012-11-30 Cima Labs Inc Formas de dosificacion oral de liberacion prolongada resistentes al alcohol y que contienen metoprolol.
CN104010630A (zh) * 2011-12-09 2014-08-27 普渡制药公司 包含聚(ε-己内酯)和聚氧乙烯的药物剂型
NZ627980A (en) * 2012-02-07 2016-12-23 Biogen Ma Inc Pharmaceutical compositions containing dimethyl fumarate
WO2014039987A2 (en) 2012-09-09 2014-03-13 Prothera Biologics, Inc. Treatment of disease using inter-alpha inhibitor proteins
EP3272837B1 (en) * 2016-07-21 2021-01-27 Bharat Petroleum Corporation Limited Fuel composition containing lubricity improver and method thereof
CN111836618A (zh) * 2018-02-08 2020-10-27 景凱生物科技股份有限公司 类阿片受体拮抗剂的固体剂型用的医药剂型

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CA2518734A1 (en) * 2003-03-14 2004-09-30 Nirmal Mulye A process for preparing sustained release tablets

Also Published As

Publication number Publication date
WO2004082615A2 (en) 2004-09-30
US20110071137A1 (en) 2011-03-24
JP2006520390A (ja) 2006-09-07
EP1603540A2 (en) 2005-12-14
AU2004222339A1 (en) 2004-09-30
NZ542303A (en) 2008-12-24
MXPA05009886A (es) 2006-05-04
CA2518734A1 (en) 2004-09-30
WO2004082615A3 (en) 2004-11-25
US20040224017A1 (en) 2004-11-11

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A ANUI DADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2129 DE 25/10/2011.