BRPI0407652A - método para acentuar a eficácia de um agente ativo, composição e método para produzir a composição - Google Patents

método para acentuar a eficácia de um agente ativo, composição e método para produzir a composição

Info

Publication number
BRPI0407652A
BRPI0407652A BRPI0407652-4A BRPI0407652A BRPI0407652A BR PI0407652 A BRPI0407652 A BR PI0407652A BR PI0407652 A BRPI0407652 A BR PI0407652A BR PI0407652 A BRPI0407652 A BR PI0407652A
Authority
BR
Brazil
Prior art keywords
composition
active agent
effectiveness
producing
enhancing
Prior art date
Application number
BRPI0407652-4A
Other languages
English (en)
Inventor
Isabelle Hansenne
Marc Cornell
Hani Fares
Peter Foltis
Original Assignee
Oreal
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Oreal filed Critical Oreal
Publication of BRPI0407652A publication Critical patent/BRPI0407652A/pt

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/67Vitamins
    • A61K8/676Ascorbic acid, i.e. vitamin C
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/34Alcohols
    • A61K8/347Phenols
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/36Carboxylic acids; Salts or anhydrides thereof
    • A61K8/368Carboxylic acids; Salts or anhydrides thereof with carboxyl groups directly bound to carbon atoms of aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/37Esters of carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/4973Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with oxygen as the only hetero atom
    • A61K8/498Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with oxygen as the only hetero atom having 6-membered rings or their condensed derivatives, e.g. coumarin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/63Steroids; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/67Vitamins
    • A61K8/671Vitamin A; Derivatives thereof, e.g. ester of vitamin A acid, ester of retinol, retinol, retinal
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/04Antipruritics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/12Keratolytics, e.g. wart or anti-corn preparations
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical & Material Sciences (AREA)
  • Birds (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Pain & Pain Management (AREA)
  • Obesity (AREA)
  • Nutrition Science (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Virology (AREA)
  • Rheumatology (AREA)
  • Medicinal Preparation (AREA)
  • Cosmetics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

"MéTODO PARA ACENTUAR A EFICáCIA DE UM AGENTE ATIVO, COMPOSIçãO E MéTODO PARA PRODUZIR A COMPOSIçãO". A presente invenção refere-se a composições que contêm pelo menos um derivado de ácido salicílico e pelo menos um agente ativo cosmético, dermatológico, farmacêutico, etc., onde o derivado de ácido salicílico aumenta, acentua, etc., a eficácia do agente ativo, bem com ao métodos de produção e uso de tais composições. A invenção também se refere a um método para acentuar a eficácia de agentes ativos com esses derivados de ácido salicílico.
BRPI0407652-4A 2003-02-19 2004-02-06 método para acentuar a eficácia de um agente ativo, composição e método para produzir a composição BRPI0407652A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/367,700 US8343519B2 (en) 2003-02-19 2003-02-19 Chemical enhancer and method
PCT/EP2004/001169 WO2004073745A1 (en) 2003-02-19 2004-02-06 Salicylic acid derivative as efficacy enhancer and method

Publications (1)

Publication Number Publication Date
BRPI0407652A true BRPI0407652A (pt) 2006-02-21

Family

ID=32850027

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0407652-4A BRPI0407652A (pt) 2003-02-19 2004-02-06 método para acentuar a eficácia de um agente ativo, composição e método para produzir a composição

Country Status (5)

Country Link
US (1) US8343519B2 (pt)
EP (1) EP1594546A1 (pt)
JP (1) JP2007523832A (pt)
BR (1) BRPI0407652A (pt)
WO (1) WO2004073745A1 (pt)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040161392A1 (en) * 2003-02-19 2004-08-19 L'oreal S.A. Skin peeling composition and method
FR2884417B1 (fr) * 2005-04-19 2007-06-15 Oreal Composition cosmetique deodorante comprenant 'association d'un derive lipophile de l'acide salicylique et d'un sel d'aluminium anti-transpirant
WO2007031117A1 (en) * 2005-04-19 2007-03-22 L'oreal Use op a lipophilic salicylic acid derivative as a deodorant active agent, process for treating body odour
FR2884416B1 (fr) * 2005-04-19 2007-06-15 Oreal Utilisation comme actif deodorant d'un derive lipophile de l'acide salicylique dans une composition deodorante ne contenant pas d'agent antitranspirant ; procede de traitement des odeurs corporelles
US20070025939A1 (en) * 2005-07-29 2007-02-01 L'oreal S.A. cosmetic compositions containing hydroquinone and various sunscreen agents
KR20090004980A (ko) * 2006-04-18 2009-01-12 디에스엠 아이피 어셋츠 비.브이. 살리실산 및 아스코브산을 포함하는 화장품 조성물
US20080082058A1 (en) * 2006-10-02 2008-04-03 Wallach Gary S Debriding Callus Foot Tissue
US8562574B2 (en) * 2006-10-02 2013-10-22 Gary S. Wallach Callus-tissue-debridement apparatus
WO2009014061A1 (ja) * 2007-07-20 2009-01-29 Rohto Pharmaceutical Co., Ltd. 乳化組成物
FR2936705B1 (fr) 2008-10-08 2010-12-17 Oreal Procede de rasage utilisant des derives de l'acide salicylique
JP5615515B2 (ja) * 2009-05-26 2014-10-29 持田製薬株式会社 洗浄用組成物
FR2990850B1 (fr) * 2012-05-25 2014-05-16 Oreal Composition cosmetique comprenant l'association d'un derive lipophile de l'acide salicylique, d'un sel ou complexe d'aluminium anti-transpirant et d'un sel d'acide amine n,n-diacide acetique
FR3012960B1 (fr) 2013-11-13 2016-07-15 Oreal Utilisation comme agent deodorant d'un derive salifie d'acide salicylique, seul ou en melange
WO2018115058A1 (en) * 2016-12-22 2018-06-28 L'oreal Preserving agent comprising 4-(3-ethoxy-4-hydroxyphenyl)-2-butanone, and use thereof in cosmetic compositions
CN109966241A (zh) * 2019-04-16 2019-07-05 浙江大学 一种促渗组合物在外用制剂经皮促渗中的应用
CN111559962B (zh) * 2020-07-14 2020-10-30 江西中医药大学 一种具有抗氧化活性的新酚酸类化合物的制备方法及应用

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2581542B1 (fr) 1985-05-07 1988-02-19 Oreal Compositions topiques destinees au traitement de la peau a base de derives de l'acide salicylique
AU618517B2 (en) * 1986-12-23 1992-01-02 Eugene J. Van Scott Additives enhancing topical actions of therapeutic agents
US5389677B1 (en) * 1986-12-23 1997-07-15 Tristrata Inc Method of treating wrinkles using glycalic acid
LU87187A1 (fr) * 1988-03-31 1989-10-26 Oreal Association de derives de pyrimidine et de derives d'acide salicylique pour induire et stimuler la croissance des cheveux et diminuer leur chute
LU87408A1 (fr) 1988-12-16 1990-07-10 Oreal Utilisation de derives salicyles pour le traitement du vieillissement de la peau
FR2653336B1 (fr) * 1989-10-20 1994-04-08 Oreal Composition pharmaceutique et cosmetiques depigmentantes a base d'acide cafeique.
BR9001880A (pt) * 1990-04-18 1991-11-12 Forjas Taurus Sa Mecanismo de desarme do cao aplicavel a pistolas semi-automaticas
ES2121947T3 (es) * 1992-05-15 1998-12-16 Shiseido Co Ltd Preparacion externa para la piel.
US5516793A (en) * 1993-04-26 1996-05-14 Avon Products, Inc. Use of ascorbic acid to reduce irritation of topically applied active ingredients
FR2714599B1 (fr) * 1993-12-30 1996-02-09 Oreal Composition pour lutter contre le vieillissement, agissant siimultanément sur les couches superficielles et profondes de la peau, son utilisation.
FR2714831B1 (fr) * 1994-01-10 1996-02-02 Oreal Composition cosmétique et/ou dermatologique contenant des dérivés d'acide salicylique et procédé de solubilisation de ces dérivés.
FR2718640B1 (fr) 1994-04-18 1996-05-15 Oreal Composition cosmétique et/ou dermatologique notamment pour dépigmenter la peau, ses utilisations.
FR2722102B1 (fr) * 1994-07-11 1996-08-23 Cird Galderma Utilisation de particules creuses deformables dans une composition cosmetique et/ou dermatologique, contenant des matieres grasses
FR2726468B1 (fr) * 1994-11-03 1996-12-13 Oreal Utilisation de derive de l'acide salicylique comme stabilisant d'une emulsion huile-dans-eau
US5687971A (en) 1995-07-07 1997-11-18 Wascana Gaming Inc. Bingo game management method
FR2740040B1 (fr) * 1995-10-23 1997-12-05 Oreal Utilisation d'au moins un agoniste beta-adrenergique en tant qu'antagoniste de substance p
US6159479A (en) * 1997-09-16 2000-12-12 L'oreal Hydrous salicylic acid solutions
FR2768622B1 (fr) 1997-09-22 1999-11-26 Oreal Extrait de rosacees en tant qu'antagoniste de bradykinine
US6200964B1 (en) * 1999-05-28 2001-03-13 Neutrogena Corporation Silicone gel containing salicylic acid
RU2266102C2 (ru) 1999-09-06 2005-12-20 Сетсуко УЕДА Состав для химического пилинга
US6566020B2 (en) * 2001-04-27 2003-05-20 Advanced Micro Devices, Inc. Dark field trench in an alternating phase shift mask to avoid phase conflict

Also Published As

Publication number Publication date
JP2007523832A (ja) 2007-08-23
US20040162272A1 (en) 2004-08-19
US8343519B2 (en) 2013-01-01
EP1594546A1 (en) 2005-11-16
WO2004073745A1 (en) 2004-09-02

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B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
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Free format text: RECONHECIDO O OBSTACULO ADMINISTRATIVO E CONCEDIDO A DEVOLUCAO DE PRAZO DE 47 DIAS , NOS TERMOS DO ARTIGO 221 2O DA LPI E DA RESOLUCAO 116/04.

B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

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B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2343 DE 01-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

B15K Others concerning applications: alteration of classification

Ipc: A61K 8/67 (2006.01), A61K 8/34 (2006.01), A61K 8/3